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—— 5-[(3R)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C21H29N3O3
5-[(3R)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— (5R)-9-[2-(2-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H22N2O4
(5R)-9-[2-(2-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[2-(2-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H22N2O4
(5S)-9-[2-(2-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3-propan-2-ylimidazol-4-yl)methyl]pyridazin-3-one —— C17H26N6O2
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3-propan-2-ylimidazol-4-yl)methyl]pyridazin-3-one
—— (5S)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H20N4O3
(5S)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-methylamino]methyl]-N,N-dimethylpyridin-2-amine —— C16H24N4S
5-[[[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-methylamino]methyl]-N,N-dimethylpyridin-2-amine
—— 5-methyl-N-[(3R)-1-[[4-(2-methylpropyl)phenyl]methyl]piperidin-3-yl]-1,2-oxazole-4-sulfonamide —— C20H29N3O3S
5-methyl-N-[(3R)-1-[[4-(2-methylpropyl)phenyl]methyl]piperidin-3-yl]-1,2-oxazole-4-sulfonamide
—— (5S)-2-(1H-indole-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C23H24N4O2
(5S)-2-(1H-indole-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O4
(5R)-9-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(3-methylsulfonylbenzoyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H18N2O5S
(5R)-9-(3-methylsulfonylbenzoyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-propyl-1H-pyrazol-4-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C21H28N4O
(5-propyl-1H-pyrazol-4-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5S)-9-(1,3-benzothiazol-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H20N2O2S
(5S)-9-(1,3-benzothiazol-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-(3-methylsulfonylbenzoyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H18N2O5S
(5S)-9-(3-methylsulfonylbenzoyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5,6-diamino-3-[(2S)-butan-2-yl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxo-1H-pyrrolo[2,3-c][2,7]naphthyridine-9-carbonitrile —— C21H27N7O2
5,6-diamino-3-[(2S)-butan-2-yl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxo-1H-pyrrolo[2,3-c][2,7]naphthyridine-9-carbonitrile
—— (5R)-3-methyl-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H17F3N4O2
(5R)-3-methyl-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N2O6
(5R)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-7-(5-methyl-1H-imidazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H16N4O3
(5R)-3-methyl-7-(5-methyl-1H-imidazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5-Methoxycarbonylfuran-2-yl)methyl 2-aminopyridin-1-ium-3-carboxylate —— C13H13N2O5+
(5-Methoxycarbonylfuran-2-yl)methyl 2-aminopyridin-1-ium-3-carboxylate
—— (5R)-9-[(2,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H25NO4
(5R)-9-[(2,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-(4-Chloro-3-morpholin-4-ylsulfonylphenyl)-1,3,4-thiadiazol-2-amine —— C12H13ClN4O3S2
5-(4-Chloro-3-morpholin-4-ylsulfonylphenyl)-1,3,4-thiadiazol-2-amine
—— 5,6-diamino-3-[(2S)-butan-2-yl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxo-1H-pyrrolo[2,3-c][2,7]naphthyridin-7-ium-9-carbonitrile —— C21H28N7O2+
5,6-diamino-3-[(2S)-butan-2-yl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxo-1H-pyrrolo[2,3-c][2,7]naphthyridin-7-ium-9-carbonitrile
—— [5-(2-chlorophenyl)-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl]methyl pentanoate —— C18H17ClN2O3S
[5-(2-chlorophenyl)-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl]methyl pentanoate
—— (5R)-5-(2-phenylethyl)-2-[2-(trifluoromethyl)phenyl]-5,6-dihydropyrazolo[3,4-e][1,3]oxazin-7-one —— C20H16F3N3O2
(5R)-5-(2-phenylethyl)-2-[2-(trifluoromethyl)phenyl]-5,6-dihydropyrazolo[3,4-e][1,3]oxazin-7-one
—— 5-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C22H28N4OS
5-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— 5-[(3S)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one —— C17H23N5O2
5-[(3S)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one
—— [5-(2-chlorophenyl)furan-2-yl]-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C17H18ClNO4
[5-(2-chlorophenyl)furan-2-yl]-[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— (5S)-9-[(2,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H25NO4
(5S)-9-[(2,5-dimethoxyphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[[[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-methylamino]methyl]-N,N-dimethylpyridin-2-amine —— C16H24N4S
5-[[[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-methylamino]methyl]-N,N-dimethylpyridin-2-amine
—— 5-ethyl-3-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H20FN3O
5-ethyl-3-[[(2R)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[(1R)-1-(4-fluorophenyl)ethyl]sulfanyl-1-(2-methoxy-5-methylphenyl)tetrazole —— C17H17FN4OS
5-[(1R)-1-(4-fluorophenyl)ethyl]sulfanyl-1-(2-methoxy-5-methylphenyl)tetrazole
—— 5-ethyl-3-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H20FN3O
5-ethyl-3-[[(2S)-2-(4-fluorophenyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5S)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N2O6
(5S)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-cyclopropyl-2-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methylsulfanyl]-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one —— C21H20N2O3S2
5-cyclopropyl-2-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methylsulfanyl]-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one
—— 5-chloro-3-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C13H18ClN3O3
5-chloro-3-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— 5-chloro-3-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C13H18ClN3O3
5-chloro-3-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— (5R)-2-(2-amino-6-methylpyrimidin-4-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H29N5O3
(5R)-2-(2-amino-6-methylpyrimidin-4-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O
(5R)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[2-ethyl-5-(2-methylpropyl)pyrazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H30N4O3
(5R)-9-[2-ethyl-5-(2-methylpropyl)pyrazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O
(5S)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1S)-1-(4-fluorophenyl)ethyl]sulfanyl-1-(2-methoxy-5-methylphenyl)tetrazole —— C17H17FN4OS
5-[(1S)-1-(4-fluorophenyl)ethyl]sulfanyl-1-(2-methoxy-5-methylphenyl)tetrazole
—— (5S)-9-[4-(1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C13H19N5O3
(5S)-9-[4-(1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[3-(2-ethylimidazol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5S)-9-[3-(2-ethylimidazol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[2-ethyl-5-(2-methylpropyl)pyrazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H30N4O3
(5S)-9-[2-ethyl-5-(2-methylpropyl)pyrazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[(3-benzylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C20H25N3O2
(5S)-9-[(3-benzylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-propyl-1H-pyrazol-4-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C21H28N4O
(5-propyl-1H-pyrazol-4-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5R)-7-(2,2-dimethylpropyl)-2-(6-methyl-4-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O3
(5R)-7-(2,2-dimethylpropyl)-2-(6-methyl-4-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-tert-butyl-4-[[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl]furan-2-carboxamide —— C16H26N2O4
5-tert-butyl-4-[[(3S)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl]furan-2-carboxamide
—— (5S)-3-methyl-7-(5-methyl-1H-imidazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H16N4O3
(5S)-3-methyl-7-(5-methyl-1H-imidazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-5-methyl-N-(5-prop-2-enylsulfanyl-1,3,4-thiadiazol-2-yl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C15H17N3OS3
(5R)-5-methyl-N-(5-prop-2-enylsulfanyl-1,3,4-thiadiazol-2-yl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one —— C17H23N5O2
5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]pyridazin-3-one