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—— 5-methyl-N-[[(2S)-1-[6-(methylamino)pyrimidin-4-yl]pyrrolidin-2-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C16H21N9
5-methyl-N-[[(2S)-1-[6-(methylamino)pyrimidin-4-yl]pyrrolidin-2-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-{[1-(Furan-2-YL)-N-(2-methoxyethyl)formamido]methyl}-2-methoxyphenyl ethane-1-sulfonate —— C18H23NO7S
5-{[1-(Furan-2-YL)-N-(2-methoxyethyl)formamido]methyl}-2-methoxyphenyl ethane-1-sulfonate
—— 5-methyl-N-[[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C13H16N8
5-methyl-N-[[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— [5-[[[(2S)-butan-2-yl]-(2-methylpropanoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C18H29NO5S
[5-[[[(2S)-butan-2-yl]-(2-methylpropanoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— 5,6-dimethyl-3-[[(6R)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridazine-4-carbonitrile —— C14H17N7
5,6-dimethyl-3-[[(6R)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridazine-4-carbonitrile
—— 5-[[(1S)-1-(3-chlorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide —— C22H25ClN3O2+
5-[[(1S)-1-(3-chlorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide
—— [5-[[[(2S)-butan-2-yl]-(tert-butylcarbamoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C20H34N2O5S
[5-[[[(2S)-butan-2-yl]-(tert-butylcarbamoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— 5,6-dimethyl-N-[[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]thieno[2,3-d]pyrimidin-4-amine —— C15H18N6S
5,6-dimethyl-N-[[(6S)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methyl]thieno[2,3-d]pyrimidin-4-amine
—— 5-[[(1R)-1-(3-chlorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide —— C22H25ClN3O2+
5-[[(1R)-1-(3-chlorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide
—— 5-({[4-(Diethylamino)-6-(methoxymethyl)pyrimidin-2-YL]sulfanyl}methyl)-N-(2-methylpropyl)furan-2-carboxamide —— C20H30N4O3S
5-({[4-(Diethylamino)-6-(methoxymethyl)pyrimidin-2-YL]sulfanyl}methyl)-N-(2-methylpropyl)furan-2-carboxamide
—— (5R)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C24H30N4O3
(5R)-N-[(2S)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[(1R)-1-(3-chlorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide —— C22H24ClN3O2
5-[[(1R)-1-(3-chlorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide
—— [5-[[[(2S)-butan-2-yl]-(ethylcarbamoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C18H30N2O5S
[5-[[[(2S)-butan-2-yl]-(ethylcarbamoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— 5-methoxy-1,3-dimethyl-4-[(2R)-pyrrolidin-2-yl]pyrazole —— C10H17N3O
5-methoxy-1,3-dimethyl-4-[(2R)-pyrrolidin-2-yl]pyrazole
—— 5-[[(1S)-1-(4-nitrophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid —— C19H17N3O5
5-[[(1S)-1-(4-nitrophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid
—— 5-[[(1S)-1-(4-nitrophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate —— C19H17N3O5
5-[[(1S)-1-(4-nitrophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate
—— [5-(methoxymethyl)-2-methylfuran-3-yl]-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C18H25N3O4
[5-(methoxymethyl)-2-methylfuran-3-yl]-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— [5-(methoxymethyl)-2-methylfuran-3-yl]-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C16H21N3O4
[5-(methoxymethyl)-2-methylfuran-3-yl]-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— [5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-pyrrolidin-1-ylmethanone —— C17H21N3O
[5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-pyrrolidin-1-ylmethanone
—— 5-[[4-(methoxymethyl)-6-morpholin-4-ylpyrimidin-2-yl]sulfanylmethyl]-N-(2-methylpropyl)furan-2-carboxamide —— C20H28N4O4S
5-[[4-(methoxymethyl)-6-morpholin-4-ylpyrimidin-2-yl]sulfanylmethyl]-N-(2-methylpropyl)furan-2-carboxamide
—— (5S)-3-(2-chloro-5-methoxyphenyl)-N-[3-oxo-3-(propylamino)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H22ClN3O4
(5S)-3-(2-chloro-5-methoxyphenyl)-N-[3-oxo-3-(propylamino)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[(1R)-1-(4-nitrophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid —— C19H17N3O5
5-[[(1R)-1-(4-nitrophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid
—— 5-[[(1R)-1-(4-nitrophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate —— C19H17N3O5
5-[[(1R)-1-(4-nitrophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate
—— 5-[[4-(4-Ethylpiperazin-4-ium-1-yl)-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C18H24N4O4S
5-[[4-(4-Ethylpiperazin-4-ium-1-yl)-6-(methoxymethyl)pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— 5-[[4-(methoxymethyl)-6-morpholin-4-ylpyrimidin-2-yl]sulfanylmethyl]-N-propan-2-ylfuran-2-carboxamide —— C19H26N4O4S
5-[[4-(methoxymethyl)-6-morpholin-4-ylpyrimidin-2-yl]sulfanylmethyl]-N-propan-2-ylfuran-2-carboxamide
—— 5-methoxy-1,3-dimethyl-4-[(2S)-pyrrolidin-2-yl]pyrazole —— C10H17N3O
5-methoxy-1,3-dimethyl-4-[(2S)-pyrrolidin-2-yl]pyrazole
—— 5-ethyl-1-(4-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-4-carboxamide —— C18H23N3O2
5-ethyl-1-(4-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-4-carboxamide
—— [5-(methoxymethyl)-2-methylfuran-3-yl]-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C17H22N2O3S
[5-(methoxymethyl)-2-methylfuran-3-yl]-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— [5-Propyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-pyrrolidin-1-ylmethanone —— C13H18F3N3O
[5-Propyl-1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-pyrrolidin-1-ylmethanone
—— [5-Ethyl-1-(4-fluorophenyl)pyrazol-4-yl]-morpholin-4-ylmethanone —— C16H18FN3O2
[5-Ethyl-1-(4-fluorophenyl)pyrazol-4-yl]-morpholin-4-ylmethanone
—— (5R)-3-(2-chloro-5-methoxyphenyl)-N-[(2S)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H20ClN3O5
(5R)-3-(2-chloro-5-methoxyphenyl)-N-[(2S)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-ethyl-1-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-4-carboxamide —— C18H23N3O2
5-ethyl-1-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-4-carboxamide
—— (5R)-3-(4-methylphenyl)-N-[(2S)-1-oxo-1-[[(2S)-oxolan-2-yl]methylamino]propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H25N3O4
(5R)-3-(4-methylphenyl)-N-[(2S)-1-oxo-1-[[(2S)-oxolan-2-yl]methylamino]propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-morpholin-4-ylmethanone —— C17H21N3O2
[5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-morpholin-4-ylmethanone
—— [5-(methoxymethyl)-2-methylfuran-3-yl]-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C18H25N3O4
[5-(methoxymethyl)-2-methylfuran-3-yl]-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— [5-Ethyl-1-(3-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C18H25N4O+
[5-Ethyl-1-(3-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5R)-3-(4-methylphenyl)-N-[(2R)-1-oxo-1-[[(2S)-oxolan-2-yl]methylamino]propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H25N3O4
(5R)-3-(4-methylphenyl)-N-[(2R)-1-oxo-1-[[(2S)-oxolan-2-yl]methylamino]propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-(2-chloro-5-methoxyphenyl)-N-[(2R)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H20ClN3O5
(5R)-3-(2-chloro-5-methoxyphenyl)-N-[(2R)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H26N4O3
(5R)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5-Ethyl-1-phenylpyrazol-4-yl)-(4-methylpiperazin-4-ium-1-yl)methanone —— C17H23N4O+
(5-Ethyl-1-phenylpyrazol-4-yl)-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5S)-3-(2-chloro-5-methoxyphenyl)-N-[(2S)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H20ClN3O5
(5S)-3-(2-chloro-5-methoxyphenyl)-N-[(2S)-1-(furan-2-ylmethylamino)-1-oxopropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-ethyl-1-(3-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-4-carboxamide —— C18H23N3O2
5-ethyl-1-(3-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-4-carboxamide
—— [5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-piperidin-1-ylmethanone —— C18H23N3O
[5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-piperidin-1-ylmethanone
—— [5-Ethyl-1-(4-methylphenyl)pyrazol-4-yl]-piperidin-1-ylmethanone —— C18H23N3O
[5-Ethyl-1-(4-methylphenyl)pyrazol-4-yl]-piperidin-1-ylmethanone
—— (5R)-3-(2-chloro-5-methoxyphenyl)-N-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H25ClN4O4
(5R)-3-(2-chloro-5-methoxyphenyl)-N-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H26N4O3
(5S)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [5-Ethyl-1-(3-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone —— C18H24N4O
[5-Ethyl-1-(3-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone
—— [5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone —— C18H24N4O
[5-Ethyl-1-(2-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone
—— (5-Ethyl-1-phenylpyrazol-4-yl)-(4-methylpiperazin-1-yl)methanone —— C17H22N4O
(5-Ethyl-1-phenylpyrazol-4-yl)-(4-methylpiperazin-1-yl)methanone
—— 5-[[4-(methoxymethyl)-6-[(2S)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C18H22N3O4S-
5-[[4-(methoxymethyl)-6-[(2S)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate