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—— [(5aS,8aS)-1-[(3-fluorophenyl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-thiophen-2-ylmethanone —— C20H23FN2OS
[(5aS,8aS)-1-[(3-fluorophenyl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-thiophen-2-ylmethanone
—— [(5aS,8aS)-1-[(4-methoxyphenyl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-pyridin-2-ylmethanone —— C22H27N3O2
[(5aS,8aS)-1-[(4-methoxyphenyl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-pyridin-2-ylmethanone
—— [(5aS,8aS)-1-(naphthalen-1-ylmethyl)-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-pyridin-2-ylmethanone —— C25H27N3O
[(5aS,8aS)-1-(naphthalen-1-ylmethyl)-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-pyridin-2-ylmethanone
—— [(5aS,8aS)-1-[(3-cyclopentyloxyphenyl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-pyridin-2-ylmethanone —— C26H33N3O2
[(5aS,8aS)-1-[(3-cyclopentyloxyphenyl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-7-yl]-pyridin-2-ylmethanone
—— 5-[1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C22H31N5O2
5-[1-[(1R,2R)-2-methylcyclopropanecarbonyl]piperidin-4-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H29N5O3
5-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H29N5O3
5-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(3R)-1-methylsulfonylpiperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C18H27N5O3S
5-[(3R)-1-methylsulfonylpiperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-bromo-N-[5-chloro-2-(dimethylamino)phenyl]thiophene-2-sulfonamide —— C12H12BrClN2O2S2
5-bromo-N-[5-chloro-2-(dimethylamino)phenyl]thiophene-2-sulfonamide
—— 5-[(3S)-1-methylsulfonylpiperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C18H27N5O3S
5-[(3S)-1-methylsulfonylpiperidin-3-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5S,10bS)-9-bromo-2,5-bis(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H21BrN2O3
(5S,10bS)-9-bromo-2,5-bis(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[1-(5-Methylthiophene-3-carbonyl)piperidin-4-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C23H29N5O2S
5-[1-(5-Methylthiophene-3-carbonyl)piperidin-4-yl]-11-propan-2-yl-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— [(5aS,8aS)-7-[(2-methylpyrimidin-5-yl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-1-yl]-(2,6-dimethoxyphenyl)methanone —— C23H30N4O3
[(5aS,8aS)-7-[(2-methylpyrimidin-5-yl)methyl]-2,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-1-yl]-(2,6-dimethoxyphenyl)methanone
—— (5R)-5-(oxan-4-yl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]isoquinoline —— C15H19NO3
(5R)-5-(oxan-4-yl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]isoquinoline
—— (5R,6S)-6-(3-fluorophenyl)-5-(furan-3-ylmethylamino)piperidin-2-one —— C16H17FN2O2
(5R,6S)-6-(3-fluorophenyl)-5-(furan-3-ylmethylamino)piperidin-2-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-6-propan-2-yl-2H-pyrazolo[3,4-b]pyridin-3-amine —— C13H15N5O
5-(3-methyl-1,2-oxazol-5-yl)-6-propan-2-yl-2H-pyrazolo[3,4-b]pyridin-3-amine
—— (5R)-N-(3,4-dimethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H21NO3S
(5R)-N-(3,4-dimethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5aS,8aS)-7-benzyl-1,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-2-one —— C15H20N2O
(5aS,8aS)-7-benzyl-1,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-2-one
—— (5aR,8aS)-7-benzyl-1,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-2-one —— C15H20N2O
(5aR,8aS)-7-benzyl-1,3,4,5,5a,6,8,8a-octahydropyrrolo[3,4-b]azepin-2-one
—— (5R,6S)-6-(2-fluorophenyl)-5-(pyridin-3-ylmethylamino)piperidin-2-one —— C17H18FN3O
(5R,6S)-6-(2-fluorophenyl)-5-(pyridin-3-ylmethylamino)piperidin-2-one
—— (5R)-5-[(2,5-dimethoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C12H13NO3S2
(5R)-5-[(2,5-dimethoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[3-(4-Fluorophenyl)-1-methylpyrazol-4-yl]methyl]-1,2-dihydropyrazol-3-one —— C14H13FN4O
5-[[3-(4-Fluorophenyl)-1-methylpyrazol-4-yl]methyl]-1,2-dihydropyrazol-3-one
—— (5R,10bS)-9-bromo-2-(4-fluorophenyl)-5-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H18BrFN2O2
(5R,10bS)-9-bromo-2-(4-fluorophenyl)-5-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,7S)-N-(1-adamantyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H29F3N4O2
(5S,7S)-N-(1-adamantyl)-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S)-5-[(2,5-dimethoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C12H13NO3S2
(5S)-5-[(2,5-dimethoxyphenyl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-cyclopropyl-2-methyl-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]furan-3-carboxamide —— C14H18N4O2
5-cyclopropyl-2-methyl-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]furan-3-carboxamide
—— (5R,6S)-6-(2-fluorophenyl)-5-(furan-2-ylmethylamino)piperidin-2-one —— C16H17FN2O2
(5R,6S)-6-(2-fluorophenyl)-5-(furan-2-ylmethylamino)piperidin-2-one
—— 5-Methyl-2-(oxan-4-yl)-7-prop-2-ynoxypyrazolo[1,5-a]pyrimidine —— C15H17N3O2
5-Methyl-2-(oxan-4-yl)-7-prop-2-ynoxypyrazolo[1,5-a]pyrimidine
—— 5-(Oxan-4-yl)-7,8-dihydro-[1,3]dioxolo[4,5-g]isoquinoline —— C15H17NO3
5-(Oxan-4-yl)-7,8-dihydro-[1,3]dioxolo[4,5-g]isoquinoline
—— 5-cyclopropyl-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-2-methylpyrazole-3-carboxamide —— C14H20N6O
5-cyclopropyl-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-2-methylpyrazole-3-carboxamide
—— 5-cyclopropyl-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide —— C13H17N5O2
5-cyclopropyl-N-[2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
—— (5R,6S)-6-(3-fluorophenyl)-5-(pyridin-4-ylmethylamino)piperidin-2-one —— C17H18FN3O
(5R,6S)-6-(3-fluorophenyl)-5-(pyridin-4-ylmethylamino)piperidin-2-one
—— 5-[2-Methoxy-4-(5-methylfuran-2-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole —— C14H13N3O3
5-[2-Methoxy-4-(5-methylfuran-2-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole
—— 5-Methyl-2-(oxan-4-yl)-7-propoxypyrazolo[1,5-a]pyrimidine —— C15H21N3O2
5-Methyl-2-(oxan-4-yl)-7-propoxypyrazolo[1,5-a]pyrimidine
—— (5R,6S)-6-(3-fluorophenyl)-5-(pyridin-2-ylmethylamino)piperidin-2-one —— C17H18FN3O
(5R,6S)-6-(3-fluorophenyl)-5-(pyridin-2-ylmethylamino)piperidin-2-one
—— (5S)-N-(3,4-dimethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H21NO3S
(5S)-N-(3,4-dimethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-methyl-3-propan-2-yl-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]-1,2-oxazole-4-carboxamide —— C13H19N5O2
5-methyl-3-propan-2-yl-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]-1,2-oxazole-4-carboxamide
—— (5S)-5-(oxan-4-yl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]isoquinoline —— C15H19NO3
(5S)-5-(oxan-4-yl)-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]isoquinoline
—— 5-bromo-2-methoxy-N-[3-(N-methylanilino)propyl]benzenesulfonamide —— C17H21BrN2O3S
5-bromo-2-methoxy-N-[3-(N-methylanilino)propyl]benzenesulfonamide
—— 5-(Pyrrolidin-1-ylmethyl)-3-(2-pyrrolidin-1-ylpyridin-3-yl)-1,2,4-oxadiazole —— C16H21N5O
5-(Pyrrolidin-1-ylmethyl)-3-(2-pyrrolidin-1-ylpyridin-3-yl)-1,2,4-oxadiazole
—— (5R,6S)-6-(3-fluorophenyl)-5-(pyridin-3-ylmethylamino)piperidin-2-one —— C17H18FN3O
(5R,6S)-6-(3-fluorophenyl)-5-(pyridin-3-ylmethylamino)piperidin-2-one
—— (5R,6S)-6-(2-fluorophenyl)-5-(pyridin-2-ylmethylamino)piperidin-2-one —— C17H18FN3O
(5R,6S)-6-(2-fluorophenyl)-5-(pyridin-2-ylmethylamino)piperidin-2-one
—— (5R,6S)-5-amino-6-[(1S)-cyclohex-3-en-1-yl]piperidin-2-one —— C11H18N2O
(5R,6S)-5-amino-6-[(1S)-cyclohex-3-en-1-yl]piperidin-2-one
—— (5-Cyclopropyl-2-methylfuran-3-yl)-[4-(2-methylprop-2-enyl)piperazin-1-yl]methanone —— C17H24N2O2
(5-Cyclopropyl-2-methylfuran-3-yl)-[4-(2-methylprop-2-enyl)piperazin-1-yl]methanone
—— 5-[4-(Furan-2-yl)-2-methylpyrimidin-5-yl]-3,4-dimethyl-1,2-oxazole —— C14H13N3O2
5-[4-(Furan-2-yl)-2-methylpyrimidin-5-yl]-3,4-dimethyl-1,2-oxazole
—— (5R,6S)-5-amino-6-[(1R)-cyclohex-3-en-1-yl]piperidin-2-one —— C11H18N2O
(5R,6S)-5-amino-6-[(1R)-cyclohex-3-en-1-yl]piperidin-2-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-[(2S)-oxolan-2-yl]-N-prop-2-enylpyrimidin-2-amine —— C15H18N4O2
5-(3-methyl-1,2-oxazol-5-yl)-4-[(2S)-oxolan-2-yl]-N-prop-2-enylpyrimidin-2-amine
—— (5-cyclopropyl-1,2-oxazol-3-yl)-(2-methyl-6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl)methanone —— C13H15N5O2
(5-cyclopropyl-1,2-oxazol-3-yl)-(2-methyl-6,8-dihydro-5H-[1,2,4]triazolo[1,5-a]pyrazin-7-yl)methanone
—— 5-(1,3-Benzodioxol-5-yl)-2-methyl-4-pyridin-3-ylpyrimidine —— C17H13N3O2
5-(1,3-Benzodioxol-5-yl)-2-methyl-4-pyridin-3-ylpyrimidine
—— 5-methyl-3-[[(2R)-pyrrolidin-2-yl]methyl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C10H14N6O
5-methyl-3-[[(2R)-pyrrolidin-2-yl]methyl]-2H-triazolo[4,5-d]pyrimidin-7-one