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—— [5-Ethyl-1-(4-fluorophenyl)-3-propylpyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C20H28FN4O+
[5-Ethyl-1-(4-fluorophenyl)-3-propylpyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5R)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H24N4O3
(5R)-N-[(2R)-1-[2-(dimethylamino)ethylamino]-1-oxopropan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-N-[2-(furan-2-ylmethylamino)-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H19N3O4
(5R)-N-[2-(furan-2-ylmethylamino)-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[3-oxo-3-[[(2S)-oxolan-2-yl]methylamino]propyl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H23N3O4
(5S)-N-[3-oxo-3-[[(2S)-oxolan-2-yl]methylamino]propyl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H24N4O3
(5S)-N-[2-[2-(dimethylamino)ethylamino]-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[2-(4-fluoroanilino)-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H18FN3O3
(5S)-N-[2-(4-fluoroanilino)-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [5-Ethyl-1-(3-fluorophenyl)-3-(2-methylpropyl)pyrazol-4-yl]-pyrrolidin-1-ylmethanone —— C20H26FN3O
[5-Ethyl-1-(3-fluorophenyl)-3-(2-methylpropyl)pyrazol-4-yl]-pyrrolidin-1-ylmethanone
—— (5S)-N-[(2S)-1-oxo-1-(propylamino)propan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H21N3O3
(5S)-N-[(2S)-1-oxo-1-(propylamino)propan-2-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-3-(4-methylphenyl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H21N3O3
(5S)-3-(4-methylphenyl)-N-[2-oxo-2-(propan-2-ylamino)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-cyclopropyl-7,8-dimethyl-N-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C21H29N3O2
(5S)-N-cyclopropyl-7,8-dimethyl-N-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— [(5R)-3-(3,4-dichlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium —— C18H16Cl2F3N2O+
[(5R)-3-(3,4-dichlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium
—— [5-Ethyl-1-(3-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone —— C22H33N4O+
[5-Ethyl-1-(3-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-(4-methylpiperazin-4-ium-1-yl)methanone
—— (5-Ethyl-1-methyl-3-propylpyrazol-4-yl)-(4-ethylpiperazin-4-ium-1-yl)methanone —— C16H29N4O+
(5-Ethyl-1-methyl-3-propylpyrazol-4-yl)-(4-ethylpiperazin-4-ium-1-yl)methanone
—— (5S)-N-(2-methoxyethyl)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H18N2O3
(5S)-N-(2-methoxyethyl)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-methyl-1-phenyl-N-propan-2-yl-3-propylpyrazole-4-carboxamide —— C17H23N3O
5-methyl-1-phenyl-N-propan-2-yl-3-propylpyrazole-4-carboxamide
—— 5-ethyl-1-methyl-N-[[(2R)-oxolan-2-yl]methyl]-3-propylpyrazole-4-carboxamide —— C15H25N3O2
5-ethyl-1-methyl-N-[[(2R)-oxolan-2-yl]methyl]-3-propylpyrazole-4-carboxamide
—— [5-Ethyl-1-(3-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone —— C22H32N4O
[5-Ethyl-1-(3-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-(4-methylpiperazin-1-yl)methanone
—— (5R)-N-cyclopropyl-7,8-dimethyl-N-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C21H29N3O2
(5R)-N-cyclopropyl-7,8-dimethyl-N-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— [5-Methyl-1-(3-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-morpholin-4-ylmethanone —— C20H27N3O2
[5-Methyl-1-(3-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-morpholin-4-ylmethanone
—— [(5S)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium —— C19H20F3N2O+
[(5S)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium
—— (5R)-N-(2-methoxyethyl)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H18N2O3
(5R)-N-(2-methoxyethyl)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5-Ethyl-1-methyl-3-propylpyrazol-4-yl)-pyrrolidin-1-ylmethanone —— C14H23N3O
(5-Ethyl-1-methyl-3-propylpyrazol-4-yl)-pyrrolidin-1-ylmethanone
—— (5S)-N-[2-(cyclopropylamino)-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H19N3O3
(5S)-N-[2-(cyclopropylamino)-2-oxoethyl]-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5-Ethyl-1-methyl-3-propylpyrazol-4-yl)-morpholin-4-ylmethanone —— C14H23N3O2
(5-Ethyl-1-methyl-3-propylpyrazol-4-yl)-morpholin-4-ylmethanone
—— 5-ethyl-1-methyl-N-[[(2S)-oxolan-2-yl]methyl]-3-propylpyrazole-4-carboxamide —— C15H25N3O2
5-ethyl-1-methyl-N-[[(2S)-oxolan-2-yl]methyl]-3-propylpyrazole-4-carboxamide
—— [(5R)-3-(3,4-dichlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[4-(trifluoromethyl)phenyl]methyl]azanium —— C18H16Cl2F3N2O+
[(5R)-3-(3,4-dichlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[4-(trifluoromethyl)phenyl]methyl]azanium
—— [(5S)-3-(1,3-benzodioxol-5-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[(3-chlorophenyl)methyl]azanium —— C18H18ClN2O3+
[(5S)-3-(1,3-benzodioxol-5-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[(3-chlorophenyl)methyl]azanium
—— 5-methyl-N-[(1R)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-4-carboxamide —— C17H17F3N6O2
5-methyl-N-[(1R)-1-(5-methyl-1,2,4-oxadiazol-3-yl)propyl]-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-4-carboxamide
—— 5-[[4-[Cyclohexyl(methyl)amino]-6-methylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate —— C18H22N3O3S-
5-[[4-[Cyclohexyl(methyl)amino]-6-methylpyrimidin-2-yl]sulfanylmethyl]furan-2-carboxylate
—— 5-chloro-N-[(2R)-2-(4-chlorophenyl)-2-(dimethylamino)ethyl]-2-piperidin-1-ylpyrimidine-4-carboxamide —— C20H25Cl2N5O
5-chloro-N-[(2R)-2-(4-chlorophenyl)-2-(dimethylamino)ethyl]-2-piperidin-1-ylpyrimidine-4-carboxamide
—— (5R)-3-(4-methylphenyl)-N-[2-oxo-2-(propylamino)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H21N3O3
(5R)-3-(4-methylphenyl)-N-[2-oxo-2-(propylamino)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[(2R)-2-methyl-4-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydroquinoxalin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C21H28N6O2
5-[[(2R)-2-methyl-4-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydroquinoxalin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— [(5R)-3-(1,3-benzodioxol-5-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[(3-chlorophenyl)methyl]azanium —— C18H18ClN2O3+
[(5R)-3-(1,3-benzodioxol-5-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[(3-chlorophenyl)methyl]azanium
—— 5,6-dimethyl-2-[[(2R)-1-[(2R)-2-(1-methylpyrrol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C22H28N4O2S2
5,6-dimethyl-2-[[(2R)-1-[(2R)-2-(1-methylpyrrol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5S)-N-[(2S)-1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H22FN3O3
(5S)-N-[(2S)-1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-N-[2-(dimethylamino)ethyl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H19N3O2
(5R)-N-[2-(dimethylamino)ethyl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-N-[(2R)-1-(cyclopropylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C22H22FN3O3
(5R)-N-[(2R)-1-(cyclopropylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [(5R)-3-(1,3-benzodioxol-5-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[(2,4-difluorophenyl)methyl]azanium —— C18H17F2N2O3+
[(5R)-3-(1,3-benzodioxol-5-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[(2,4-difluorophenyl)methyl]azanium
—— 5,6-dimethyl-2-[[(2R)-1-[(2S)-2-(1-methylpyrrol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C22H28N4O2S2
5,6-dimethyl-2-[[(2R)-1-[(2S)-2-(1-methylpyrrol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— [(5R)-3-phenyl-4,5-dihydro-1,2-oxazol-5-yl]-pyrrolidin-1-ylmethanone —— C14H16N2O2
[(5R)-3-phenyl-4,5-dihydro-1,2-oxazol-5-yl]-pyrrolidin-1-ylmethanone
—— (5S)-N-[(2S)-1-(cyclopropylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C22H22FN3O3
(5S)-N-[(2S)-1-(cyclopropylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5S)-N-[2-(dimethylamino)ethyl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C14H19N3O2
(5S)-N-[2-(dimethylamino)ethyl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-chloro-N-[(2S)-2-(4-chlorophenyl)-2-(dimethylamino)ethyl]-2-piperidin-1-ylpyrimidine-4-carboxamide —— C20H25Cl2N5O
5-chloro-N-[(2S)-2-(4-chlorophenyl)-2-(dimethylamino)ethyl]-2-piperidin-1-ylpyrimidine-4-carboxamide
—— 5,6-dimethyl-2-[[(2S)-1-[(2R)-2-(1-methylpyrrol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C22H28N4O2S2
5,6-dimethyl-2-[[(2S)-1-[(2R)-2-(1-methylpyrrol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— [(5S)-3-(3,4-dichlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium —— C18H16Cl2F3N2O+
[(5S)-3-(3,4-dichlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium
—— [(5R)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium —— C19H20F3N2O+
[(5R)-3-(4-methylphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl-[[3-(trifluoromethyl)phenyl]methyl]azanium
—— (5S)-N-[(2R)-1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H22FN3O3
(5S)-N-[(2R)-1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-N-[(2S)-1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H22FN3O3
(5R)-N-[(2S)-1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[[(2S)-2-methyl-4-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydroquinoxalin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole —— C21H28N6O2
5-[[(2S)-2-methyl-4-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydroquinoxalin-1-yl]methyl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5S)-N-[(2R)-1-(cyclopropylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C22H22FN3O3
(5S)-N-[(2R)-1-(cyclopropylamino)-1-oxo-3-phenylpropan-2-yl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide