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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-3-methyl-9-(3-methyl-1-benzothiophene-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22N2O3S
(5S)-3-methyl-9-(3-methyl-1-benzothiophene-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-5-(naphthalen-1-yloxymethyl)-N-(2-phenylethyl)-3-propan-2-yl-1,3-thiazolidin-2-imine —— C25H28N2OS
(5R)-5-(naphthalen-1-yloxymethyl)-N-(2-phenylethyl)-3-propan-2-yl-1,3-thiazolidin-2-imine
—— 5-(2-fluorophenyl)-N-[(4-sulfamoylphenyl)methyl]furan-2-carboxamide —— C18H15FN2O4S
5-(2-fluorophenyl)-N-[(4-sulfamoylphenyl)methyl]furan-2-carboxamide
—— (5R)-3-methyl-9-(3-pyridin-2-ylpropanoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H23N3O3
(5R)-3-methyl-9-(3-pyridin-2-ylpropanoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5-chloropyridin-2-yl)-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C21H25ClFN3O
(5-chloropyridin-2-yl)-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— (5S,10bS)-5-(4-methylphenyl)-2-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H19N3O
(5S,10bS)-5-(4-methylphenyl)-2-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(1S)-1-(benzylsulfamoylamino)ethyl]-1,3,4-thiadiazol-2-amine —— C11H15N5O2S2
5-[(1S)-1-(benzylsulfamoylamino)ethyl]-1,3,4-thiadiazol-2-amine
—— (5R)-9-[2-(2-phenylimidazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O3
(5R)-9-[2-(2-phenylimidazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R,7R)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H16BrFN4O
(5R,7R)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5R)-3-methyl-7-(7-oxo-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H14N4O4S
(5R)-3-methyl-7-(7-oxo-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-9-[2-(1,2,4-triazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C13H19N5O3
(5S)-3-methyl-9-[2-(1,2,4-triazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H21N3O5
(5R)-9-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[(2,3-difluorophenyl)methyl]-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H21F2N3O3
(5S)-7-[(2,3-difluorophenyl)methyl]-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-N-(3-methoxyphenyl)-5-(naphthalen-1-yloxymethyl)-3-propan-2-yl-1,3-thiazolidin-2-imine —— C24H26N2O2S
(5S)-N-(3-methoxyphenyl)-5-(naphthalen-1-yloxymethyl)-3-propan-2-yl-1,3-thiazolidin-2-imine
—— (5R)-7-[(2,3-difluorophenyl)methyl]-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H21F2N3O3
(5R)-7-[(2,3-difluorophenyl)methyl]-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(2-phenylimidazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O3
(5S)-9-[2-(2-phenylimidazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-9-[(4-methylsulfonylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N2O4S
(5R)-3-methyl-9-[(4-methylsulfonylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-5-(4-nitrophenyl)-N-(2-phenylethyl)-4,5-dihydro-1,3-thiazol-2-amine —— C17H17N3O2S
(5R)-5-(4-nitrophenyl)-N-(2-phenylethyl)-4,5-dihydro-1,3-thiazol-2-amine
—— (5R,7R)-7-(1,3-benzodioxol-5-yl)-5-(4-bromophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H15BrN4O2
(5R,7R)-7-(1,3-benzodioxol-5-yl)-5-(4-bromophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5S,7S)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H16BrFN4O
(5S,7S)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5R,10bS)-5-(4-methylphenyl)-2-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H19N3O
(5R,10bS)-5-(4-methylphenyl)-2-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,7R)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H16BrFN4O
(5S,7R)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5-chloropyridin-2-yl)-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C21H25ClFN3O
(5-chloropyridin-2-yl)-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— (5S)-9-[(2-pyrazol-1-ylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H23N3O2
(5S)-9-[(2-pyrazol-1-ylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C11H20N2O2
(5R)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,7S)-7-(2,3-dichlorophenyl)-5-thiophen-2-yl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C15H12Cl2N4S
(5S,7S)-7-(2,3-dichlorophenyl)-5-thiophen-2-yl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyridin-2-one —— C20H23N3O2
5-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyridin-2-one
—— 5-chloro-N'-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfonyl)-2-hydroxybenzohydrazide —— C16H15ClN2O6S
5-chloro-N'-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfonyl)-2-hydroxybenzohydrazide
—— (5S)-3-methyl-7-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H19N3O3S
(5S)-3-methyl-7-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R,7S)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H16BrFN4O
(5R,7S)-7-(5-bromo-2-methoxyphenyl)-5-(4-fluorophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(dimethylamino)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O4
(5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(dimethylamino)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[4-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-6-oxopyridazin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide —— C17H23N5O3
5-[[4-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-6-oxopyridazin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide
—— (5R)-9-[[3-(5-methylfuran-2-yl)phenyl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H24N2O3
(5R)-9-[[3-(5-methylfuran-2-yl)phenyl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C11H20N2O2
(5S)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[[3-(5-methylfuran-2-yl)phenyl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H24N2O3
(5S)-9-[[3-(5-methylfuran-2-yl)phenyl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3S)-3-(3-propan-2-yloxybenzoyl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H23N3O4
5-[(3S)-3-(3-propan-2-yloxybenzoyl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-[4-(4-Methoxyphenyl)piperazin-1-yl]-2-methyl-[1,2]oxazolo[2,3-a]pyrimidin-7-one —— C18H20N4O3
5-[4-(4-Methoxyphenyl)piperazin-1-yl]-2-methyl-[1,2]oxazolo[2,3-a]pyrimidin-7-one
—— 5-[(3R)-3-(3-propan-2-yloxybenzoyl)piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H23N3O4
5-[(3R)-3-(3-propan-2-yloxybenzoyl)piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-chloro-2-(1H-indol-3-ylmethylsulfanyl)-1,3-benzothiazole —— C16H11ClN2S2
5-chloro-2-(1H-indol-3-ylmethylsulfanyl)-1,3-benzothiazole
—— 5-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyridin-2-one —— C20H23N3O2
5-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyridin-2-one
—— (5S)-3-methyl-9-[(4-methylsulfonylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N2O4S
(5S)-3-methyl-9-[(4-methylsulfonylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[3-(3-oxo-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H21N3O5
(5R)-9-[3-(3-oxo-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[3-(3-oxo-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H21N3O5
(5S)-9-[3-(3-oxo-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-7-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H19N3O3S
(5R)-3-methyl-7-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-5-(naphthalen-1-yloxymethyl)-N-(2-phenylethyl)-3-propan-2-yl-1,3-thiazolidin-2-imine —— C25H28N2OS
(5S)-5-(naphthalen-1-yloxymethyl)-N-(2-phenylethyl)-3-propan-2-yl-1,3-thiazolidin-2-imine
—— 5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C32H56N6O9S2
5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aR,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— 5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide —— C32H56N6O9S2
5-[(3aS,4S,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[2-[2-[2-[2-[2-[2-[5-[(3aS,4R,6aS)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]pentanamide
—— (5R)-N-cyclohexyl-5-(4-nitrophenyl)-4,5-dihydro-1,3-thiazol-2-amine —— C15H19N3O2S
(5R)-N-cyclohexyl-5-(4-nitrophenyl)-4,5-dihydro-1,3-thiazol-2-amine
—— (5E)-5-[[benzyl(methyl)amino]methylidene]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C16H19N3O3S
(5E)-5-[[benzyl(methyl)amino]methylidene]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(dimethylamino)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O4
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(dimethylamino)acetyl]-2,7-diazaspiro[4.5]decan-6-one