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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-Ethyl-1-(3-fluorophenyl)-3-(2-methylpropyl)pyrazole-4-carboxylic acid —— C16H19FN2O2
5-Ethyl-1-(3-fluorophenyl)-3-(2-methylpropyl)pyrazole-4-carboxylic acid
—— (5-fluoro-2-methylphenyl)-[4-[(2S)-1-methoxypropan-2-yl]piperazin-1-yl]methanone —— C16H23FN2O2
(5-fluoro-2-methylphenyl)-[4-[(2S)-1-methoxypropan-2-yl]piperazin-1-yl]methanone
—— 5-ethyl-3-[(3R)-1-(4-methylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C14H19N5O
5-ethyl-3-[(3R)-1-(4-methylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(2R)-1-(4-methylpyrimidin-2-yl)pyrrolidin-2-yl]-1,2,4-oxadiazole —— C13H17N5O
5-ethyl-3-[(2R)-1-(4-methylpyrimidin-2-yl)pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-(4-fluorophenyl)-N-[(1R,2S)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide —— C19H22FN3O2
5-(4-fluorophenyl)-N-[(1R,2S)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide
—— 5-ethyl-3-[(3S)-1-(4-methylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C14H19N5O
5-ethyl-3-[(3S)-1-(4-methylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— (5-chloropyridin-2-yl)-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C16H19ClN4O2
(5-chloropyridin-2-yl)-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— (5R,6R)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C21H20N6O2
(5R,6R)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— (5S,6S)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C21H20N6O2
(5S,6S)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— (5S,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C25H25N5O3
(5S,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5R,6S)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C21H20N6O2
(5R,6S)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— 5-(4-fluorophenyl)-N-[(1R,2R)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide —— C19H22FN3O2
5-(4-fluorophenyl)-N-[(1R,2R)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide
—— 5-bromo-N-[(1R)-1-(1-methylbenzimidazol-2-yl)ethyl]furan-2-carboxamide —— C15H14BrN3O2
5-bromo-N-[(1R)-1-(1-methylbenzimidazol-2-yl)ethyl]furan-2-carboxamide
—— 5-bromo-N-[(1S)-1-(1-methylbenzimidazol-2-yl)ethyl]furan-2-carboxamide —— C15H14BrN3O2
5-bromo-N-[(1S)-1-(1-methylbenzimidazol-2-yl)ethyl]furan-2-carboxamide
—— 5-Ethyl-1-(3-fluorophenyl)-3-(2-methylpropyl)pyrazole-4-carboxylate —— C16H18FN2O2-
5-Ethyl-1-(3-fluorophenyl)-3-(2-methylpropyl)pyrazole-4-carboxylate
—— 5-(4-fluorophenyl)-N-[(1S,2R)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide —— C19H22FN3O2
5-(4-fluorophenyl)-N-[(1S,2R)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide
—— 5-[(4-Fluorophenyl)methyl]-2,4-dimethyl-6-(4-propan-2-ylsulfonylpiperazin-1-yl)pyrimidine —— C20H27FN4O2S
5-[(4-Fluorophenyl)methyl]-2,4-dimethyl-6-(4-propan-2-ylsulfonylpiperazin-1-yl)pyrimidine
—— (5R,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C24H24N6O3
(5R,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-ethyl-4-methyl-N'-[2-[(2S)-2-methylmorpholin-4-yl]acetyl]thiophene-2-carbohydrazide —— C15H23N3O3S
5-ethyl-4-methyl-N'-[2-[(2S)-2-methylmorpholin-4-yl]acetyl]thiophene-2-carbohydrazide
—— 5-[1-(3,4-dimethylphenyl)sulfonylcyclopentyl]-3-[(1S)-1-ethoxyethyl]-1,2,4-oxadiazole —— C19H26N2O4S
5-[1-(3,4-dimethylphenyl)sulfonylcyclopentyl]-3-[(1S)-1-ethoxyethyl]-1,2,4-oxadiazole
—— 5-(4-fluorophenyl)-N-[(1S,2S)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide —— C19H22FN3O2
5-(4-fluorophenyl)-N-[(1S,2S)-2-imidazol-1-ylcyclopentyl]-5-oxopentanamide
—— [5-[[Cyclobutanecarbonyl(cyclopropyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C18H25NO5S
[5-[[Cyclobutanecarbonyl(cyclopropyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— 5-{[(4-Fluorobenzyl)(isobutyryl)amino]methyl}-2-methoxyphenyl 1-ethanesulfonate —— C21H26FNO5S
5-{[(4-Fluorobenzyl)(isobutyryl)amino]methyl}-2-methoxyphenyl 1-ethanesulfonate
—— 5-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate —— C21H20N2O5
5-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate
—— 5-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid —— C21H20N2O5
5-[[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid
—— [5-[[tert-butylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C20H32N2O6S
[5-[[tert-butylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— [5-[[tert-butylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C20H32N2O6S
[5-[[tert-butylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— 5-[1-(3,4-dimethylphenyl)sulfonylcyclopentyl]-3-[(1R)-1-ethoxyethyl]-1,2,4-oxadiazole —— C19H26N2O4S
5-[1-(3,4-dimethylphenyl)sulfonylcyclopentyl]-3-[(1R)-1-ethoxyethyl]-1,2,4-oxadiazole
—— 5-[(1R)-1-[(5-phenyl-1H-imidazol-2-yl)sulfonyl]ethyl]-3-propyl-1,2,4-oxadiazole —— C16H18N4O3S
5-[(1R)-1-[(5-phenyl-1H-imidazol-2-yl)sulfonyl]ethyl]-3-propyl-1,2,4-oxadiazole
—— 5-methyl-1-phenyl-N-propan-2-ylpyrazole-4-carboxamide —— C14H17N3O
5-methyl-1-phenyl-N-propan-2-ylpyrazole-4-carboxamide
—— 5-[[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate —— C21H20N2O5
5-[[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]furan-2-carboxylate
—— 5-[[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid —— C21H20N2O5
5-[[(1S)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]furan-2-carboxylic acid
—— 5-methyl-N-(2-methylpropyl)-1-(4-nitrophenyl)pyrazole-4-carboxamide —— C15H18N4O3
5-methyl-N-(2-methylpropyl)-1-(4-nitrophenyl)pyrazole-4-carboxamide
—— (5-chloropyridin-2-yl)-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C16H19ClN4O2
(5-chloropyridin-2-yl)-[(3S)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— (5R,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C25H25N5O3
(5R,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C24H24N6O3
(5S,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C24H24N6O3
(5S,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S,6R)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one —— C21H20N6O2
(5S,6R)-5-(3-isoquinolin-1-yl-1,2,4-oxadiazol-5-yl)-1-methyl-6-(1-methylpyrazol-4-yl)piperidin-2-one
—— 5-{[Cyclopropyl(2-fluorobenzoyl)amino]methyl}-2-methoxyphenyl 1-ethanesulfonate —— C20H22FNO5S
5-{[Cyclopropyl(2-fluorobenzoyl)amino]methyl}-2-methoxyphenyl 1-ethanesulfonate
—— (5R,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C25H25N5O3
(5R,6S)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-Ethyl-1-(4-methoxyphenyl)-3-(2-methylpropyl)pyrazole-4-carboxylic acid —— C17H22N2O3
5-Ethyl-1-(4-methoxyphenyl)-3-(2-methylpropyl)pyrazole-4-carboxylic acid
—— (5S,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C25H25N5O3
(5S,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(phenoxymethyl)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5R,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C24H24N6O3
(5R,6R)-1-methyl-6-(1-methylpyrazol-4-yl)-5-[3-[4-(pyridin-3-ylmethoxy)phenyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-[(N-Cyclopropyl-3-methylbutanamido)methyl]-2-methoxyphenyl ethane-1-sulfonate —— C18H27NO5S
5-[(N-Cyclopropyl-3-methylbutanamido)methyl]-2-methoxyphenyl ethane-1-sulfonate
—— [5-Methyl-1-(4-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone —— C17H22N4O
[5-Methyl-1-(4-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone
—— (5S,7S)-5-(4-ethylphenyl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H23F3N4O2
(5S,7S)-5-(4-ethylphenyl)-N-(2-methoxyethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-(3-Methoxycarbonylphenyl)furan-2-carboxylate —— C13H9O5-
5-(3-Methoxycarbonylphenyl)furan-2-carboxylate
—— 5-[(N-Cyclopropyl-3,3-dimethylbutanamido)methyl]-2-methoxyphenyl ethane-1-sulfonate —— C19H29NO5S
5-[(N-Cyclopropyl-3,3-dimethylbutanamido)methyl]-2-methoxyphenyl ethane-1-sulfonate
—— 5-[[(2R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)-3,3-dimethylbutan-2-yl]carbamoylamino]-2-fluoro-N-methylbenzamide —— C24H31FN4O2
5-[[(2R)-1-(3,4-dihydro-1H-isoquinolin-2-yl)-3,3-dimethylbutan-2-yl]carbamoylamino]-2-fluoro-N-methylbenzamide
—— 5,6-dichloro-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methylpropyl]pyridine-3-carboxamide —— C18H18Cl2N2O3
5,6-dichloro-N-[(1R)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methylpropyl]pyridine-3-carboxamide