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—— 5-ethyl-N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine —— C17H24N6O
5-ethyl-N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
—— (5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)prop-2-enoate —— C22H18ClNO5
(5-phenyl-1,3-oxazol-2-yl)methyl (E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)prop-2-enoate
—— 5-(4-fluorophenyl)-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H19FN6
5-(4-fluorophenyl)-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine —— C17H24N6O
5-ethyl-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-N,5-dimethyl-N-[(1R)-1-(3-nitrophenyl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C19H22N2O3S
(5S)-N,5-dimethyl-N-[(1R)-1-(3-nitrophenyl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(1R)-1-[[2-(furan-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl]amino]ethyl]-1,3,4-thiadiazol-2-amine —— C16H19N7OS
5-[(1R)-1-[[2-(furan-2-yl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl]amino]ethyl]-1,3,4-thiadiazol-2-amine
—— (5R)-N,5-dimethyl-N-[(1R)-1-(3-nitrophenyl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C19H22N2O3S
(5R)-N,5-dimethyl-N-[(1R)-1-(3-nitrophenyl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-ethyl-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H20N6
5-ethyl-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(4-fluorophenyl)-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H19FN6
5-(4-fluorophenyl)-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-N,5-dimethyl-N-[(1S)-1-(3-nitrophenyl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C19H22N2O3S
(5R)-N,5-dimethyl-N-[(1S)-1-(3-nitrophenyl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-ethyl-2,3-dimethyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H22N4O
5-ethyl-2,3-dimethyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H20N6
5-ethyl-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(1-Ethyl-2-oxoindol-3-ylidene)-2-(4-hexoxyphenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C26H26N4O3S
5-(1-Ethyl-2-oxoindol-3-ylidene)-2-(4-hexoxyphenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— (5S)-9-(1-benzofuran-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H20N2O3
(5S)-9-(1-benzofuran-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-N-(3,4-dimethoxyphenyl)-7-oxo-3-thiophen-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C18H17N5O4S
(5R)-N-(3,4-dimethoxyphenyl)-7-oxo-3-thiophen-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— (5S)-N-(3,4-dimethoxyphenyl)-7-oxo-3-thiophen-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C18H17N5O4S
(5S)-N-(3,4-dimethoxyphenyl)-7-oxo-3-thiophen-2-yl-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— [5-(4-methoxyphenyl)-2-methylpyrazol-3-yl]-[(2S)-2-phenylmorpholin-4-yl]methanone —— C22H23N3O3
[5-(4-methoxyphenyl)-2-methylpyrazol-3-yl]-[(2S)-2-phenylmorpholin-4-yl]methanone
—— (5R)-5-[2-(3-carboxyanilino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C19H15FN2O6
(5R)-5-[2-(3-carboxyanilino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5S)-5-[2-(3-carboxyanilino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C19H15FN2O6
(5S)-5-[2-(3-carboxyanilino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5Z)-2-imino-5-[2-(4-methoxyphenyl)-2-oxoethylidene]-1,3-thiazolidin-4-one —— C12H10N2O3S
(5Z)-2-imino-5-[2-(4-methoxyphenyl)-2-oxoethylidene]-1,3-thiazolidin-4-one
—— (5-Chloroquinolin-8-yl) 4-(2-oxopyrrolidin-1-yl)benzoate —— C20H15ClN2O3
(5-Chloroquinolin-8-yl) 4-(2-oxopyrrolidin-1-yl)benzoate
—— (5-Chloroquinolin-8-yl) 3-(1,3-benzothiazol-2-yl)propanoate —— C19H13ClN2O2S
(5-Chloroquinolin-8-yl) 3-(1,3-benzothiazol-2-yl)propanoate
—— (5-Chloroquinolin-8-yl) 3-methyl-4-oxophthalazine-1-carboxylate —— C19H12ClN3O3
(5-Chloroquinolin-8-yl) 3-methyl-4-oxophthalazine-1-carboxylate
—— (5-chloroquinolin-8-yl) 2-(2,3-dihydro-1H-inden-5-yloxy)acetate —— C20H16ClNO3
(5-chloroquinolin-8-yl) 2-(2,3-dihydro-1H-inden-5-yloxy)acetate
—— 5-bromo-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]pyridine-3-carboxamide —— C15H14BrN3O3
5-bromo-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]pyridine-3-carboxamide
—— 5-fluoro-1-methyl-N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]indole-2-carboxamide —— C16H15FN4O2S
5-fluoro-1-methyl-N-[5-[(2R)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]indole-2-carboxamide
—— (5R)-N-(3,4-difluorophenyl)-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C16H11F2N5O3
(5R)-N-(3,4-difluorophenyl)-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— (5S)-5-[2-(2,1,3-benzoxadiazol-4-ylamino)-2-oxoethyl]-3-(2-chlorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C18H13ClN4O5
(5S)-5-[2-(2,1,3-benzoxadiazol-4-ylamino)-2-oxoethyl]-3-(2-chlorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5S)-5-(2-anilino-2-oxoethyl)-3-(4-methoxyphenyl)-4H-1,2-oxazole-5-carboxylic acid —— C19H18N2O5
(5S)-5-(2-anilino-2-oxoethyl)-3-(4-methoxyphenyl)-4H-1,2-oxazole-5-carboxylic acid
—— 5-bromo-N-methyl-N-[(1R)-1-(3-nitrophenyl)ethyl]pyridine-3-carboxamide —— C15H14BrN3O3
5-bromo-N-methyl-N-[(1R)-1-(3-nitrophenyl)ethyl]pyridine-3-carboxamide
—— [5-(3-chlorophenyl)-2-methylpyrazol-3-yl]-[(2S)-2-phenylmorpholin-4-yl]methanone —— C21H20ClN3O2
[5-(3-chlorophenyl)-2-methylpyrazol-3-yl]-[(2S)-2-phenylmorpholin-4-yl]methanone
—— (5R)-5-[2-(2,1,3-benzoxadiazol-4-ylamino)-2-oxoethyl]-3-(2-chlorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C18H13ClN4O5
(5R)-5-[2-(2,1,3-benzoxadiazol-4-ylamino)-2-oxoethyl]-3-(2-chlorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5R)-N-[2-(difluoromethoxy)phenyl]-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C17H13F2N5O4
(5R)-N-[2-(difluoromethoxy)phenyl]-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— 5-[(4R)-1-benzyl-3,6-dimethyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]-3-methoxybenzene-1,2-diol —— C21H21N3O3S
5-[(4R)-1-benzyl-3,6-dimethyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]-3-methoxybenzene-1,2-diol
—— 5-fluoro-1-methyl-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]indole-2-carboxamide —— C16H15FN4O2S
5-fluoro-1-methyl-N-[5-[(2S)-oxolan-2-yl]-1,3,4-thiadiazol-2-yl]indole-2-carboxamide
—— (5R)-5-[2-(2,1,3-benzoxadiazol-4-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C18H13FN4O5
(5R)-5-[2-(2,1,3-benzoxadiazol-4-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5R)-5-[2-(4-carboxyanilino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C19H15FN2O6
(5R)-5-[2-(4-carboxyanilino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5S)-N-[2-(difluoromethoxy)phenyl]-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C17H13F2N5O4
(5S)-N-[2-(difluoromethoxy)phenyl]-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— (5S)-N-(3,4-difluorophenyl)-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C16H11F2N5O3
(5S)-N-(3,4-difluorophenyl)-3-(furan-2-yl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— 5-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]pentanenitrile —— C17H18N2O2S
5-[4-(5-Acetyl-4-methyl-1,3-thiazol-2-yl)phenoxy]pentanenitrile
—— [5-(3-chlorophenyl)-2-methylpyrazol-3-yl]-[(2R)-2-phenylmorpholin-4-yl]methanone —— C21H20ClN3O2
[5-(3-chlorophenyl)-2-methylpyrazol-3-yl]-[(2R)-2-phenylmorpholin-4-yl]methanone
—— 5-[(4S)-1-benzyl-3,6-dimethyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]-3-methoxybenzene-1,2-diol —— C21H21N3O3S
5-[(4S)-1-benzyl-3,6-dimethyl-4H-pyrazolo[3,4-d][1,3]thiazin-4-yl]-3-methoxybenzene-1,2-diol
—— 5-(1,3-benzothiazol-2-yl)-N-[[2-[(dimethylamino)methyl]phenyl]methyl]pentanamide —— C22H27N3OS
5-(1,3-benzothiazol-2-yl)-N-[[2-[(dimethylamino)methyl]phenyl]methyl]pentanamide
—— (5R)-3-(furan-2-yl)-7-oxo-N-[4-(trifluoromethoxy)phenyl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C17H12F3N5O4
(5R)-3-(furan-2-yl)-7-oxo-N-[4-(trifluoromethoxy)phenyl]-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— (5S)-5-[2-(2,1,3-benzothiadiazol-4-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C18H13FN4O4S
(5S)-5-[2-(2,1,3-benzothiadiazol-4-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5R)-5-[2-(2,1,3-benzothiadiazol-5-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C18H13FN4O4S
(5R)-5-[2-(2,1,3-benzothiadiazol-5-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5S)-3-(4-fluorophenyl)-5-[2-(2-methoxycarbonylanilino)-2-oxoethyl]-4H-1,2-oxazole-5-carboxylic acid —— C20H17FN2O6
(5S)-3-(4-fluorophenyl)-5-[2-(2-methoxycarbonylanilino)-2-oxoethyl]-4H-1,2-oxazole-5-carboxylic acid
—— (5S)-5-[2-(2,1,3-benzothiadiazol-5-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid —— C18H13FN4O4S
(5S)-5-[2-(2,1,3-benzothiadiazol-5-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4H-1,2-oxazole-5-carboxylic acid
—— (5S)-3-(furan-2-yl)-N-(3-methoxyphenyl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide —— C17H15N5O4
(5S)-3-(furan-2-yl)-N-(3-methoxyphenyl)-7-oxo-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrimidine-5-carboxamide
—— 5-chloro-N-[[2-[(dimethylamino)methyl]phenyl]methyl]-1-benzofuran-2-carboxamide —— C19H19ClN2O2
5-chloro-N-[[2-[(dimethylamino)methyl]phenyl]methyl]-1-benzofuran-2-carboxamide