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—— 5-(4-bromophenyl)-2-[(2R)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H21BrN4O
5-(4-bromophenyl)-2-[(2R)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(2-methoxyphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C23H20N4O2
5-(2-methoxyphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(1,3-benzodioxol-5-yl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H18N4O4
5-(1,3-benzodioxol-5-yl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-bromophenyl)prop-2-enoate —— C18H15BrN2O4
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(4-bromophenyl)prop-2-enoate
—— 5-(2-methoxyphenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O2
5-(2-methoxyphenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-methylsulfonyl-N-[2-(4-methyl-1,2,4-triazol-3-yl)ethyl]-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine —— C15H23N7O2S
5-methylsulfonyl-N-[2-(4-methyl-1,2,4-triazol-3-yl)ethyl]-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine
—— 5-[(2,6-Dichlorophenyl)sulfanylmethyl]-3-(2-methoxyphenyl)-1,2,4-oxadiazole —— C16H12Cl2N2O2S
5-[(2,6-Dichlorophenyl)sulfanylmethyl]-3-(2-methoxyphenyl)-1,2,4-oxadiazole
—— 5-(3,4-dimethoxyphenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C21H24N4O3
5-(3,4-dimethoxyphenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C24H22N4O3
5-(3,4-dimethoxyphenyl)-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(1,3-benzodioxol-5-yl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H20N4O3
5-(1,3-benzodioxol-5-yl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3-methoxyphenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H20N4O3
5-(3-methoxyphenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(1,3-benzodioxol-5-yl)-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C23H18N4O3
5-(1,3-benzodioxol-5-yl)-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-fluorophenyl)-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C22H17FN4O
5-(4-fluorophenyl)-2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-chlorophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C18H17ClN4O2
5-(4-chlorophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C21H24N4O3
5-(3,4-dimethoxyphenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O4
5-(3,4-dimethoxyphenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-fluorophenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H19FN4O
5-(4-fluorophenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[(2S)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C22H26N4O3
5-(3,4-dimethoxyphenyl)-2-[(2S)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C22H26N4O3
5-(3,4-dimethoxyphenyl)-2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-bromophenyl)-2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H21BrN4O
5-(4-bromophenyl)-2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(2-methoxyphenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O2
5-(2-methoxyphenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-bromophenyl)-2-[(2S)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H19BrN4O
5-(4-bromophenyl)-2-[(2S)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C24H22N4O3
5-(3,4-dimethoxyphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-chlorophenyl)-2-[(2R)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H21ClN4O
5-(4-chlorophenyl)-2-[(2R)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-fluorophenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H19FN4O
5-(4-fluorophenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O4
5-(3,4-dimethoxyphenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-fluorophenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C22H17FN4O
5-(4-fluorophenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(2-fluorophenyl)prop-2-enoate —— C18H15FN2O4
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(2-fluorophenyl)prop-2-enoate
—— 5-(4-fluorophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C18H17FN4O2
5-(4-fluorophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-chlorophenyl)-2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H21ClN4O
5-(4-chlorophenyl)-2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-chlorophenyl)-2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H21ClN4O
5-(4-chlorophenyl)-2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-bromophenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C18H17BrN4O2
5-(4-bromophenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-chlorophenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C18H17ClN4O2
5-(4-chlorophenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3,4-dimethoxyphenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C21H24N4O3
5-(3,4-dimethoxyphenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-[3-[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one —— C21H28N4O3
5-[3-[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-3-oxopropyl]-4,6-dimethyl-1H-pyrimidin-2-one
—— 5-(4-bromophenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H19BrN4O
5-(4-bromophenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(3-nitrophenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C18H17N5O4
5-(3-nitrophenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-chlorophenyl)-2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H21ClN4O
5-(4-chlorophenyl)-2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-bromophenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C22H17BrN4O
5-(4-bromophenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-bromophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C18H17BrN4O2
5-(4-bromophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-[[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C14H15N5O2S2
5-[[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— 5-(4-bromophenyl)-2-[(2S)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H21BrN4O
5-(4-bromophenyl)-2-[(2S)-2-ethylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-methylphenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O
5-(4-methylphenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-methylphenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H20N4O2
5-(4-methylphenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(2-methylpropyl)-3-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-1,2,4-oxadiazole —— C14H20N4O2
5-(2-methylpropyl)-3-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]-1,2,4-oxadiazole
—— 5-naphthalen-2-yl-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C22H20N4O2
5-naphthalen-2-yl-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-methylphenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C19H20N4O2
5-(4-methylphenyl)-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— [5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 1H-indole-2-carboxylate —— C18H15N3O4
[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 1H-indole-2-carboxylate
—— 5-(4-nitrophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C18H17N5O4
5-(4-nitrophenyl)-2-[[(2R)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-naphthalen-2-yl-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one —— C22H20N4O2
5-naphthalen-2-yl-2-[[(2S)-oxolan-2-yl]methylamino]-1H-pyrido[2,3-d]pyrimidin-4-one