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—— 5-[[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-N-(4-methylphenyl)-1,3,4-thiadiazol-2-amine —— C18H17N5O2S2
5-[[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-N-(4-methylphenyl)-1,3,4-thiadiazol-2-amine
—— 5-[[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-(3-methylphenyl)-1,3,4-thiadiazol-2-amine —— C19H17N5O2S2
5-[[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-(3-methylphenyl)-1,3,4-thiadiazol-2-amine
—— (5R,7R)-N-[1-(1,3-benzodioxol-5-yl)cyclopentyl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H23F3N4O3
(5R,7R)-N-[1-(1,3-benzodioxol-5-yl)cyclopentyl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 1-(4-fluorophenyl)-2,5-dimethylpyrrole-3-carboxylate —— C22H20FN3O4
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 1-(4-fluorophenyl)-2,5-dimethylpyrrole-3-carboxylate
—— 5-(3-Fluorophenyl)-4-(5-methylpyridin-2-yl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)-1,2,4-triazol-3-one —— C20H20FN5O2
5-(3-Fluorophenyl)-4-(5-methylpyridin-2-yl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)-1,2,4-triazol-3-one
—— (5-Tert-butyl-3-methylfuran-2-yl)-(4-pyridin-4-ylpiperidin-1-yl)methanone —— C20H26N2O2
(5-Tert-butyl-3-methylfuran-2-yl)-(4-pyridin-4-ylpiperidin-1-yl)methanone
—— 5-(3-Fluorophenyl)-4-(6-methylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-1,2,4-triazol-3-one —— C20H16FN5O
5-(3-Fluorophenyl)-4-(6-methylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-1,2,4-triazol-3-one
—— [5-[(4-Chloropyrazol-1-yl)methyl]furan-2-yl]-(4-pyridin-4-ylpiperidin-1-yl)methanone —— C19H19ClN4O2
[5-[(4-Chloropyrazol-1-yl)methyl]furan-2-yl]-(4-pyridin-4-ylpiperidin-1-yl)methanone
—— (5S,7R)-N-[1-(1,3-benzodioxol-5-yl)cyclopentyl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H23F3N4O3
(5S,7R)-N-[1-(1,3-benzodioxol-5-yl)cyclopentyl]-5-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-(2-methylphenyl)-1,3,4-thiadiazol-2-amine —— C19H17N5O2S2
5-[[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-(2-methylphenyl)-1,3,4-thiadiazol-2-amine
—— (5-Cyclopropyl-2-methylfuran-3-yl)-(4-pyridin-4-ylpiperidin-1-yl)methanone —— C19H22N2O2
(5-Cyclopropyl-2-methylfuran-3-yl)-(4-pyridin-4-ylpiperidin-1-yl)methanone
—— 5-bromo-N'-[(2S)-2-(2,3-dimethylphenoxy)propanoyl]pyridine-3-carbohydrazide —— C17H18BrN3O3
5-bromo-N'-[(2S)-2-(2,3-dimethylphenoxy)propanoyl]pyridine-3-carbohydrazide
—— 5-bromo-N'-[(2R)-2-(2,3-dimethylphenoxy)propanoyl]pyridine-3-carbohydrazide —— C17H18BrN3O3
5-bromo-N'-[(2R)-2-(2,3-dimethylphenoxy)propanoyl]pyridine-3-carbohydrazide
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2,5-dimethyl-1-phenylpyrrole-3-carboxylate —— C22H21N3O4
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2,5-dimethyl-1-phenylpyrrole-3-carboxylate
—— 5-(2-Methylfuran-3-yl)-3-(quinolin-2-ylmethyl)-1,3,4-oxadiazol-2-one —— C17H13N3O3
5-(2-Methylfuran-3-yl)-3-(quinolin-2-ylmethyl)-1,3,4-oxadiazol-2-one
—— 5-(3-Fluorophenyl)-4-pyridin-4-yl-2-(pyridin-3-ylmethyl)-1,2,4-triazol-3-one —— C19H14FN5O
5-(3-Fluorophenyl)-4-pyridin-4-yl-2-(pyridin-3-ylmethyl)-1,2,4-triazol-3-one
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(2-methoxyphenyl)cyclopentyl]pentanamide —— C22H31N3O3S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(2-methoxyphenyl)cyclopentyl]pentanamide
—— 5-ethoxy-N-[1-(4-fluorophenyl)cyclopentyl]furan-2-carboxamide —— C18H20FNO3
5-ethoxy-N-[1-(4-fluorophenyl)cyclopentyl]furan-2-carboxamide
—— 5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(4-fluorophenyl)cyclopentyl]pentanamide —— C21H28FN3O2S
5-[(3aR,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(4-fluorophenyl)cyclopentyl]pentanamide
—— 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(1,3-benzodioxol-5-yl)cyclopentyl]pentanamide —— C22H29N3O4S
5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(1,3-benzodioxol-5-yl)cyclopentyl]pentanamide
—— 5-bromo-N'-[(2S)-2-(2,3-dimethylphenoxy)propanoyl]-2-fluorobenzohydrazide —— C18H18BrFN2O3
5-bromo-N'-[(2S)-2-(2,3-dimethylphenoxy)propanoyl]-2-fluorobenzohydrazide
—— 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(4-fluorophenyl)cyclopentyl]pentanamide —— C21H28FN3O2S
5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(4-fluorophenyl)cyclopentyl]pentanamide
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 4-(dimethylamino)benzoate —— C19H17ClN2O3
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 4-(dimethylamino)benzoate
—— 5-(5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3,4-oxadiazol-2-one —— C15H17N3O3S
5-(5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3,4-oxadiazol-2-one
—— 5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(2-methoxyphenyl)cyclopentyl]pentanamide —— C22H31N3O3S
5-[(3aR,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[1-(2-methoxyphenyl)cyclopentyl]pentanamide
—— 5-Isoquinolin-1-yl-3-(pyridin-4-ylmethyl)-1,3,4-oxadiazol-2-one —— C17H12N4O2
5-Isoquinolin-1-yl-3-(pyridin-4-ylmethyl)-1,3,4-oxadiazol-2-one
—— 5-(4-methoxyphenyl)-4-[(3S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-2-amine —— C20H24N6O3S
5-(4-methoxyphenyl)-4-[(3S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-2-amine
—— 5-[(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22ClN5O2
5-[(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22ClN5O2
5-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-(4-chlorophenyl)-4-[(3S)-1-(oxan-4-yl)piperidin-3-yl]pyrimidin-2-amine —— C20H25ClN4O
5-(4-chlorophenyl)-4-[(3S)-1-(oxan-4-yl)piperidin-3-yl]pyrimidin-2-amine
—— 5-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-[(3R)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(3R)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-(4-methoxyphenyl)-4-[(3R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-2-amine —— C20H24N6O3S
5-(4-methoxyphenyl)-4-[(3R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-2-amine
—— 5-[(3S)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(3S)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-(3-fluorophenyl)-4-[(3R)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C24H24FN5
5-(3-fluorophenyl)-4-[(3R)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-fluorophenyl)-N-(5-pyridin-3-yl-1,3-thiazol-2-yl)-1,3-oxazole-4-carboxamide —— C18H11FN4O2S
5-(4-fluorophenyl)-N-(5-pyridin-3-yl-1,3-thiazol-2-yl)-1,3-oxazole-4-carboxamide
—— 5-(3-fluorophenyl)-4-[(3S)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C24H24FN5
5-(3-fluorophenyl)-4-[(3S)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-methoxyphenyl)sulfonyl-1-methyl-3-phenyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine —— C20H21N3O3S
5-(4-methoxyphenyl)sulfonyl-1-methyl-3-phenyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine
—— 5-(4-chlorophenyl)-4-[(3R)-1-(quinoxalin-6-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C24H23ClN6
5-(4-chlorophenyl)-4-[(3R)-1-(quinoxalin-6-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-fluorophenyl)-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H22FN5
5-(4-fluorophenyl)-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-methoxyphenyl)-4-[(3S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]pyrimidin-2-amine —— C23H28N6O
5-(4-methoxyphenyl)-4-[(3S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-methoxyphenyl)-4-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]pyrimidin-2-amine —— C23H28N6O
5-(4-methoxyphenyl)-4-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-methoxyphenyl)-4-[(3S)-1-(oxan-4-yl)piperidin-3-yl]pyrimidin-2-amine —— C21H28N4O2
5-(4-methoxyphenyl)-4-[(3S)-1-(oxan-4-yl)piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-chlorophenyl)-4-[(3S)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-3-yl]pyrimidin-2-amine —— C22H25ClN6
5-(4-chlorophenyl)-4-[(3S)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-chlorophenyl)-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H22ClN5
5-(4-chlorophenyl)-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-methoxyphenyl)-4-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]pyrimidin-2-amine —— C24H28N4O2
5-(4-methoxyphenyl)-4-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-chlorophenyl)-4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H22ClN5
5-(4-chlorophenyl)-4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 5-(3-fluorophenyl)-4-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]pyrimidin-2-amine —— C22H22F2N4
5-(3-fluorophenyl)-4-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]pyrimidin-2-amine
—— 5-(4-fluorophenyl)-4-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]pyrimidin-2-amine —— C22H22F2N4
5-(4-fluorophenyl)-4-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]pyrimidin-2-amine
—— 5-(3-fluorophenyl)-4-[(3R)-1-(4-fluorophenyl)sulfonylpiperidin-3-yl]pyrimidin-2-amine —— C21H20F2N4O2S
5-(3-fluorophenyl)-4-[(3R)-1-(4-fluorophenyl)sulfonylpiperidin-3-yl]pyrimidin-2-amine