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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-3-methyl-9-[2-(2-methylphenyl)sulfanylacetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H22N2O3S
(5R)-3-methyl-9-[2-(2-methylphenyl)sulfanylacetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-chloro-3-methyl-1-phenyl-N-(2,3,5,6-tetrafluorophenyl)pyrazole-4-carboxamide —— C17H10ClF4N3O
5-chloro-3-methyl-1-phenyl-N-(2,3,5,6-tetrafluorophenyl)pyrazole-4-carboxamide
—— (5S)-3-methyl-7-(1-oxo-3,4-dihydro-2H-[1]benzothiolo[2,3-c]pyridine-6-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C19H19N3O4S
(5S)-3-methyl-7-(1-oxo-3,4-dihydro-2H-[1]benzothiolo[2,3-c]pyridine-6-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[(4-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C19H23FN4
(5R)-9-[(4-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— (5R)-7-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O3S
(5R)-7-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[(4-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C19H23FN4
(5S)-9-[(4-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— (5S)-9-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C12H17N5O3S
(5S)-9-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[2-[(3R)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C19H23N5O
5-[[2-[(3R)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— (5S)-9-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H24N4O3
(5S)-9-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(1-phenyltetrazol-5-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H18N6O2
(5R)-9-(1-phenyltetrazol-5-yl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-7-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O3S
(5S)-7-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-N-(1-benzofuran-5-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C17H19N3O4
(5S)-N-(1-benzofuran-5-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— (5R)-9-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C12H17N5O3S
(5R)-9-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[2-[(3S)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole —— C19H23N5O
5-[[2-[(3S)-1-ethylpiperidin-3-yl]imidazol-1-yl]methyl]-3-pyridin-2-yl-1,2-oxazole
—— (5S)-3-methyl-9-(1-methylimidazol-4-yl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C13H20N4O4S
(5S)-3-methyl-9-(1-methylimidazol-4-yl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-(Phenoxymethyl)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene —— C8H7N4O-
5-(Phenoxymethyl)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene
—— (5S)-2-(1,3-benzoxazol-2-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H22FN3O2
(5S)-2-(1,3-benzoxazol-2-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-methyl-9-(1-methylimidazol-4-yl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C13H20N4O4S
(5R)-3-methyl-9-(1-methylimidazol-4-yl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5Z)-5-[(4-fluorophenyl)methylidene]-3-(furan-2-ylmethyl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylimidazol-4-one —— C21H20FN3O3S
(5Z)-5-[(4-fluorophenyl)methylidene]-3-(furan-2-ylmethyl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanylimidazol-4-one
—— [(5S,7R)-3-chloro-1-adamantyl]-(1-methyl-3,4-dihydro-2H-[1,4]diazepino[2,3-b]quinoxalin-5-yl)methanone —— C23H27ClN4O
[(5S,7R)-3-chloro-1-adamantyl]-(1-methyl-3,4-dihydro-2H-[1,4]diazepino[2,3-b]quinoxalin-5-yl)methanone
—— (5-propyl-1,2-oxazol-3-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C21H27N3O2
(5-propyl-1,2-oxazol-3-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5R)-2-(1,3-benzoxazol-2-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H22FN3O2
(5R)-2-(1,3-benzoxazol-2-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-5-oxopentanamide —— C20H30FN3O2
5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-5-oxopentanamide
—— 5-(2,5-dichlorothiophen-3-yl)-2,3-dihydro-1H-pyrazin-6-one —— C8H6Cl2N2OS
5-(2,5-dichlorothiophen-3-yl)-2,3-dihydro-1H-pyrazin-6-one
—— (5S)-9-[[3-fluoro-2-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H19F4NO2
(5S)-9-[[3-fluoro-2-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5E)-5-(furan-2-ylmethylidene)-2-sulfanylidene-3-[4-(trifluoromethoxy)phenyl]imidazolidin-4-one —— C15H9F3N2O3S
(5E)-5-(furan-2-ylmethylidene)-2-sulfanylidene-3-[4-(trifluoromethoxy)phenyl]imidazolidin-4-one
—— (5S)-9-(4-pyrazol-1-ylphenyl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20N4O4S
(5S)-9-(4-pyrazol-1-ylphenyl)sulfonyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-N-(1-benzofuran-5-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C17H19N3O4
(5R)-N-(1-benzofuran-5-yl)-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— (5S)-9-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H21N3O3
(5S)-9-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[[5-(1,5-dimethylpyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H21N5O3
(5S)-9-[[5-(1,5-dimethylpyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-Methyl-12-phenyl-10-(trifluoromethyl)-2,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4,10,12-pentaen-8-one —— C17H11F3N4O
5-Methyl-12-phenyl-10-(trifluoromethyl)-2,6,7,13-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4,10,12-pentaen-8-one
—— 5-cyano-2-methyl-6-oxo-N-[(3R)-1-(2-phenylethyl)piperidin-3-yl]-1H-pyridine-3-carboxamide —— C21H24N4O2
5-cyano-2-methyl-6-oxo-N-[(3R)-1-(2-phenylethyl)piperidin-3-yl]-1H-pyridine-3-carboxamide
—— (5R)-2-(5,6-dimethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H33N5O2
(5R)-2-(5,6-dimethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(5-fluoro-2-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H22FNO2
(5S)-9-[(5-fluoro-2-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(3R)-3-(3,4-dihydro-1H-isoquinolin-2-yl)piperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one —— C20H23N3O3
5-[(3R)-3-(3,4-dihydro-1H-isoquinolin-2-yl)piperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one
—— (5R)-9-[(5-fluoro-2-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H22FNO2
(5R)-9-[(5-fluoro-2-methylphenyl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[(3S)-3-(3,4-dihydro-1H-isoquinolin-2-yl)piperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one —— C20H23N3O3
5-[(3S)-3-(3,4-dihydro-1H-isoquinolin-2-yl)piperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one
—— (5R)-3-methyl-9-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H21N3O4
(5R)-3-methyl-9-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[2-(2-ethoxyphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H27NO4
(5S)-9-[2-(2-ethoxyphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-2-(5,6-dimethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H33N5O2
(5S)-2-(5,6-dimethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[[3-fluoro-2-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H19F4NO2
(5R)-9-[[3-fluoro-2-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-ethyl-N-[(1S)-2-imidazol-1-yl-1-phenylethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H20N6
5-ethyl-N-[(1S)-2-imidazol-1-yl-1-phenylethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-N-[(1R)-2-imidazol-1-yl-1-phenylethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H20N6
5-ethyl-N-[(1R)-2-imidazol-1-yl-1-phenylethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5-methylpyridin-3-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C21H25N3O
(5-methylpyridin-3-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5S)-3-methyl-N-(pyrazolo[1,5-a]pyridin-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C13H14N4O2
(5S)-3-methyl-N-(pyrazolo[1,5-a]pyridin-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-chloro-3-methyl-N-[[(6R)-1,4-oxazepan-6-yl]methyl]-1-benzothiophene-2-sulfonamide —— C15H19ClN2O3S2
5-chloro-3-methyl-N-[[(6R)-1,4-oxazepan-6-yl]methyl]-1-benzothiophene-2-sulfonamide
—— 5-[(3S)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H28N4O3
5-[(3S)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— (5S)-3-methyl-9-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H21N3O4
(5S)-3-methyl-9-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5-propyl-1,2-oxazol-3-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C21H27N3O2
(5-propyl-1,2-oxazol-3-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— 5-[(3R)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H28N4O2
5-[(3R)-3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl]-1H-pyridin-2-one