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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S,7S)-N,N-diethyl-5-(4-ethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H25F3N4O
(5S,7S)-N,N-diethyl-5-(4-ethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7R)-N,N-diethyl-5-(4-ethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H25F3N4O
(5R,7R)-N,N-diethyl-5-(4-ethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S)-3-(2,4-dimethoxyphenyl)-N-(2,5-dimethoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C20H22N2O6
(5S)-3-(2,4-dimethoxyphenyl)-N-(2,5-dimethoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R,7R)-5-(4-ethylphenyl)-N-[(2S)-1-methoxypropan-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H25F3N4O2
(5R,7R)-5-(4-ethylphenyl)-N-[(2S)-1-methoxypropan-2-yl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R)-5-[(3S)-3-(1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C13H17N3O2S
(5R)-5-[(3S)-3-(1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
—— (5R,7S)-N,N-diethyl-5-(4-ethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H25F3N4O
(5R,7S)-N,N-diethyl-5-(4-ethylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R)-3-cyclopentyl-5-[(3-methylpyridin-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-1-ium-4-one —— C21H22F3N4O+
(5R)-3-cyclopentyl-5-[(3-methylpyridin-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-1-ium-4-one
—— 5-Methyl-3-phenyl-7-(4-pyridin-1-ium-2-ylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine —— C22H23N6+
5-Methyl-3-phenyl-7-(4-pyridin-1-ium-2-ylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine
—— (5R)-3-cyclopentyl-5-[(6-methylpyridin-1-ium-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-1-ium-4-one —— C21H23F3N4O+2
(5R)-3-cyclopentyl-5-[(6-methylpyridin-1-ium-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-1-ium-4-one
—— 5-[(3-Methoxyphenoxy)methyl]-3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazole —— C17H13F3N2O4
5-[(3-Methoxyphenoxy)methyl]-3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazole
—— (5S)-3-cyclopentyl-5-[(6-methylpyridin-1-ium-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-4-one —— C21H22F3N4O+
(5S)-3-cyclopentyl-5-[(6-methylpyridin-1-ium-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-4-one
—— 5,6-dimethyl-N-[2-(morpholin-4-yl)ethyl]-7-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine —— C22H29N5O
5,6-dimethyl-N-[2-(morpholin-4-yl)ethyl]-7-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
—— 5-ethyl-N-{(2S)-1-[(3-hydroxypropyl)amino]-3-methyl-1-oxobutan-2-yl}-8-oxo-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide —— C21H27N3O6
5-ethyl-N-{(2S)-1-[(3-hydroxypropyl)amino]-3-methyl-1-oxobutan-2-yl}-8-oxo-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide
—— 5,6-dimethyl-N,7-bis[2-(morpholin-4-yl)ethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine —— C20H32N6O2
5,6-dimethyl-N,7-bis[2-(morpholin-4-yl)ethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
—— 5-[(E)-2-(2-chlorophenyl)ethenyl]-N,N-dimethyl-3-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-1,2,4-triazole-2-sulfonamide —— C18H17ClN4O3S
5-[(E)-2-(2-chlorophenyl)ethenyl]-N,N-dimethyl-3-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-1,2,4-triazole-2-sulfonamide
—— 5-{[(4-chlorophenyl)sulfonyl]methyl}-1-[3-(trifluoromethyl)phenyl]-1H-tetrazole —— C15H10ClF3N4O2S
5-{[(4-chlorophenyl)sulfonyl]methyl}-1-[3-(trifluoromethyl)phenyl]-1H-tetrazole
—— 5,5-dimethyl-2-{[(4-methylpiperidin-1-yl)carbonyl]amino}-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid —— C17H24N2O4S
5,5-dimethyl-2-{[(4-methylpiperidin-1-yl)carbonyl]amino}-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid
—— 5,6-dimethyl-N,7-bis(2-morpholin-4-ium-4-ylethyl)pyrrolo[2,3-d]pyrimidin-4-amine —— C20H34N6O2+2
5,6-dimethyl-N,7-bis(2-morpholin-4-ium-4-ylethyl)pyrrolo[2,3-d]pyrimidin-4-amine
—— (5R,7R)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C14H13F3N4O
(5R,7R)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-ethyl-N-[2-(isopentylamino)-1-methyl-2-oxoethyl]-8-oxo-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide —— C21H27N3O5
5-ethyl-N-[2-(isopentylamino)-1-methyl-2-oxoethyl]-8-oxo-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide
—— (5S)-3-cyclopentyl-5-[(6-methylpyridin-1-ium-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-1-ium-4-one —— C21H23F3N4O+2
(5S)-3-cyclopentyl-5-[(6-methylpyridin-1-ium-2-yl)amino]-2-phenyl-5-(trifluoromethyl)imidazol-1-ium-4-one
—— 5-Chloro-1-(2-piperidin-1-ium-1-ylethyl)indole-2,3-dione —— C15H18ClN2O2+
5-Chloro-1-(2-piperidin-1-ium-1-ylethyl)indole-2,3-dione
—— 5-[(2,4-dichlorophenoxy)methyl]-1-(2,4-dimethylphenyl)-1H-tetrazole —— C16H14Cl2N4O
5-[(2,4-dichlorophenoxy)methyl]-1-(2,4-dimethylphenyl)-1H-tetrazole
—— 5-ethyl-8-oxo-N-[3-oxo-3-(propan-2-ylamino)propyl]-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide —— C19H23N3O5
5-ethyl-8-oxo-N-[3-oxo-3-(propan-2-ylamino)propyl]-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide
—— (5R,7S)-5-(furan-2-yl)-N-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H17F3N4O2
(5R,7S)-5-(furan-2-yl)-N-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5,5-dimethyl-2-{[{[2-(morpholin-4-yl)ethyl]amino}(oxo)acetyl]amino}-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid —— C18H25N3O6S
5,5-dimethyl-2-{[{[2-(morpholin-4-yl)ethyl]amino}(oxo)acetyl]amino}-4,7-dihydro-5H-thieno[2,3-c]pyran-3-carboxylic acid
—— (5S)-3-(3,4-dimethoxyphenyl)-N-quinolin-5-yl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H19N3O4
(5S)-3-(3,4-dimethoxyphenyl)-N-quinolin-5-yl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S,7R)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C14H13F3N4O
(5S,7R)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R)-5-[(3R)-3-(1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C13H17N3O2S
(5R)-5-[(3R)-3-(1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
—— 5-chloro-3-(2-(3,4-dihydroquinolin-1(2H)-yl)-2-oxoethyl)benzo[d]oxazol-2(3H)-one —— C18H15ClN2O3
5-chloro-3-(2-(3,4-dihydroquinolin-1(2H)-yl)-2-oxoethyl)benzo[d]oxazol-2(3H)-one
—— 5-chloro-3-(2-(3,4-dihydroisoquinolin-2(1H)-yl)-2-oxoethyl)benzo[d]oxazol-2(3H)-one —— C18H15ClN2O3
5-chloro-3-(2-(3,4-dihydroisoquinolin-2(1H)-yl)-2-oxoethyl)benzo[d]oxazol-2(3H)-one
—— 5-[[(3R)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C16H20N6O
5-[[(3R)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5S,7S)-N-benzyl-N-methyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H21F3N4O
(5S,7S)-N-benzyl-N-methyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7S)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C14H13F3N4O
(5S,7S)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5Z)-5-(1H-indol-3-ylmethylidene)-2-pyrrolidin-1-yl-1,3-thiazol-4-one —— C16H15N3OS
(5Z)-5-(1H-indol-3-ylmethylidene)-2-pyrrolidin-1-yl-1,3-thiazol-4-one
—— 5-chloro-3-(3-(3,4-dihydroquinolin-1(2H)-yl)-3-oxopropyl)benzo[d]oxazol-2(3H)-one —— C19H17ClN2O3
5-chloro-3-(3-(3,4-dihydroquinolin-1(2H)-yl)-3-oxopropyl)benzo[d]oxazol-2(3H)-one
—— 5-ethyl-N-{2-[(3-methoxypropyl)amino]-2-oxoethyl}-8-oxo-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide —— C19H23N3O6
5-ethyl-N-{2-[(3-methoxypropyl)amino]-2-oxoethyl}-8-oxo-5,8-dihydro[1,3]dioxolo[4,5-g]quinoline-7-carboxamide
—— 5-ethoxy-1-[3-(4-fluorophenyl)-3-oxopropyl]-1H-indole-2,3-dione —— C19H16FNO4
5-ethoxy-1-[3-(4-fluorophenyl)-3-oxopropyl]-1H-indole-2,3-dione
—— (5R)-5-(4-fluorophenyl)-1,3,7-trimethyl-2,4-dioxo-N-phenyl-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide —— C23H21FN4O3
(5R)-5-(4-fluorophenyl)-1,3,7-trimethyl-2,4-dioxo-N-phenyl-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide
—— 5-(4-chlorophenyl)-N,N-dimethylthieno[2,3-d]pyrimidin-4-amine —— C14H12ClN3S
5-(4-chlorophenyl)-N,N-dimethylthieno[2,3-d]pyrimidin-4-amine
—— 5-[[(3S)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C16H20N6O
5-[[(3S)-3-(2-methylpyrazol-3-yl)piperidin-1-yl]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5R,7S)-N-benzyl-N-methyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H21F3N4O
(5R,7S)-N-benzyl-N-methyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[(4-Methylphenoxy)methyl]-3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazole —— C17H13F3N2O3
5-[(4-Methylphenoxy)methyl]-3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazole
—— (5R)-5-[(5-chloro-2-propan-2-yloxybenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide —— C20H22ClN3O4
(5R)-5-[(5-chloro-2-propan-2-yloxybenzoyl)amino]-2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carboxamide
—— 5-chloro-2-[[4-[(2R)-2-methylpiperidin-1-yl]sulfonylbenzoyl]amino]benzamide —— C20H22ClN3O4S
5-chloro-2-[[4-[(2R)-2-methylpiperidin-1-yl]sulfonylbenzoyl]amino]benzamide
—— 5-Methyl-3-(4-methylphenyl)-7-(4-pyridin-2-ylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine —— C23H24N6
5-Methyl-3-(4-methylphenyl)-7-(4-pyridin-2-ylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine
—— (5R,7R)-5-(furan-2-yl)-N-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H17F3N4O2
(5R,7R)-5-(furan-2-yl)-N-(4-methylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-Methyl-3-(4-methylphenyl)-7-(4-pyridin-1-ium-2-ylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine —— C23H25N6+
5-Methyl-3-(4-methylphenyl)-7-(4-pyridin-1-ium-2-ylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine
—— (5S,7S)-5-(1,3-benzodioxol-5-yl)-7-(3-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine —— C18H17N5O3
(5S,7S)-5-(1,3-benzodioxol-5-yl)-7-(3-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine
—— (5R,7R)-5-(1,3-benzodioxol-5-yl)-7-(3-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine —— C18H17N5O3
(5R,7R)-5-(1,3-benzodioxol-5-yl)-7-(3-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine