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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(5R)-9-[(4-fluorophenyl)methyl]-2,9-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-1H-pyridin-4-one —— C22H26FN3O2
5-[(5R)-9-[(4-fluorophenyl)methyl]-2,9-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-1H-pyridin-4-one
—— 5-ethyl-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H24N6
5-ethyl-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(5S)-9-[(4-fluorophenyl)methyl]-2,9-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-1H-pyridin-4-one —— C22H26FN3O2
5-[(5S)-9-[(4-fluorophenyl)methyl]-2,9-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5S)-9-[(6,8-dimethyl-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H25N3O3
(5S)-9-[(6,8-dimethyl-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C23H27N3O4
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H19N5O3
(5S)-7-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[(6-chloro-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H19ClN2O4
(5S)-9-[(6-chloro-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[(6,8-dimethyl-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H25N3O3
(5R)-9-[(6,8-dimethyl-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone —— C17H21ClN2O4
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone
—— (5R)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O
(5R)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(5-propyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H19N3O4
(5S)-9-(5-propyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[(3-methoxyphenyl)methyl]-2-(2-methylsulfanylpyrimidin-4-yl)-2,9-diazaspiro[4.5]decane —— C21H28N4OS
(5S)-9-[(3-methoxyphenyl)methyl]-2-(2-methylsulfanylpyrimidin-4-yl)-2,9-diazaspiro[4.5]decane
—— 5-[(1S)-1-[2-(2-butyl-1H-imidazol-5-yl)imidazol-1-yl]ethyl]-2-methylpyridine —— C18H23N5
5-[(1S)-1-[2-(2-butyl-1H-imidazol-5-yl)imidazol-1-yl]ethyl]-2-methylpyridine
—— (5-chloropyridin-2-yl)-[4-[(3R)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone —— C16H22ClN3O2
(5-chloropyridin-2-yl)-[4-[(3R)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone
—— (5R)-3-methyl-9-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H24N4O3
(5R)-3-methyl-9-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[2-(hydroxymethyl)-3H-benzimidazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O4
(5S)-9-[2-(hydroxymethyl)-3H-benzimidazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H20N2O4
(5S)-7-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5-chloropyridin-2-yl)-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone —— C16H22ClN3O2
(5-chloropyridin-2-yl)-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone
—— (5S)-3-methyl-7-[2-(2-oxo-1,3-benzoxazol-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H17N3O5
(5S)-3-methyl-7-[2-(2-oxo-1,3-benzoxazol-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[(3-methoxyphenyl)methyl]-2-(2-methylsulfanylpyrimidin-4-yl)-2,9-diazaspiro[4.5]decane —— C21H28N4OS
(5R)-9-[(3-methoxyphenyl)methyl]-2-(2-methylsulfanylpyrimidin-4-yl)-2,9-diazaspiro[4.5]decane
—— 5-[[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C20H18N4OS
5-[[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— (5R)-9-[2-[(4-methylphenyl)methyl]benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C23H26N2O3
(5R)-9-[2-[(4-methylphenyl)methyl]benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C20H18N4OS
5-[[(2S)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— 5-[[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C21H35N5O
5-[[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (5S)-7-[2-[(3,5-dimethylphenyl)methylsulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H24N2O3S
(5S)-7-[2-[(3,5-dimethylphenyl)methylsulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H19N5O3
(5R)-7-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-(2,3-Dihydro-1,4-benzodioxin-6-yl)-1,2-oxazole-3-carboxylate —— C12H8NO5-
5-(2,3-Dihydro-1,4-benzodioxin-6-yl)-1,2-oxazole-3-carboxylate
—— (5S)-9-[2-(3-acetylindol-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H25N3O4
(5S)-9-[2-(3-acetylindol-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-7-(3-methylsulfonylbenzoyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H18N2O5S
(5R)-3-methyl-7-(3-methylsulfonylbenzoyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-2-methylsulfonyl-9-[(4-propan-2-ylphenyl)methyl]-2,9-diazaspiro[4.5]decane —— C19H30N2O2S
(5R)-2-methylsulfonyl-9-[(4-propan-2-ylphenyl)methyl]-2,9-diazaspiro[4.5]decane
—— 5-[[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine —— C21H28N6
5-[[(3R)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine
—— 5-[[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-N-propylpyrimidin-2-amine —— C20H24N6O
5-[[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl]-N-propylpyrimidin-2-amine
—— 5-[(1R)-1-[2-(2-butyl-1H-imidazol-5-yl)imidazol-1-yl]ethyl]-2-methylpyridine —— C18H23N5
5-[(1R)-1-[2-(2-butyl-1H-imidazol-5-yl)imidazol-1-yl]ethyl]-2-methylpyridine
—— (5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone —— C17H21ClN2O4
(5-chloro-7-methoxy-1-benzofuran-2-yl)-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl]methanone
—— 5-[[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine —— C21H28N6
5-[[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine
—— 5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]pyridazin-3-one —— C15H22N6O2
5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]pyridazin-3-one
—— (5R)-9-(5-propyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H19N3O4
(5R)-9-(5-propyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(2H-benzotriazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H17N5O3
(5R)-9-(2H-benzotriazole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[2-oxo-2-[(3S)-3-(4-propan-2-ylanilino)piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione —— C20H26N4O3
5-[2-oxo-2-[(3S)-3-(4-propan-2-ylanilino)piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione
—— 5-[2-oxo-2-[(3R)-3-(4-propan-2-ylanilino)piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione —— C20H26N4O3
5-[2-oxo-2-[(3R)-3-(4-propan-2-ylanilino)piperidin-1-yl]ethyl]-1H-pyrimidine-2,4-dione
—— (5R)-7-[(6-chloro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H18ClN3O3
(5R)-7-[(6-chloro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-[2-[(3,5-dimethylphenyl)methylsulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H24N2O3S
(5R)-7-[2-[(3,5-dimethylphenyl)methylsulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(naphthalen-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C20H23NO2
(5S)-9-(naphthalen-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-9-[2-(hydroxymethyl)-3H-benzimidazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O4
(5R)-9-[2-(hydroxymethyl)-3H-benzimidazole-5-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[2-(3-acetylindol-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H25N3O4
(5R)-9-[2-(3-acetylindol-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H28N4O3
(5R)-9-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[3-(4-methylpyrazol-1-yl)propyl]pyridazin-3-one —— C16H24N6O
5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[3-(4-methylpyrazol-1-yl)propyl]pyridazin-3-one
—— 5-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-2-[[(2S)-2-methylpyrrolidin-1-yl]methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine —— C21H28N6
5-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-2-[[(2S)-2-methylpyrrolidin-1-yl]methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine
—— (5S)-9-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H28N4O3
(5S)-9-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-7-(3-phenoxypropanoyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H20N2O4
(5R)-3-methyl-7-(3-phenoxypropanoyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one