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—— (5S)-3-(4-chlorophenyl)-N-[3-oxo-3-(propan-2-ylamino)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20ClN3O3
(5S)-3-(4-chlorophenyl)-N-[3-oxo-3-(propan-2-ylamino)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(4-chlorophenyl)-N-[(2S)-1-oxo-1-(propylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20ClN3O3
(5R)-3-(4-chlorophenyl)-N-[(2S)-1-oxo-1-(propylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[4-[Cyclohexyl(methyl)amino]-6-(trifluoromethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylic acid —— C18H20F3N3O3S
5-[[4-[Cyclohexyl(methyl)amino]-6-(trifluoromethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylic acid
—— (5S)-3-(4-chlorophenyl)-N-[3-oxo-3-[[(2S)-oxolan-2-yl]methylamino]propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H22ClN3O4
(5S)-3-(4-chlorophenyl)-N-[3-oxo-3-[[(2S)-oxolan-2-yl]methylamino]propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-chloro-N-[(2R,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2R,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— (5R)-N-[(1S)-3-amino-1-cyclohexyl-3-oxopropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C19H25N3O3
(5R)-N-[(1S)-3-amino-1-cyclohexyl-3-oxopropyl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5-chloro-N-[(2S,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2S,3S)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— (5R)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H23FN4O3
(5R)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-chloro-N-[(2S,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2S,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— (5S)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H27FN4O3
(5S)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-bromo-N-[(1S,3S)-3-butoxy-2,2-dimethylcyclobutyl]-N-methylpyridine-3-carboxamide —— C17H25BrN2O2
5-bromo-N-[(1S,3S)-3-butoxy-2,2-dimethylcyclobutyl]-N-methylpyridine-3-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-[(2R)-1-oxo-1-(propylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20ClN3O3
(5S)-3-(4-chlorophenyl)-N-[(2R)-1-oxo-1-(propylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[4-[Benzyl(methyl)amino]-6-propan-2-ylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C21H22N3O3S-
5-[[4-[Benzyl(methyl)amino]-6-propan-2-ylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— (5S)-3-(4-fluorophenyl)-N-[(2R)-1-(2-methoxyethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20FN3O4
(5S)-3-(4-fluorophenyl)-N-[(2R)-1-(2-methoxyethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(4-chlorophenyl)-N-[(2R)-1-(ethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C15H18ClN3O3
(5R)-3-(4-chlorophenyl)-N-[(2R)-1-(ethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-bromo-N-[[4-(dimethylamino)oxan-4-yl]methyl]-2-methyl-3-sulfamoylbenzamide —— C16H24BrN3O4S
5-bromo-N-[[4-(dimethylamino)oxan-4-yl]methyl]-2-methyl-3-sulfamoylbenzamide
—— (5R)-3-(4-chlorophenyl)-N-[3-(2-methoxyethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20ClN3O4
(5R)-3-(4-chlorophenyl)-N-[3-(2-methoxyethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-fluorophenyl)-N-[(2R)-1-oxo-1-(propylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20FN3O3
(5S)-3-(4-fluorophenyl)-N-[(2R)-1-oxo-1-(propylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-[(2S)-1-(cyclopropylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H18ClN3O3
(5S)-3-(4-chlorophenyl)-N-[(2S)-1-(cyclopropylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-chloro-N-[(2R,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide —— C21H26Cl2N4O
5-chloro-N-[(2R,3R)-3-(4-chlorophenyl)butan-2-yl]-N-methyl-2-piperidin-1-ylpyrimidine-4-carboxamide
—— (5S)-3-(4-fluorophenyl)-N-[(2S)-1-(2-methoxyethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20FN3O4
(5S)-3-(4-fluorophenyl)-N-[(2S)-1-(2-methoxyethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-[3-(2-methoxyethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20ClN3O4
(5S)-3-(4-chlorophenyl)-N-[3-(2-methoxyethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(4-chlorophenyl)-N-[(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H18ClN3O3
(5R)-3-(4-chlorophenyl)-N-[(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-bromo-N-[(1R,3R)-3-butoxy-2,2-dimethylcyclobutyl]-N-methylpyridine-3-carboxamide —— C17H25BrN2O2
5-bromo-N-[(1R,3R)-3-butoxy-2,2-dimethylcyclobutyl]-N-methylpyridine-3-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-[(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H18ClN3O3
(5S)-3-(4-chlorophenyl)-N-[(2R)-1-(cyclopropylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-[(2R)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H23ClN4O3
(5S)-3-(4-chlorophenyl)-N-[(2R)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(4-chlorophenyl)-N-[3-oxo-3-[[(2R)-oxolan-2-yl]methylamino]propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H22ClN3O4
(5R)-3-(4-chlorophenyl)-N-[3-oxo-3-[[(2R)-oxolan-2-yl]methylamino]propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [5-[[4-Methyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-morpholin-4-ylmethanone —— C19H26N4O3S
[5-[[4-Methyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-morpholin-4-ylmethanone
—— (5R)-3-(4-chlorophenyl)-N-[(2R)-1-(4-methylpiperazin-4-ium-1-yl)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H24ClN4O3+
(5R)-3-(4-chlorophenyl)-N-[(2R)-1-(4-methylpiperazin-4-ium-1-yl)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[4-[Cyclohexyl(methyl)amino]-6-propan-2-ylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C20H26N3O3S-
5-[[4-[Cyclohexyl(methyl)amino]-6-propan-2-ylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— (5S)-3-(4-chlorophenyl)-N-[3-(2-methylpropylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H22ClN3O3
(5S)-3-(4-chlorophenyl)-N-[3-(2-methylpropylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H28N4O3
(5S)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-bromo-N-[(2S)-3,3-dimethylbutan-2-yl]-2-methyl-3-sulfamoylbenzamide —— C14H21BrN2O3S
5-bromo-N-[(2S)-3,3-dimethylbutan-2-yl]-2-methyl-3-sulfamoylbenzamide
—— (5S)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H28N4O3
(5S)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[(2R)-1-oxo-3-phenyl-1-(propylamino)propan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C22H25N3O3
(5S)-N-[(2R)-1-oxo-3-phenyl-1-(propylamino)propan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-bromo-N-[(1S,3R)-3-butoxy-2,2-dimethylcyclobutyl]-N-methylpyridine-3-carboxamide —— C17H25BrN2O2
5-bromo-N-[(1S,3R)-3-butoxy-2,2-dimethylcyclobutyl]-N-methylpyridine-3-carboxamide
—— 5-methyl-1-(3-methylphenyl)-N,3-bis(2-methylpropyl)pyrazole-4-carboxamide —— C20H29N3O
5-methyl-1-(3-methylphenyl)-N,3-bis(2-methylpropyl)pyrazole-4-carboxamide
—— (5R)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H28N4O3
(5R)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(4-chlorophenyl)-N-[(2S)-1-(4-fluoroanilino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H17ClFN3O3
(5R)-3-(4-chlorophenyl)-N-[(2S)-1-(4-fluoroanilino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(1,3-benzodioxol-5-yl)-N-[3-(furan-2-ylmethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H19N3O6
(5S)-3-(1,3-benzodioxol-5-yl)-N-[3-(furan-2-ylmethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-(2-morpholin-4-yl-2-oxoethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H18ClN3O4
(5S)-3-(4-chlorophenyl)-N-(2-morpholin-4-yl-2-oxoethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(2-methylphenyl)-N-[(2S)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C24H27N3O3
(5S)-3-(2-methylphenyl)-N-[(2S)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [(5R)-3-(2-chloro-5-methoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]-morpholin-4-ylmethanone —— C15H17ClN2O4
[(5R)-3-(2-chloro-5-methoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]-morpholin-4-ylmethanone
—— (5R)-3-(4-chlorophenyl)-N-[(2S)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H18ClN3O4
(5R)-3-(4-chlorophenyl)-N-[(2S)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(1,3-benzodioxol-5-yl)-N-[3-(furan-2-ylmethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H19N3O6
(5R)-3-(1,3-benzodioxol-5-yl)-N-[3-(furan-2-ylmethylamino)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[(2S)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]-3-(2-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H23N3O3
(5S)-N-[(2S)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]-3-(2-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-[(2S)-1-(2-methoxyethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20ClN3O4
(5S)-3-(4-chlorophenyl)-N-[(2S)-1-(2-methoxyethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(4-chlorophenyl)-N-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H20ClN3O4
(5R)-3-(4-chlorophenyl)-N-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-chlorophenyl)-N-[(2S)-1-oxo-1-(propan-2-ylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H20ClN3O3
(5S)-3-(4-chlorophenyl)-N-[(2S)-1-oxo-1-(propan-2-ylamino)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(4-chlorophenyl)-N-[(2R)-1-(4-fluoroanilino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H17ClFN3O3
(5R)-3-(4-chlorophenyl)-N-[(2R)-1-(4-fluoroanilino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide