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中文名称 英文名称 CAS号 化学式 结构式图片
—— [5-Methyl-1-(4-methylphenyl)pyrazol-4-yl]-morpholin-4-ylmethanone —— C16H19N3O2
[5-Methyl-1-(4-methylphenyl)pyrazol-4-yl]-morpholin-4-ylmethanone
—— (5R)-3-(3-fluorophenyl)-N-[(2S)-1-(2-methylpropylamino)-1-oxo-3-phenylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H26FN3O3
(5R)-3-(3-fluorophenyl)-N-[(2S)-1-(2-methylpropylamino)-1-oxo-3-phenylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-5-tert-butyl-N-[3-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H26N4O2S
(5S)-5-tert-butyl-N-[3-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— [(5S)-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C15H19FN3O2+
[(5S)-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5S)-3-(3-fluorophenyl)-N-[(2R)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C20H20FN3O3
(5S)-3-(3-fluorophenyl)-N-[(2R)-1-(methylamino)-1-oxo-3-phenylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(3-fluorophenyl)-N-[(2S)-1-(2-methylpropylamino)-1-oxo-3-phenylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H26FN3O3
(5S)-3-(3-fluorophenyl)-N-[(2S)-1-(2-methylpropylamino)-1-oxo-3-phenylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H27FN4O3
(5R)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-N-[2-(6-fluoro-1H-benzimidazol-2-yl)ethyl]-5-methyl-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide —— C20H19FN6O2
(5R)-N-[2-(6-fluoro-1H-benzimidazol-2-yl)ethyl]-5-methyl-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide
—— (5S)-3-(3-fluorophenyl)-N-[(2S)-1-oxo-1-[[(2R)-oxolan-2-yl]methylamino]propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H22FN3O4
(5S)-3-(3-fluorophenyl)-N-[(2S)-1-oxo-1-[[(2R)-oxolan-2-yl]methylamino]propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [(5S)-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-1-yl)methanone —— C15H18FN3O2
[(5S)-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-1-yl)methanone
—— [(5R)-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C15H19FN3O2+
[(5R)-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5R)-N-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H18FN3O2
(5R)-N-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(3-fluorophenyl)-N-[(2R)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C23H24FN3O3
(5S)-3-(3-fluorophenyl)-N-[(2R)-1-oxo-3-phenyl-1-pyrrolidin-1-ylpropan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[4-(Diethylamino)-6-phenylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C20H20N3O3S-
5-[[4-(Diethylamino)-6-phenylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— (5E)-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-2-(4-phenylpiperazin-1-yl)-1,3-thiazol-4-one —— C23H25N3O3S
(5E)-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-2-(4-phenylpiperazin-1-yl)-1,3-thiazol-4-one
—— 5-[(4-Phenyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-carboxylate —— C20H18N3O3S-
5-[(4-Phenyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-carboxylate
—— 5-[(4-Phenyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-carboxylic acid —— C20H19N3O3S
5-[(4-Phenyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-carboxylic acid
—— 5-[(4-tert-butyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]-N-[2-(dimethylamino)ethyl]furan-2-carboxamide —— C22H33N5O2S
5-[(4-tert-butyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]-N-[2-(dimethylamino)ethyl]furan-2-carboxamide
—— 5-[[4-ethyl-6-[(2S)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C18H22N3O3S-
5-[[4-ethyl-6-[(2S)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— 5-({[4-Tert-butyl-6-(morpholin-4-YL)pyrimidin-2-YL]sulfanyl}methyl)-N-(propan-2-YL)furan-2-carboxamide —— C21H30N4O3S
5-({[4-Tert-butyl-6-(morpholin-4-YL)pyrimidin-2-YL]sulfanyl}methyl)-N-(propan-2-YL)furan-2-carboxamide
—— (5R)-5-tert-butyl-N-[3-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H26N4O2S
(5R)-5-tert-butyl-N-[3-(5-oxo-1,4-dihydro-1,2,4-triazol-3-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[[4-ethyl-6-[(2S)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylic acid —— C18H23N3O3S
5-[[4-ethyl-6-[(2S)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylic acid
—— [5-[(4-Tert-butyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-yl]-pyrrolidin-1-ylmethanone —— C22H30N4O2S
[5-[(4-Tert-butyl-6-pyrrolidin-1-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-yl]-pyrrolidin-1-ylmethanone
—— 5-[[4-ethyl-6-[(2R)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C18H22N3O3S-
5-[[4-ethyl-6-[(2R)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— 5-[[4-ethyl-6-[(2R)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylic acid —— C18H23N3O3S
5-[[4-ethyl-6-[(2R)-2-methylpiperidin-1-yl]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylic acid
—— 5-chloro-2-propan-2-yl-N-[(1S)-1-(1H-1,2,4-triazol-5-yl)ethyl]pyrimidine-4-carboxamide —— C12H15ClN6O
5-chloro-2-propan-2-yl-N-[(1S)-1-(1H-1,2,4-triazol-5-yl)ethyl]pyrimidine-4-carboxamide
—— (5-bromo-2-fluoro-3-morpholin-4-ylsulfonylphenyl)-[(2R)-2-methylpiperidin-1-yl]methanone —— C17H22BrFN2O4S
(5-bromo-2-fluoro-3-morpholin-4-ylsulfonylphenyl)-[(2R)-2-methylpiperidin-1-yl]methanone
—— (5S)-N-[2-(6-fluoro-1H-benzimidazol-2-yl)ethyl]-5-methyl-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide —— C20H19FN6O2
(5S)-N-[2-(6-fluoro-1H-benzimidazol-2-yl)ethyl]-5-methyl-6-oxo-1-phenyl-2,5-dihydro-1,2,4-triazine-3-carboxamide
—— [5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-[(2R)-2-(1-propan-2-ylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone —— C26H29N5O
[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-[(2R)-2-(1-propan-2-ylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone
—— 5-chloro-N-[(4R)-4-(1,3-dioxolan-2-yl)-4-methylheptyl]-6-propan-2-yloxypyridine-3-carboxamide —— C20H31ClN2O4
5-chloro-N-[(4R)-4-(1,3-dioxolan-2-yl)-4-methylheptyl]-6-propan-2-yloxypyridine-3-carboxamide
—— [5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-[(2S)-2-(1-propan-2-ylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone —— C26H29N5O
[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]-[(2S)-2-(1-propan-2-ylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone
—— 5-chloro-N-[(4S)-4-(1,3-dioxolan-2-yl)-4-methylheptyl]-6-propan-2-yloxypyridine-3-carboxamide —— C20H31ClN2O4
5-chloro-N-[(4S)-4-(1,3-dioxolan-2-yl)-4-methylheptyl]-6-propan-2-yloxypyridine-3-carboxamide
—— 5-tert-butyl-N-[(2S)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-1,3-oxazole-2-carboxamide —— C16H26N2O4
5-tert-butyl-N-[(2S)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-1,3-oxazole-2-carboxamide
—— [5-[[4-Ethyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-(4-methylpiperazin-1-yl)methanone —— C21H31N5O2S
[5-[[4-Ethyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-(4-methylpiperazin-1-yl)methanone
—— 5-tert-butyl-N-[(2R)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-1,3-oxazole-2-carboxamide —— C16H26N2O4
5-tert-butyl-N-[(2R)-2-methyl-3-(2-methyl-1,3-dioxolan-2-yl)propyl]-1,3-oxazole-2-carboxamide
—— 5-[[4-Ethyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C16H20N3O3S-
5-[[4-Ethyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— 5-[[4-ethyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]-N-(furan-2-ylmethyl)furan-2-carboxamide —— C21H26N4O3S
5-[[4-ethyl-6-[methyl(propyl)amino]pyrimidin-2-yl]sulfanylmethyl]-N-(furan-2-ylmethyl)furan-2-carboxamide
—— 5-[[4-(diethylamino)-6-methylpyrimidin-2-yl]sulfanylmethyl]-N-(furan-2-ylmethyl)furan-2-carboxamide —— C20H24N4O3S
5-[[4-(diethylamino)-6-methylpyrimidin-2-yl]sulfanylmethyl]-N-(furan-2-ylmethyl)furan-2-carboxamide
—— [5-Ethyl-3-methyl-1-(2-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C19H27N4O+
[5-Ethyl-3-methyl-1-(2-methylphenyl)pyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5R)-N-(3-chloro-2-morpholin-4-ylphenyl)-5-(trifluoromethyl)-1,4-diazepane-1-carboxamide —— C17H22ClF3N4O2
(5R)-N-(3-chloro-2-morpholin-4-ylphenyl)-5-(trifluoromethyl)-1,4-diazepane-1-carboxamide
—— 5-[(1R)-1-(5-fluoro-2-nitrophenoxy)ethyl]-3-(2-methylphenyl)-1,2,4-oxadiazole —— C17H14FN3O4
5-[(1R)-1-(5-fluoro-2-nitrophenoxy)ethyl]-3-(2-methylphenyl)-1,2,4-oxadiazole
—— 5-[[4-tert-butyl-6-(4-ethylpiperazin-4-ium-1-yl)pyrimidin-2-yl]sulfanylmethyl]-N-ethylfuran-2-carboxamide —— C22H34N5O2S+
5-[[4-tert-butyl-6-(4-ethylpiperazin-4-ium-1-yl)pyrimidin-2-yl]sulfanylmethyl]-N-ethylfuran-2-carboxamide
—— 5-[[4-ethyl-6-(4-ethylpiperazin-4-ium-1-yl)pyrimidin-2-yl]sulfanylmethyl]-N-propan-2-ylfuran-2-carboxamide —— C21H32N5O2S+
5-[[4-ethyl-6-(4-ethylpiperazin-4-ium-1-yl)pyrimidin-2-yl]sulfanylmethyl]-N-propan-2-ylfuran-2-carboxamide
—— 5-[[4-tert-butyl-6-(4-ethylpiperazin-1-yl)pyrimidin-2-yl]sulfanylmethyl]-N-ethylfuran-2-carboxamide —— C22H33N5O2S
5-[[4-tert-butyl-6-(4-ethylpiperazin-1-yl)pyrimidin-2-yl]sulfanylmethyl]-N-ethylfuran-2-carboxamide
—— [5-[[4-Ethyl-6-(4-ethylpiperazin-4-ium-1-yl)pyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-pyrrolidin-1-ylmethanone —— C22H32N5O2S+
[5-[[4-Ethyl-6-(4-ethylpiperazin-4-ium-1-yl)pyrimidin-2-yl]sulfanylmethyl]furan-2-yl]-pyrrolidin-1-ylmethanone
—— (5S)-N-(3-chloro-2-morpholin-4-ylphenyl)-5-(trifluoromethyl)-1,4-diazepane-1-carboxamide —— C17H22ClF3N4O2
(5S)-N-(3-chloro-2-morpholin-4-ylphenyl)-5-(trifluoromethyl)-1,4-diazepane-1-carboxamide
—— 5-[[4-tert-butyl-6-[cyclohexyl(methyl)amino]pyrimidin-2-yl]sulfanylmethyl]-N-ethylfuran-2-carboxamide —— C23H34N4O2S
5-[[4-tert-butyl-6-[cyclohexyl(methyl)amino]pyrimidin-2-yl]sulfanylmethyl]-N-ethylfuran-2-carboxamide
—— 5-[(4-Tert-butyl-6-morpholin-4-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-carboxylic acid —— C18H23N3O4S
5-[(4-Tert-butyl-6-morpholin-4-ylpyrimidin-2-yl)sulfanylmethyl]furan-2-carboxylic acid
—— 5-[(5,6-dimethylpyridazin-3-yl)oxymethyl]-3-[(1R)-1-(2-methylpropoxy)ethyl]-1,2,4-oxadiazole —— C15H22N4O3
5-[(5,6-dimethylpyridazin-3-yl)oxymethyl]-3-[(1R)-1-(2-methylpropoxy)ethyl]-1,2,4-oxadiazole
—— 5-({[4-Tert-butyl-6-(diethylamino)pyrimidin-2-YL]sulfanyl}methyl)-N-cyclopropylfuran-2-carboxamide —— C21H30N4O2S
5-({[4-Tert-butyl-6-(diethylamino)pyrimidin-2-YL]sulfanyl}methyl)-N-cyclopropylfuran-2-carboxamide