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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H16F4N2O2
(5R)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(3S)-1-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C17H26ClN5O2
5-[(3S)-1-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— (5R)-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H23N5O3
(5R)-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-methyl-2-(1H-pyrrolo[2,3-b]pyridin-6-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H20N4O
(5R)-7-methyl-2-(1H-pyrrolo[2,3-b]pyridin-6-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H16F4N2O2
(5S)-7-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-9-[(3-propan-2-ylimidazol-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H24N4O2
(5S)-3-methyl-9-[(3-propan-2-ylimidazol-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C13H22N2O
(5R)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(1-benzylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22N4O3
(5S)-9-(1-benzylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H23N5O3
(5S)-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(cyclopropylmethyl)-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C16H24N4
(5S)-9-(cyclopropylmethyl)-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— (5R)-9-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H27N5O2
(5R)-9-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[(3-pyridin-2-ylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H23N3O2
(5R)-9-[(3-pyridin-2-ylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-7-[3-(6-oxo-1H-pyridazin-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H18N4O4
(5S)-3-methyl-7-[3-(6-oxo-1H-pyridazin-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methoxy-2-[[(2R)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1H-pyridin-4-one —— C20H26N2O2
5-methoxy-2-[[(2R)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1H-pyridin-4-one
—— (5R)-9-(cyclopropylmethyl)-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C16H24N4
(5R)-9-(cyclopropylmethyl)-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-methoxy-2-[[(2S)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1H-pyridin-4-one —— C20H26N2O2
5-methoxy-2-[[(2S)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1H-pyridin-4-one
—— 5-[(3R)-1-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C17H26ClN5O2
5-[(3R)-1-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— (5R)-3-methyl-7-[3-(6-oxo-1H-pyridazin-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H18N4O4
(5R)-3-methyl-7-[3-(6-oxo-1H-pyridazin-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C13H19N3O2S
(5S)-9-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H21N3O3S
(5S)-9-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H21N3O3S
(5R)-9-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(4S)-4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C17H21N3O4
5-[(4S)-4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— 5-[[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole —— C20H28N4OS
5-[[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole
—— (5S)-9-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H25N3O5
(5S)-9-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(5-fluoropyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H16FN3O3
(5S)-9-(5-fluoropyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-(2-methylsulfanylpyrimidin-4-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H20N4O2S
(5S)-3-methyl-9-(2-methylsulfanylpyrimidin-4-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5R)-3-methyl-9-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole —— C20H28N4OS
5-[[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyrrolidin-1-yl-1,3-thiazole
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,6-dichlorophenyl)acetate —— C15H10Cl2N2O4
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,6-dichlorophenyl)acetate
—— 5-[(4R)-4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C17H21N3O4
5-[(4R)-4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— (5S)-3-methyl-9-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5S)-3-methyl-9-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— [(5R)-9-(2-methoxyethyl)-2,9-diazaspiro[4.5]decan-2-yl]-quinoxalin-5-ylmethanone —— C20H26N4O2
[(5R)-9-(2-methoxyethyl)-2,9-diazaspiro[4.5]decan-2-yl]-quinoxalin-5-ylmethanone
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-(2,6-dichlorophenyl)acetate —— C18H13Cl2NO3
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-(2,6-dichlorophenyl)acetate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 3,4,5-trimethoxybenzoate —— C20H19NO6
(5-Phenyl-1,3-oxazol-2-yl)methyl 3,4,5-trimethoxybenzoate
—— 5-[[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H21F3N4O2
5-[[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5S)-3-methyl-9-[5-(6-oxocyclohexa-2,4-dien-1-ylidene)-1,2-dihydropyrazole-3-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22N4O4
(5S)-3-methyl-9-[5-(6-oxocyclohexa-2,4-dien-1-ylidene)-1,2-dihydropyrazole-3-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C18H21F3N4O2
5-[[(3S)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5-Fluoro-2-methoxyphenyl)methyl 3,4,5-trimethoxybenzoate —— C18H19FO6
(5-Fluoro-2-methoxyphenyl)methyl 3,4,5-trimethoxybenzoate
—— (5R)-9-(5-fluoropyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H16FN3O3
(5R)-9-(5-fluoropyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-7-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H21N5O3
(5S)-3-methyl-7-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H30N4O3
(5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C20H24F3N5O2
5-[(3S)-3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— (5S)-3-methyl-9-(2-pyridin-2-ylethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H23N3O2
(5S)-3-methyl-9-(2-pyridin-2-ylethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-propan-2-yl-N-[(2S)-2-pyrrolidin-1-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H25N5
5-propan-2-yl-N-[(2S)-2-pyrrolidin-1-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(2S)-2-(cyclopropylcarbamoyl)piperazine-1-carbonyl]-4-oxo-1-propan-2-ylpyridine-3-carboxylic acid —— C18H24N4O5
5-[(2S)-2-(cyclopropylcarbamoyl)piperazine-1-carbonyl]-4-oxo-1-propan-2-ylpyridine-3-carboxylic acid
—— (5R)-3-methyl-7-[2-(2-methylphenoxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H20N2O4
(5R)-3-methyl-7-[2-(2-methylphenoxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[(2-fluoro-3-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H22FNO2
(5S)-9-[(2-fluoro-3-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C23H27N3O4
(5S)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-methyl-7-(2-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O3S
(5R)-3-methyl-7-(2-methyl-5-thiophen-2-ylpyrazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-7-[3-(5-methyltetrazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H20N6O2
(5S)-3-methyl-7-[3-(5-methyltetrazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one