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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C20H18FN5O
5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— 5-[(2-butyl-1H-imidazol-5-yl)methyl]-2-[[(2S)-2-methylpyrrolidin-1-yl]methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine —— C21H34N6
5-[(2-butyl-1H-imidazol-5-yl)methyl]-2-[[(2S)-2-methylpyrrolidin-1-yl]methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine
—— (5R)-9-[(3,4-difluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C19H22F2N4
(5R)-9-[(3,4-difluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-[(2R)-2-(2-phenylethyl)piperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione —— C17H21N3O4S
5-[(2R)-2-(2-phenylethyl)piperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione
—— (5R)-7-(1-methyl-6-propylpyrazolo[3,4-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decane —— C17H26N6
(5R)-7-(1-methyl-6-propylpyrazolo[3,4-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decane
—— (5R)-3-methyl-7-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H21N5O3
(5R)-3-methyl-7-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[(2-fluoro-3-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H22FNO2
(5R)-9-[(2-fluoro-3-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-2-ethylsulfonyl-9-[(2-fluoro-5-methoxyphenyl)methyl]-2,9-diazaspiro[4.5]decane —— C18H27FN2O3S
(5R)-2-ethylsulfonyl-9-[(2-fluoro-5-methoxyphenyl)methyl]-2,9-diazaspiro[4.5]decane
—— 5-cyclopropyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-phenyl-N-propylpyrazole-3-carboxamide —— C20H25N3O3S
5-cyclopropyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-phenyl-N-propylpyrazole-3-carboxamide
—— 5-[1-[[(2R)-oxolan-2-yl]methyl]triazol-4-yl]-3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazole —— C18H28N6O2
5-[1-[[(2R)-oxolan-2-yl]methyl]triazol-4-yl]-3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazole
—— (5S)-7-(1-methyl-6-propylpyrazolo[3,4-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decane —— C17H26N6
(5S)-7-(1-methyl-6-propylpyrazolo[3,4-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decane
—— (5R)-2-(4,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O4
(5R)-2-(4,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,6-dichlorophenyl)acetate —— C17H11Cl3N2O3
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,6-dichlorophenyl)acetate
—— (5S)-9-[(3,4-difluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C19H22F2N4
(5S)-9-[(3,4-difluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-[(3R)-3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C20H24F3N5O2
5-[(3R)-3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— 5-[1-[[(2S)-oxolan-2-yl]methyl]triazol-4-yl]-3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazole —— C18H28N6O2
5-[1-[[(2S)-oxolan-2-yl]methyl]triazol-4-yl]-3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazole
—— 5-[(2S)-2-(2-phenylethyl)piperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione —— C17H21N3O4S
5-[(2S)-2-(2-phenylethyl)piperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione
—— 5-(2,3-dihydroindol-1-ylsulfonyl)-2-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide —— C21H24N2O5S
5-(2,3-dihydroindol-1-ylsulfonyl)-2-methoxy-N-[[(2S)-oxolan-2-yl]methyl]benzamide
—— 5-ethoxy-3-methyl-N-(4-methylsulfonylphenyl)-1-benzofuran-2-carboxamide —— C19H19NO5S
5-ethoxy-3-methyl-N-(4-methylsulfonylphenyl)-1-benzofuran-2-carboxamide
—— (5R)-3-methyl-9-(2-pyridin-2-ylethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H23N3O2
(5R)-3-methyl-9-(2-pyridin-2-ylethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-7-(2-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O3S
(5S)-3-methyl-7-(2-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-N-(3,4-diethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H25NO3S
(5R)-N-(3,4-diethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-chloro-5-methylsulfanylbenzoate —— C18H14ClNO3S
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-chloro-5-methylsulfanylbenzoate
—— 5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide —— C20H25FN2O2
5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide
—— (5R)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane —— C22H34N2O2
(5R)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
—— (5S)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane —— C22H34N2O2
(5S)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H30N4O3
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C14H20N2O2S
(5S)-9-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-N-(3,4-diethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H25NO3S
(5S)-N-(3,4-diethoxyphenyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(2R)-2-(cyclopropylcarbamoyl)piperazine-1-carbonyl]-4-oxo-1-propan-2-ylpyridine-3-carboxylic acid —— C18H24N4O5
5-[(2R)-2-(cyclopropylcarbamoyl)piperazine-1-carbonyl]-4-oxo-1-propan-2-ylpyridine-3-carboxylic acid
—— [(5S)-9-(2-methoxyethyl)-2,9-diazaspiro[4.5]decan-2-yl]-quinoxalin-5-ylmethanone —— C20H26N4O2
[(5S)-9-(2-methoxyethyl)-2,9-diazaspiro[4.5]decan-2-yl]-quinoxalin-5-ylmethanone
—— (5-bromo-2-methoxyphenyl)methyl-[2-[[(1S)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl]-methylazanium —— C17H23BrN3O2+
(5-bromo-2-methoxyphenyl)methyl-[2-[[(1S)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl]-methylazanium
—— (5S)-2-(4,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O4
(5S)-2-(4,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-methyl-7-[3-(5-methyltetrazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H20N6O2
(5R)-3-methyl-7-[3-(5-methyltetrazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C20H18FN5O
5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— 5-(4-acetylphenyl)-N-(5-methylpyridin-2-yl)furan-2-carboxamide —— C19H16N2O3
5-(4-acetylphenyl)-N-(5-methylpyridin-2-yl)furan-2-carboxamide
—— 5-[[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide —— C20H25FN2O2
5-[[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide
—— (5R)-3-methyl-9-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H26N2O3S
(5R)-3-methyl-9-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C23H27N3O4
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl)-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone —— C17H27N5O
(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl)-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone
—— 5-phenyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H18N6
5-phenyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-3-methyl-9-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H26N2O3S
(5S)-3-methyl-9-[[5-(4-methylphenyl)sulfanylfuran-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(1S)-1-[(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine —— C15H15N9S
5-[(1S)-1-[(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine
—— (5S)-3-methyl-9-[2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O5
(5S)-3-methyl-9-[2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N2O4
(5S)-9-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-ethyl-6-methyl-N-[[(6R)-4-methyl-1,4-oxazepan-6-yl]methyl]thieno[2,3-d]pyrimidin-4-amine —— C16H24N4OS
5-ethyl-6-methyl-N-[[(6R)-4-methyl-1,4-oxazepan-6-yl]methyl]thieno[2,3-d]pyrimidin-4-amine
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(cyclopropylmethyl)pyridazin-3-one —— C14H22N4O2
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(cyclopropylmethyl)pyridazin-3-one
—— 5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]pyridine-2-carbonitrile —— C22H25FN4O
5-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]pyridine-2-carbonitrile
—— (5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl)-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone —— C17H27N5O
(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-3-yl)-[(3S)-3-pyrrolidin-1-ylpiperidin-1-yl]methanone
—— (5R)-3-methyl-9-[2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O5
(5R)-3-methyl-9-[2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one