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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-N-cyclohexyl-5-(4-nitrophenyl)-4,5-dihydro-1,3-thiazol-2-amine —— C15H19N3O2S
(5S)-N-cyclohexyl-5-(4-nitrophenyl)-4,5-dihydro-1,3-thiazol-2-amine
—— [5-(1H-benzimidazol-2-yl)-1H-pyrrol-3-yl]-(2-hydroxy-5-methylphenyl)methanone —— C19H15N3O2
[5-(1H-benzimidazol-2-yl)-1H-pyrrol-3-yl]-(2-hydroxy-5-methylphenyl)methanone
—— 5-chloro-4-(4-fluoroanilino)-1H-pyridazin-6-one —— C10H7ClFN3O
5-chloro-4-(4-fluoroanilino)-1H-pyridazin-6-one
—— 5-Chloro-4-[(4-phenylphenoxy)methyl]thiadiazole —— C15H11ClN2OS
5-Chloro-4-[(4-phenylphenoxy)methyl]thiadiazole
—— 5-[(4-chlorophenyl)methoxy]-6-oxo-1H-pyrazine-2,3-dicarbonitrile —— C13H7ClN4O2
5-[(4-chlorophenyl)methoxy]-6-oxo-1H-pyrazine-2,3-dicarbonitrile
—— 5-Chloro-4-[[4-(3,4-dimethylphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]thiadiazole —— C19H16ClN5S2
5-Chloro-4-[[4-(3,4-dimethylphenyl)-5-phenyl-1,2,4-triazol-3-yl]sulfanylmethyl]thiadiazole
—— 5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C32H56N6O9S2
5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— 5-(4-Imidazo[2,1-b][1,3]thiazol-6-ylanilino)-5-oxopentanoate —— C16H14N3O3S-
5-(4-Imidazo[2,1-b][1,3]thiazol-6-ylanilino)-5-oxopentanoate
—— (5-Fluoro-2-hydroxyphenyl)-pyridazino[1,6-a]benzimidazol-3-ylmethanone —— C17H10FN3O2
(5-Fluoro-2-hydroxyphenyl)-pyridazino[1,6-a]benzimidazol-3-ylmethanone
—— 5-(4-acetylphenyl)-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methylfuran-2-carboxamide —— C23H22N2O5
5-(4-acetylphenyl)-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methylfuran-2-carboxamide
—— (5R)-3-methyl-9-(2,4,5-trifluorophenyl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H17F3N2O4S
(5R)-3-methyl-9-(2,4,5-trifluorophenyl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-7-[4-(2-methyltetrazol-5-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N6O3
(5R)-3-methyl-7-[4-(2-methyltetrazol-5-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-3-methyl-9-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H19N5O3
(5R)-3-methyl-9-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-(2,4,5-trifluorophenyl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H17F3N2O4S
(5S)-3-methyl-9-(2,4,5-trifluorophenyl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(2,4-dimethyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H19N3O3S
(5S)-9-(2,4-dimethyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(4R)-4-(dimethylamino)azepane-1-carbonyl]-1H-pyridin-2-one —— C14H21N3O2
5-[(4R)-4-(dimethylamino)azepane-1-carbonyl]-1H-pyridin-2-one
—— 5-tert-butyl-2-methoxy-N-[[(6S)-1,4-oxazepan-6-yl]methyl]benzenesulfonamide —— C17H28N2O4S
5-tert-butyl-2-methoxy-N-[[(6S)-1,4-oxazepan-6-yl]methyl]benzenesulfonamide
—— 5-Phenyl-2-[[2-[(4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]thiophene-3-carboxamide —— C18H17N5O2S2
5-Phenyl-2-[[2-[(4-prop-2-enyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]thiophene-3-carboxamide
—— (5R)-9-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H24FNO4
(5R)-9-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-9-(2,4-dimethyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H19N3O3S
(5R)-9-(2,4-dimethyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-fluoro-1-methyl-2-[[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]indole —— C21H24FN3O
5-fluoro-1-methyl-2-[[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]indole
—— (5S)-3-methyl-7-[4-(2-methyltetrazol-5-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N6O3
(5S)-3-methyl-7-[4-(2-methyltetrazol-5-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H24FNO4
(5S)-9-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-3-methyl-9-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H19N5O3
(5S)-3-methyl-9-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[2-(1-methylindol-3-yl)sulfanylacetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O3S
(5S)-9-[2-(1-methylindol-3-yl)sulfanylacetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H25N3O3
(5R)-9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H27N5O2
(5R)-9-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-methyl-1-[(3R)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]hexan-1-one —— C22H35N3O
5-methyl-1-[(3R)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl]hexan-1-one
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide —— C20H24F2N2O2
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide
—— (5R)-9-(2-methoxypyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H19N3O4
(5R)-9-(2-methoxypyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[methyl(2-phenylethyl)amino]-2-[2-[(3R)-oxolan-3-yl]ethyl]pyridazin-3-one —— C19H25N3O2
5-[methyl(2-phenylethyl)amino]-2-[2-[(3R)-oxolan-3-yl]ethyl]pyridazin-3-one
—— (5S)-3-methyl-9-[(1-methylimidazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H22N4O2
(5S)-3-methyl-9-[(1-methylimidazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— [(5R)-5-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl]-(3-pyridin-4-ylazetidin-1-yl)methanone —— C17H20N4O
[(5R)-5-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl]-(3-pyridin-4-ylazetidin-1-yl)methanone
—— (5R)-9-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H27N5O2
(5R)-9-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— [5,6-dimethyl-4-[[(1R)-1-pyridin-2-ylethyl]amino]thieno[2,3-d]pyrimidin-2-yl]methyl-diethylazanium —— C20H28N5S+
[5,6-dimethyl-4-[[(1R)-1-pyridin-2-ylethyl]amino]thieno[2,3-d]pyrimidin-2-yl]methyl-diethylazanium
—— (5S)-9-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H27N5O2
(5S)-9-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-(methylsulfanylmethyl)-1,2,4-oxadiazole —— C16H18FN5OS
5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-(methylsulfanylmethyl)-1,2,4-oxadiazole
—— (5R)-9-[2-(1-methylindol-3-yl)sulfanylacetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O3S
(5R)-9-[2-(1-methylindol-3-yl)sulfanylacetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl]-(3-pyridin-4-ylazetidin-1-yl)methanone —— C17H20N4O
[(5S)-5-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl]-(3-pyridin-4-ylazetidin-1-yl)methanone
—— (5S)-9-(2-methoxypyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H19N3O4
(5S)-9-(2-methoxypyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O2
(5S)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-fluoropyridin-3-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C20H22FN3O
(5-fluoropyridin-3-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5S)-9-(2,3-dimethyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O4S
(5S)-9-(2,3-dimethyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H28N2O
(5S)-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5,6-dimethyl-4-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[2,3-d]pyrimidin-2-yl]methyl-diethylazanium —— C20H28N5S+
[5,6-dimethyl-4-[[(1S)-1-pyridin-2-ylethyl]amino]thieno[2,3-d]pyrimidin-2-yl]methyl-diethylazanium
—— 5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-(methylsulfanylmethyl)-1,2,4-oxadiazole —— C16H18FN5OS
5-[[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-(methylsulfanylmethyl)-1,2,4-oxadiazole
—— (5R)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O2
(5R)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(2-methoxy-6,7-dihydro-5H-cyclopenta[b]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H23N3O4
(5R)-9-(2-methoxy-6,7-dihydro-5H-cyclopenta[b]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(2,3-dimethyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O4S
(5R)-9-(2,3-dimethyl-5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide —— C20H24F2N2O2
5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide