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中文名称 英文名称 CAS号 化学式 结构式图片
—— [3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 4-propan-2-yloxybenzoate —— C19H17ClN2O4
[3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl 4-propan-2-yloxybenzoate
—— 1-(4-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(2-methylpropylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid —— C26H31FN4O6S
1-(4-fluorophenyl)-4-methyl-5-[4-[[(2R)-2-methylbutanoyl]amino]-2-(2-methylpropylsulfamoyl)phenoxy]pyrazole-3-carboxylic acid
—— 6-amino-5-[(2R)-2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione —— C26H27ClN6O3S
6-amino-5-[(2R)-2-[[5-(4-chlorophenyl)-4-(2-propan-2-ylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione
—— (2R)-N-(4-ethylphenyl)-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H31N5O3S2
(2R)-N-(4-ethylphenyl)-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[[3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-phenyl-1,3,4-oxadiazole —— C17H11ClN4O2S
2-[[3-(2-Chlorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-5-phenyl-1,3,4-oxadiazole
—— (2S)-N-(4-ethylphenyl)-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C29H31N5O3S2
(2S)-N-(4-ethylphenyl)-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C32H33N5O4S
2-[(4S)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide —— C33H34N4O5S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-1-(2,4-dimethylphenyl)-7-oxo-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(3-methoxypropyl)acetamide
—— (2R)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-2-phenyl-1-pyrrolidin-1-ylethanone —— C21H23N5OS
(2R)-2-[1-(2,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-2-phenyl-1-pyrrolidin-1-ylethanone
—— (2R)-2-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide —— C14H17ClN4OS
(2R)-2-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethylpropanamide
—— (2R)-2-[[4-amino-5-(4-tert-butylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylpropanamide —— C17H25N5OS
(2R)-2-[[4-amino-5-(4-tert-butylphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylpropanamide
—— 2-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3,5-trimethylpyrazol-4-yl)acetamide —— C17H19FN6OS
2-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3,5-trimethylpyrazol-4-yl)acetamide
—— 2-(4-fluorophenyl)-5-[(1S)-1-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1,3,4-oxadiazole —— C19H15F2N5OS
2-(4-fluorophenyl)-5-[(1S)-1-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1,3,4-oxadiazole
—— (4R)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one —— C36H40N4O4S
(4R)-4-(2,5-dimethoxyphenyl)-1-(2,4-dimethylphenyl)-8-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3-phenyl-4H-pyrazolo[3,4-e][1,4]thiazepin-7-one
—— (2R)-3-[(2R)-butan-2-yl]-2-(1-phenyl-3-pyridin-4-ylpyrazol-4-yl)-1,2-dihydroquinazolin-4-one —— C26H25N5O
(2R)-3-[(2R)-butan-2-yl]-2-(1-phenyl-3-pyridin-4-ylpyrazol-4-yl)-1,2-dihydroquinazolin-4-one
—— (2R)-N-(2-chloro-4-nitrophenyl)-2-phenyl-2-[(4-phenyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide —— C26H18ClN5O3S2
(2R)-N-(2-chloro-4-nitrophenyl)-2-phenyl-2-[(4-phenyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl]acetamide
—— 2-[(1S)-1-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole —— C20H18ClN5OS
2-[(1S)-1-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole
—— 2-[[4-(3-chloro-4-fluorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]ethanone —— C28H28ClFN4O3S
2-[[4-(3-chloro-4-fluorophenyl)-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-1-[2,5-dimethyl-1-[[(2S)-oxolan-2-yl]methyl]pyrrol-3-yl]ethanone
—— 2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide —— C32H33N5O4S
2-[(4R)-4-(1,3-benzodioxol-5-yl)-3-tert-butyl-1-(4-methylphenyl)-7-oxo-4H-pyrazolo[3,4-e][1,4]thiazepin-8-yl]-N-(pyridin-2-ylmethyl)acetamide
—— [(1R,2R,5S)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C27H31Cl2N3O2S
[(1R,2R,5S)-5-methyl-2-propan-2-ylcyclohexyl] 2-[[4-(3-chloro-4-methylphenyl)-5-(4-chlorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— (2R)-2-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylpropanamide —— C14H17ClN4OS
(2R)-2-[[5-(4-chlorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N,N-dimethylpropanamide
—— [2-[[(1S)-1-(1-benzofuran-2-yl)ethyl]amino]-2-oxoethyl] 3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoate —— C23H21N3O5
[2-[[(1S)-1-(1-benzofuran-2-yl)ethyl]amino]-2-oxoethyl] 3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoate
—— 2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[2-(1H-indol-3-yl)ethyl]acetamide —— C21H22N6OS
2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[2-(1H-indol-3-yl)ethyl]acetamide
—— (2S)-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanyl-N,N-dimethylpropanamide —— C14H19N5OS
(2S)-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanyl-N,N-dimethylpropanamide
—— N-cyclopropyl-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide —— C18H23N5O3S2
N-cyclopropyl-2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[(3R)-1,1-dioxothiolan-3-yl]acetamide
—— [2-[(2-Fluorophenyl)methyl-methylamino]-2-oxoethyl] 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate —— C21H19FN2O3S
[2-[(2-Fluorophenyl)methyl-methylamino]-2-oxoethyl] 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate
—— N-[(1S)-1-phenylethyl]-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C28H29N5O3S2
N-[(1S)-1-phenylethyl]-2-[[4-phenyl-5-(3-pyrrolidin-1-ylsulfonylphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (7,8-dimethyl-2-oxochromen-4-yl)methyl (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C32H26N2O6
(7,8-dimethyl-2-oxochromen-4-yl)methyl (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate —— C21H17N3O3S
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate
—— (2S)-2-[[4-(4-chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide —— C27H24ClN7O2S
(2S)-2-[[4-(4-chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide
—— [(2S)-1-[(5-chloropyridin-2-yl)amino]-1-oxopropan-2-yl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H23ClN4O5
[(2S)-1-[(5-chloropyridin-2-yl)amino]-1-oxopropan-2-yl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-acetyl-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C20H21N3O6
[3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl 4-acetyl-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— [2-oxo-2-[3-(2-oxopyrrolidin-1-yl)propylamino]ethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C29H30N4O6
[2-oxo-2-[3-(2-oxopyrrolidin-1-yl)propylamino]ethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H29N3O7S
[2-[[(3S)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— 2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-prop-2-ynylacetamide —— C14H15N5OS
2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-prop-2-ynylacetamide
—— 2-(4-fluorophenyl)-5-[(1S)-1-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1,3,4-oxadiazole —— C19H15F2N5OS
2-(4-fluorophenyl)-5-[(1S)-1-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-1,3,4-oxadiazole
—— (3S)-3-[(E)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoyl]-6-methylpyran-2,4-dione —— C25H20N2O5
(3S)-3-[(E)-3-[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoyl]-6-methylpyran-2,4-dione
—— (3aS,7aS)-2-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-3a,4,7,7a-tetrahydroisoindole-1,3-dione —— C18H15ClN2O3
(3aS,7aS)-2-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]-3a,4,7,7a-tetrahydroisoindole-1,3-dione
—— (3S)-5-[2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]-3-methyl-1,3-dihydroindol-2-one —— C20H19N5O2S
(3S)-5-[2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]-3-methyl-1,3-dihydroindol-2-one
—— (2R)-2-[[4-(4-chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide —— C27H24ClN7O2S
(2R)-2-[[4-(4-chlorophenyl)-5-pyridin-4-yl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)propanamide
—— 3-Cyclopropyl-5-[(1,3-diphenylpyrazol-4-yl)methylsulfanyl]-4-methyl-1,2,4-triazole —— C22H21N5S
3-Cyclopropyl-5-[(1,3-diphenylpyrazol-4-yl)methylsulfanyl]-4-methyl-1,2,4-triazole
—— N-[2-[(5E)-5-[(2-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-2-[1-(2-methoxy-5-methylphenyl)tetrazol-5-yl]sulfanylacetamide —— C23H21FN6O4S2
N-[2-[(5E)-5-[(2-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]-2-[1-(2-methoxy-5-methylphenyl)tetrazol-5-yl]sulfanylacetamide
—— [2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C30H23N3O7
[2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[[4-(Dimethylamino)phenyl]methylamino]-2-oxoethyl] 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate —— C22H23N3O3S
[2-[[4-(Dimethylamino)phenyl]methylamino]-2-oxoethyl] 2-(4-methylphenyl)-1,3-thiazole-4-carboxylate
—— 2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-cyclopropylethyl]acetamide —— C17H23N5O2S
2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-[(1S)-1-cyclopropylethyl]acetamide
—— 2-[(1R)-1-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole —— C20H18FN5OS
2-[(1R)-1-[[5-(4-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]ethyl]-5-(4-methylphenyl)-1,3,4-oxadiazole
—— 2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylbutan-2-yl)acetamide —— C17H25N5O2S
2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methylbutan-2-yl)acetamide
—— [(2R)-1-[(5-chloropyridin-2-yl)amino]-1-oxopropan-2-yl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H23ClN4O5
[(2R)-1-[(5-chloropyridin-2-yl)amino]-1-oxopropan-2-yl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— [2-[[(3R)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate —— C28H29N3O7S
[2-[[(3R)-1,1-dioxothiolan-3-yl]-ethylamino]-2-oxoethyl] (Z)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]prop-2-enoate
—— (3aS,7aS)-2-[[2-(3-fluorophenyl)-1,3-oxazol-4-yl]methyl]-3a,4,7,7a-tetrahydroisoindole-1,3-dione —— C18H15FN2O3
(3aS,7aS)-2-[[2-(3-fluorophenyl)-1,3-oxazol-4-yl]methyl]-3a,4,7,7a-tetrahydroisoindole-1,3-dione