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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine —— C21H29N5O
5-[[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine
—— (5S)-9-(2-benzyl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H19N3O3S
(5S)-9-(2-benzyl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-(1-tert-butylpyrrole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H23N3O3
(5R)-7-(1-tert-butylpyrrole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-ethylbenzoate —— C16H14N2O4
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 4-ethylbenzoate
—— 5-(2-fluorophenyl)-N-[(1S)-1-pyrimidin-4-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H15FN6
5-(2-fluorophenyl)-N-[(1S)-1-pyrimidin-4-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18F4N2O2
(5S)-9-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18F4N2O2
(5R)-9-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine —— C18H31N5
5-[[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine
—— 5-[[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine —— C18H31N5
5-[[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine
—— (5S)-3-methyl-7-[1-(2-piperazin-1-ylethyl)triazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H25N7O3
(5S)-3-methyl-7-[1-(2-piperazin-1-ylethyl)triazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(2R)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine —— C21H29N5O
5-[[(2R)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-ylpyrimidine
—— (5R)-3-methyl-7-[1-(2-piperazin-1-ylethyl)triazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H25N7O3
(5R)-3-methyl-7-[1-(2-piperazin-1-ylethyl)triazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N4O3S
(5R)-9-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20N4O3
(5S)-3-methyl-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-[3-(4-chlorophenyl)-4-methyl-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H19ClN4O3
(5R)-7-[3-(4-chlorophenyl)-4-methyl-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-methyl-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H21N5O2
(5R)-7-methyl-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-ethylbenzoate —— C18H15N3O5
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 4-ethylbenzoate
—— (5R)-9-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H19N3O4
(5R)-9-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H19N3O4
(5S)-9-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C18H18FN7O
5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— (5S)-9-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N4O3S
(5S)-9-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[2-(2,3-dihydro-1,4-benzoxazin-4-yl)-2-oxoethyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H23N3O4
(5S)-9-[2-(2,3-dihydro-1,4-benzoxazin-4-yl)-2-oxoethyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[(3-ethylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H23N3O2
(5S)-9-[(3-ethylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-7-methyl-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H21N5O2
(5S)-7-methyl-2-(2-methylimidazo[1,2-a]pyrimidine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H19N5O4
(5R)-7-[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-3-methyl-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20N4O3
(5R)-3-methyl-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H25N3O2S
(5R)-3-methyl-9-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(2-phenoxybenzoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H22N2O4
(5S)-9-(2-phenoxybenzoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-(furan-2-yl)pyrimidine —— C18H26N4O
5-[[(3S)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-(furan-2-yl)pyrimidine
—— (5R)-9-(2-phenoxybenzoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H22N2O4
(5R)-9-(2-phenoxybenzoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C18H18FN7O
5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— (5R)-5-(1H-imidazol-5-ylmethyl)-7-methyl-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C15H22N6O
(5R)-5-(1H-imidazol-5-ylmethyl)-7-methyl-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— (5R)-9-[(3-ethylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H23N3O2
(5R)-9-[(3-ethylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-3-methyl-9-[2-(4-propan-2-ylphenyl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H26N2O3
(5S)-3-methyl-9-[2-(4-propan-2-ylphenyl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-9-(5-propan-2-ylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N2O3S
(5R)-3-methyl-9-(5-propan-2-ylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[2-(hydroxymethyl)-3H-benzimidazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O4
(5R)-7-[2-(hydroxymethyl)-3H-benzimidazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H19N5O3
(5R)-9-(5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[2-[(3R)-3-(4-fluoroanilino)piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one —— C19H23FN4O2
5-[2-[(3R)-3-(4-fluoroanilino)piperidin-1-yl]-2-oxoethyl]-2,4-dimethyl-1H-pyrimidin-6-one
—— (5S)-3-methyl-9-(5-propan-2-ylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N2O3S
(5S)-3-methyl-9-(5-propan-2-ylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-[[2-(methylamino)-1,3-thiazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C13H20N4O2S
(5S)-3-methyl-9-[[2-(methylamino)-1,3-thiazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— [5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]-[(3R)-3-morpholin-4-ylpiperidin-1-yl]methanone —— C21H33N3O3
[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]-[(3R)-3-morpholin-4-ylpiperidin-1-yl]methanone
—— [5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]-[(3S)-3-morpholin-4-ylpiperidin-1-yl]methanone —— C21H33N3O3
[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]-[(3S)-3-morpholin-4-ylpiperidin-1-yl]methanone
—— (5R)-9-(1,3-thiazol-4-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C13H18N2O2S
(5R)-9-(1,3-thiazol-4-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-7-[3-(4-chlorophenyl)-4-methyl-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H19ClN4O3
(5S)-7-[3-(4-chlorophenyl)-4-methyl-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-(furan-2-yl)pyrimidine —— C18H26N4O
5-[[(3R)-3-ethyl-4-propan-2-ylpiperazin-1-yl]methyl]-2-(furan-2-yl)pyrimidine
—— (5S)-7-[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H19N5O4
(5S)-7-[5-(1,5-dimethylpyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(1,3-thiazol-4-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C13H18N2O2S
(5S)-9-(1,3-thiazol-4-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[(9-hydroxy-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O4
(5S)-9-[(9-hydroxy-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H25N3O2S
(5S)-3-methyl-9-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-(pyridin-3-ylmethyl)amino]methyl]-N,N-dimethylfuran-2-carboxamide —— C21H28N4O2
5-[[[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-(pyridin-3-ylmethyl)amino]methyl]-N,N-dimethylfuran-2-carboxamide