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—— 5-chloro-1-methyl-N-[(5S)-2-methyl-5,6,7,8-tetrahydroquinazolin-5-yl]pyrazole-4-carboxamide —— C14H16ClN5O
5-chloro-1-methyl-N-[(5S)-2-methyl-5,6,7,8-tetrahydroquinazolin-5-yl]pyrazole-4-carboxamide
—— 5-[(2,2-dimethylpyrrolidin-1-yl)methyl]-N,N-dimethylfuran-2-sulfonamide —— C13H22N2O3S
5-[(2,2-dimethylpyrrolidin-1-yl)methyl]-N,N-dimethylfuran-2-sulfonamide
—— (5R)-1-(furan-2-ylmethyl)-5-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one —— C16H14N4O3
(5R)-1-(furan-2-ylmethyl)-5-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
—— 5-[[(R)-cyclohexylmethylsulfinyl]methyl]-3-(3-methylphenyl)-1,2,4-oxadiazole —— C17H22N2O2S
5-[[(R)-cyclohexylmethylsulfinyl]methyl]-3-(3-methylphenyl)-1,2,4-oxadiazole
—— 5-propan-2-yl-N-[(4R)-1-pyridin-4-yl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide —— C19H21N5O2
5-propan-2-yl-N-[(4R)-1-pyridin-4-yl-4,5,6,7-tetrahydroindazol-4-yl]-1,2-oxazole-3-carboxamide
—— 5-[[(S)-cyclohexylmethylsulfinyl]methyl]-3-(3-methylphenyl)-1,2,4-oxadiazole —— C17H22N2O2S
5-[[(S)-cyclohexylmethylsulfinyl]methyl]-3-(3-methylphenyl)-1,2,4-oxadiazole
—— (5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(2R)-2-methylpiperidine-1-carbonyl]piperidin-2-one —— C20H28N2O3
(5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(2R)-2-methylpiperidine-1-carbonyl]piperidin-2-one
—— (5R)-1-(furan-2-ylmethyl)-5-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one —— C16H14N4O3
(5R)-1-(furan-2-ylmethyl)-5-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
—— (5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(piperidine-1-carbonyl)piperidin-2-one —— C19H26N2O3
(5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(piperidine-1-carbonyl)piperidin-2-one
—— (5S,6S)-5-(4-ethylpiperazine-1-carbonyl)-6-(3-fluorophenyl)-1-methylpiperidin-2-one —— C19H26FN3O2
(5S,6S)-5-(4-ethylpiperazine-1-carbonyl)-6-(3-fluorophenyl)-1-methylpiperidin-2-one
—— 5-cyclopropyl-1-methyl-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide —— C16H21N5O
5-cyclopropyl-1-methyl-N-[(4R)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]pyrazole-3-carboxamide
—— (5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperazine-1-carbonyl)piperidin-2-one —— C19H27N3O3
(5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperazine-1-carbonyl)piperidin-2-one
—— (5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(morpholine-4-carbonyl)piperidin-2-one —— C18H24N2O4
(5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(morpholine-4-carbonyl)piperidin-2-one
—— (5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one —— C20H28N2O3
(5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one
—— (5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one —— C20H28N2O3
(5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one
—— (5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one —— C24H29N3O3
(5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one
—— (5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one —— C24H29N3O3
(5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one
—— (5S,6S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one —— C24H28FN3O3
(5S,6S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one
—— (5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperazine-1-carbonyl)piperidin-2-one —— C19H27N3O3
(5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperazine-1-carbonyl)piperidin-2-one
—— (5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(3R)-3-methylpiperidine-1-carbonyl]piperidin-2-one —— C20H28N2O3
(5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(3R)-3-methylpiperidine-1-carbonyl]piperidin-2-one
—— (5R)-1-(furan-2-ylmethyl)-5-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one —— C16H14N4O3
(5R)-1-(furan-2-ylmethyl)-5-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
—— (5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one —— C18H24N2O3
(5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one
—— 5-ethyl-3-[(2S)-1-(2-pyridin-2-ylethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole —— C15H20N4O
5-ethyl-3-[(2S)-1-(2-pyridin-2-ylethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
—— (5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(thiomorpholine-4-carbonyl)piperidin-2-one —— C18H24N2O3S
(5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(thiomorpholine-4-carbonyl)piperidin-2-one
—— (5R,6S)-5-(azepane-1-carbonyl)-6-(3-fluorophenyl)-1-methylpiperidin-2-one —— C19H25FN2O2
(5R,6S)-5-(azepane-1-carbonyl)-6-(3-fluorophenyl)-1-methylpiperidin-2-one
—— (5R,6S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one —— C24H28FN3O3
(5R,6S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one
—— (5S,6R)-6-(3-fluorophenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one —— C17H21FN2O2
(5S,6R)-6-(3-fluorophenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one
—— (5S,6S)-6-(3-fluorophenyl)-1-methyl-5-(thiomorpholine-4-carbonyl)piperidin-2-one —— C17H21FN2O2S
(5S,6S)-6-(3-fluorophenyl)-1-methyl-5-(thiomorpholine-4-carbonyl)piperidin-2-one
—— (5R,6S)-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-(3-fluorophenyl)-1-methylpiperidin-2-one —— C19H25FN2O3
(5R,6S)-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-(3-fluorophenyl)-1-methylpiperidin-2-one
—— (5R,6R)-6-(3-fluorophenyl)-1-methyl-5-(piperidine-1-carbonyl)piperidin-2-one —— C18H23FN2O2
(5R,6R)-6-(3-fluorophenyl)-1-methyl-5-(piperidine-1-carbonyl)piperidin-2-one
—— (5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(morpholine-4-carbonyl)piperidin-2-one —— C18H24N2O4
(5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(morpholine-4-carbonyl)piperidin-2-one
—— (5S,6R)-5-(3-fluorophenyl)-4-methyl-6-(thiomorpholine-4-carbonyl)morpholin-3-one —— C16H19FN2O3S
(5S,6R)-5-(3-fluorophenyl)-4-methyl-6-(thiomorpholine-4-carbonyl)morpholin-3-one
—— (5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-(morpholine-4-carbonyl)piperidin-2-one —— C18H24N2O4
(5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-(morpholine-4-carbonyl)piperidin-2-one
—— (5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one —— C20H28N2O3
(5R,6S)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one
—— (5R,6S)-5-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-(3-fluorophenyl)-1-methylpiperidin-2-one —— C19H25FN2O3
(5R,6S)-5-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-(3-fluorophenyl)-1-methylpiperidin-2-one
—— (5S,6R)-6-(3-fluorophenyl)-1-methyl-5-(thiomorpholine-4-carbonyl)piperidin-2-one —— C17H21FN2O2S
(5S,6R)-6-(3-fluorophenyl)-1-methyl-5-(thiomorpholine-4-carbonyl)piperidin-2-one
—— (5S,6R)-5-(azepane-1-carbonyl)-6-(3-fluorophenyl)-1-methylpiperidin-2-one —— C19H25FN2O2
(5S,6R)-5-(azepane-1-carbonyl)-6-(3-fluorophenyl)-1-methylpiperidin-2-one
—— (5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one —— C18H24N2O3
(5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one
—— (5R,6R)-6-(3-fluorophenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one —— C17H21FN2O2
(5R,6R)-6-(3-fluorophenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one
—— (5S,6R)-5-(4-benzylpiperazine-1-carbonyl)-6-(4-methoxyphenyl)-1-methylpiperidin-2-one —— C25H31N3O3
(5S,6R)-5-(4-benzylpiperazine-1-carbonyl)-6-(4-methoxyphenyl)-1-methylpiperidin-2-one
—— (5S,6R)-6-(3-fluorophenyl)-1-methyl-5-(piperidine-1-carbonyl)piperidin-2-one —— C18H23FN2O2
(5S,6R)-6-(3-fluorophenyl)-1-methyl-5-(piperidine-1-carbonyl)piperidin-2-one
—— (5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(2R)-2-methylpiperidine-1-carbonyl]piperidin-2-one —— C20H28N2O3
(5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(2R)-2-methylpiperidine-1-carbonyl]piperidin-2-one
—— (5R,6S)-6-(3-fluorophenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one —— C17H21FN2O2
(5R,6S)-6-(3-fluorophenyl)-1-methyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one
—— (5S,6R)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one —— C24H28FN3O3
(5S,6R)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one
—— (5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(3R)-3-methylpiperidine-1-carbonyl]piperidin-2-one —— C20H28N2O3
(5S,6S)-6-(4-methoxyphenyl)-1-methyl-5-[(3R)-3-methylpiperidine-1-carbonyl]piperidin-2-one
—— (5R,6S)-5-(4-benzylpiperazine-1-carbonyl)-6-(4-methoxyphenyl)-1-methylpiperidin-2-one —— C25H31N3O3
(5R,6S)-5-(4-benzylpiperazine-1-carbonyl)-6-(4-methoxyphenyl)-1-methylpiperidin-2-one
—— (5S,6S)-6-(3-fluorophenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one —— C23H26FN3O2
(5S,6S)-6-(3-fluorophenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one
—— (5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one —— C20H28N2O3
(5R,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-methylpiperidine-1-carbonyl)piperidin-2-one
—— (5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one —— C24H29N3O3
(5S,6R)-6-(4-methoxyphenyl)-1-methyl-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one
—— 5-methyl-N-(2-morpholin-4-ium-4-ylethyl)-N-[3-oxo-3-(pyridin-2-ylmethylamino)propyl]pyrazine-2-carboxamide —— C21H29N6O3+
5-methyl-N-(2-morpholin-4-ium-4-ylethyl)-N-[3-oxo-3-(pyridin-2-ylmethylamino)propyl]pyrazine-2-carboxamide