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—— (5R)-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O2
(5R)-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H28N2O4
(5R)-9-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-(4-fluorophenyl)-N-[(1S)-1-pyridin-2-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(4-fluorophenyl)-N-[(1S)-1-pyridin-2-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-3-methyl-9-(pyridin-4-ylmethyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H19N3O2
(5R)-3-methyl-9-(pyridin-4-ylmethyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(4,6-dimethoxypyrimidin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H20N4O4
(5S)-9-(4,6-dimethoxypyrimidin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[2-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H24N4O4
5-[2-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (5S)-9-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H25N5O3
(5S)-9-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-methyl-1-[3-[2-[5-[(2R)-oxan-2-yl]furan-2-yl]imidazol-1-yl]phenyl]tetrazole —— C20H20N6O2
5-methyl-1-[3-[2-[5-[(2R)-oxan-2-yl]furan-2-yl]imidazol-1-yl]phenyl]tetrazole
—— (5R)-9-(4,6-dimethoxypyrimidin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H20N4O4
(5R)-9-(4,6-dimethoxypyrimidin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5,6-bis(4-methylphenyl)-3-[[(2R)-oxolan-2-yl]methylsulfanyl]-1,2,4-triazine —— C22H23N3OS
5,6-bis(4-methylphenyl)-3-[[(2R)-oxolan-2-yl]methylsulfanyl]-1,2,4-triazine
—— (5R)-7-(furan-2-ylmethyl)-5-(1H-imidazol-5-ylmethyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H24N6O2
(5R)-7-(furan-2-ylmethyl)-5-(1H-imidazol-5-ylmethyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methanone —— C18H21ClN4O2
(5-chloro-2-methylpyrimidin-4-yl)-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methanone
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C19H17FN2O5
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— (5S)-7-(furan-2-ylmethyl)-5-(1H-imidazol-5-ylmethyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H24N6O2
(5S)-7-(furan-2-ylmethyl)-5-(1H-imidazol-5-ylmethyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 5-[2-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H24N4O4
5-[2-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-(4-fluorophenyl)-N-[(1R)-1-pyridin-2-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(4-fluorophenyl)-N-[(1R)-1-pyridin-2-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-fluoro-2-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine —— C19H27FN6
5-fluoro-2-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine
—— 5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyridin-2-amine —— C19H22N6O
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyridin-2-amine
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-2-(4-propan-2-ylpiperazin-1-yl)pyrimidine —— C17H29N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-2-(4-propan-2-ylpiperazin-1-yl)pyrimidine
—— 5-fluoro-2-[(3S)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine —— C19H27FN6
5-fluoro-2-[(3S)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methanone —— C18H21ClN4O2
(5-chloro-2-methylpyrimidin-4-yl)-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methanone
—— (5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C20H16FNO4
(5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— [5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C20H15ClFNO4
[5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— 5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyridin-2-amine —— C19H22N6O
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyridin-2-amine
—— (5S)-9-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H20ClFN2O3
(5S)-9-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— [5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone —— C18H18N4OS
[5-(5-methylthiophen-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(3-pyrazol-1-ylpropyl)pyrimidin-2-amine —— C16H24N6O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(3-pyrazol-1-ylpropyl)pyrimidin-2-amine
—— (5S)-7-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H20ClN3O2
(5S)-7-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[(2,2-difluoro-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H16F2N2O4
(5S)-9-[(2,2-difluoro-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[(2,2-difluoro-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H16F2N2O4
(5R)-9-[(2,2-difluoro-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(3S)-4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C17H23N5O3
5-[[(3S)-4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5R)-9-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H20ClFN2O3
(5R)-9-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-2-(4-propan-2-ylpiperazin-1-yl)pyrimidine —— C17H29N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-2-(4-propan-2-ylpiperazin-1-yl)pyrimidine
—— 5-[(3S)-1-(5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl)piperidin-3-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C20H28N6O
5-[(3S)-1-(5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl)piperidin-3-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-ethyl-2,3-dimethyl-N-[(2R)-2-(4-methylpiperazin-1-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H32N6
5-ethyl-2,3-dimethyl-N-[(2R)-2-(4-methylpiperazin-1-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-7-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H20ClN3O2
(5R)-7-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— [5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C19H14ClFN2O4
[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— [5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C17H13FN2O5
[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— 5,6-dimethyl-3-[[(2S)-oxolan-2-yl]methyl]thieno[2,3-d]pyrimidin-4-one —— C13H16N2O2S
5,6-dimethyl-3-[[(2S)-oxolan-2-yl]methyl]thieno[2,3-d]pyrimidin-4-one
—— (5-acetyl-2-ethoxyphenyl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C21H21FO5
(5-acetyl-2-ethoxyphenyl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— (5R)-7-[(6-ethoxyquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C19H23N3O3
(5R)-7-[(6-ethoxyquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[[4-[(dimethylamino)methyl]thiophen-2-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H25N3O2S
(5S)-9-[[4-[(dimethylamino)methyl]thiophen-2-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-phenyl-1,3,4-oxadiazol-2-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C19H15FN2O4
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— (5R)-9-[[4-[(dimethylamino)methyl]thiophen-2-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H25N3O2S
(5R)-9-[[4-[(dimethylamino)methyl]thiophen-2-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C17H13FN2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— [5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C20H17FN2O4
[5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 2-(2,5-difluorophenyl)sulfanylacetate —— C18H13F2NO3S
(5-Phenyl-1,2-oxazol-3-yl)methyl 2-(2,5-difluorophenyl)sulfanylacetate
—— 5-(furan-2-yl)-2-[[(2S)-oxolan-2-yl]methylsulfanyl]-3-phenylthieno[2,3-d]pyrimidin-4-one —— C21H18N2O3S2
5-(furan-2-yl)-2-[[(2S)-oxolan-2-yl]methylsulfanyl]-3-phenylthieno[2,3-d]pyrimidin-4-one
—— 5-(furan-2-yl)-2-[[(2R)-oxolan-2-yl]methylsulfanyl]-3-phenylthieno[2,3-d]pyrimidin-4-one —— C21H18N2O3S2
5-(furan-2-yl)-2-[[(2R)-oxolan-2-yl]methylsulfanyl]-3-phenylthieno[2,3-d]pyrimidin-4-one
—— (5-methylpyrazin-2-yl)-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone —— C17H26N4O2
(5-methylpyrazin-2-yl)-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]methanone