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—— 5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-2-methylbenzamide —— C15H21N3O3S
5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-2-methylbenzamide
—— 5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-2-chlorobenzonitrile —— C14H16ClN3O2S
5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-2-chlorobenzonitrile
—— [5-(2-fluorophenyl)-1,2-oxazol-3-yl]-[(2R)-2-(1-methylpyrrol-2-yl)azepan-1-yl]methanone —— C21H22FN3O2
[5-(2-fluorophenyl)-1,2-oxazol-3-yl]-[(2R)-2-(1-methylpyrrol-2-yl)azepan-1-yl]methanone
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C15H20N4O2
(5-propan-2-yl-1,3-oxazol-4-yl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— 5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-1,3-dimethylpyrimidine-2,4-dione —— C13H20N4O4S
5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-2-fluorobenzonitrile —— C14H16FN3O2S
5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-2-fluorobenzonitrile
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C15H20N4O2
(5-propan-2-yl-1,3-oxazol-4-yl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(3S)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone —— C14H19N5O2
(5-propan-2-yl-1,3-oxazol-4-yl)-[(3S)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone
—— 5-methyl-3-[(3S)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole —— C15H20N4O
5-methyl-3-[(3S)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-propan-2-yl-3-[(3R)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole —— C17H24N4O
5-propan-2-yl-3-[(3R)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-methyl-3-[(3R)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole —— C15H20N4O
5-methyl-3-[(3R)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-{[(Ethylcarbamoyl)(propan-2-YL)amino]methyl}-2-methoxyphenyl propane-2-sulfonate —— C17H28N2O5S
5-{[(Ethylcarbamoyl)(propan-2-YL)amino]methyl}-2-methoxyphenyl propane-2-sulfonate
—— [5-[[cyclobutanecarbonyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C20H29NO6S
[5-[[cyclobutanecarbonyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— [5-[[Cyclopropyl-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C19H20FNO5S
[5-[[Cyclopropyl-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— [5-[[acetyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C18H27NO6S
[5-[[acetyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— 5-[[(1S)-1-(4-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide —— C22H24FN3O2
5-[[(1S)-1-(4-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide
—— [5-[[[(2S)-butan-2-yl]-(3,3-dimethylbutanoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C20H33NO5S
[5-[[[(2S)-butan-2-yl]-(3,3-dimethylbutanoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— (5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2S)-2-[(1R)-1-phenylpropyl]pyrrolidin-1-yl]methanone —— C22H27ClN4O
(5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2S)-2-[(1R)-1-phenylpropyl]pyrrolidin-1-yl]methanone
—— 5-[[(1R)-1-(4-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide —— C22H24FN3O2
5-[[(1R)-1-(4-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide
—— [5-[[Cyclopropyl(3-methylbutanoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C19H29NO5S
[5-[[Cyclopropyl(3-methylbutanoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— 5-[(N-Cyclopropyl-3,3-dimethylbutanamido)methyl]-2-methoxyphenyl methanesulfonate —— C18H27NO5S
5-[(N-Cyclopropyl-3,3-dimethylbutanamido)methyl]-2-methoxyphenyl methanesulfonate
—— (5-propan-2-yl-1,3-oxazol-4-yl)-[(3R)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone —— C14H19N5O2
(5-propan-2-yl-1,3-oxazol-4-yl)-[(3R)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone
—— (5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2S)-2-[(1S)-1-phenylpropyl]pyrrolidin-1-yl]methanone —— C22H27ClN4O
(5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2S)-2-[(1S)-1-phenylpropyl]pyrrolidin-1-yl]methanone
—— 5-[[(1S)-1-(4-fluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide —— C22H25FN3O2+
5-[[(1S)-1-(4-fluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-propan-2-ylfuran-2-carboxamide
—— [5-[[[(2R)-butan-2-yl]-(3,3-dimethylbutanoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C20H33NO5S
[5-[[[(2R)-butan-2-yl]-(3,3-dimethylbutanoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— (5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2R)-2-[(1S)-1-phenylpropyl]pyrrolidin-1-yl]methanone —— C22H27ClN4O
(5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2R)-2-[(1S)-1-phenylpropyl]pyrrolidin-1-yl]methanone
—— [5-[[tert-butylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate —— C19H30N2O6S
[5-[[tert-butylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] methanesulfonate
—— [5-[[acetyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C18H27NO6S
[5-[[acetyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— (5R)-N-[1-[2-(cyclopentylamino)-2-oxoethyl]pyrazol-4-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C20H23N5O3
(5R)-N-[1-[2-(cyclopentylamino)-2-oxoethyl]pyrazol-4-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— [5-[[[(2S)-butan-2-yl]-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C20H24FNO5S
[5-[[[(2S)-butan-2-yl]-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— 5-[2-chloro-5-[(2R)-2-(4-ethoxyphenyl)pyrrolidin-1-yl]sulfonylphenyl]-2H-tetrazole —— C19H20ClN5O3S
5-[2-chloro-5-[(2R)-2-(4-ethoxyphenyl)pyrrolidin-1-yl]sulfonylphenyl]-2H-tetrazole
—— [5-[[Cyclopropyl-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C21H24FNO5S
[5-[[Cyclopropyl-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— [5-[[Tert-butylcarbamoyl(2-methylpropyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C18H30N2O5S
[5-[[Tert-butylcarbamoyl(2-methylpropyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— 5-[[(1S)-1-(4-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propylfuran-2-carboxamide —— C22H24FN3O2
5-[[(1S)-1-(4-fluorophenyl)-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-N-propylfuran-2-carboxamide
—— [5-[[Cyclopropyl(propan-2-ylcarbamoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C18H28N2O5S
[5-[[Cyclopropyl(propan-2-ylcarbamoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— 5-({N-[2-(Dimethylamino)ethyl]-3-methylbutanamido}methyl)-2-methoxyphenyl propane-2-sulfonate —— C20H34N2O5S
5-({N-[2-(Dimethylamino)ethyl]-3-methylbutanamido}methyl)-2-methoxyphenyl propane-2-sulfonate
—— 5-{[1-(2-Fluorophenyl)-N-(propan-2-YL)formamido]methyl}-2-methoxyphenyl ethane-1-sulfonate —— C20H24FNO5S
5-{[1-(2-Fluorophenyl)-N-(propan-2-YL)formamido]methyl}-2-methoxyphenyl ethane-1-sulfonate
—— 5-[2-chloro-5-[(2S)-2-(4-ethoxyphenyl)pyrrolidin-1-yl]sulfonylphenyl]-2H-tetrazole —— C19H20ClN5O3S
5-[2-chloro-5-[(2S)-2-(4-ethoxyphenyl)pyrrolidin-1-yl]sulfonylphenyl]-2H-tetrazole
—— [5-[[2-(Dimethylamino)ethyl-(propan-2-ylcarbamoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate —— C18H31N3O5S
[5-[[2-(Dimethylamino)ethyl-(propan-2-ylcarbamoyl)amino]methyl]-2-methoxyphenyl] ethanesulfonate
—— [5-[[[(2S)-butan-2-yl]-(3-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C20H24FNO5S
[5-[[[(2S)-butan-2-yl]-(3-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— (5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2R)-2-[(1R)-1-phenylpropyl]pyrrolidin-1-yl]methanone —— C22H27ClN4O
(5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)-[(2R)-2-[(1R)-1-phenylpropyl]pyrrolidin-1-yl]methanone
—— [5-[[[(2R)-butan-2-yl]-(2-methylpropanoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C19H31NO5S
[5-[[[(2R)-butan-2-yl]-(2-methylpropanoyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— [5-[[[(2R)-butan-2-yl]-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C20H24FNO5S
[5-[[[(2R)-butan-2-yl]-(2-fluorobenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— 5-[4-(4-Fluorophenyl)piperazine-1-carbonyl]-1-methanesulfonyl-2,3-dihydro-1H-indole —— C20H22FN3O3S
5-[4-(4-Fluorophenyl)piperazine-1-carbonyl]-1-methanesulfonyl-2,3-dihydro-1H-indole
—— [5-[[Cyclopropyl-(2-methoxyacetyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C17H25NO6S
[5-[[Cyclopropyl-(2-methoxyacetyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— [5-[[[(2S)-butan-2-yl]-(cyclobutanecarbonyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C20H31NO5S
[5-[[[(2S)-butan-2-yl]-(cyclobutanecarbonyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— 5-[(4-Chlorophenyl)methyl]-4-(methoxymethyl)-2-methyl-6-(4-methylsulfonylpiperazin-1-yl)pyrimidine —— C19H25ClN4O3S
5-[(4-Chlorophenyl)methyl]-4-(methoxymethyl)-2-methyl-6-(4-methylsulfonylpiperazin-1-yl)pyrimidine
—— 5-[[(1S)-1-(4-fluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-(2-methylpropyl)furan-2-carboxamide —— C23H27FN3O2+
5-[[(1S)-1-(4-fluorophenyl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-2-ium-2-yl]methyl]-N-(2-methylpropyl)furan-2-carboxamide
—— 5-fluoro-2-[[methyl-[(3S)-1-(6-methylpyridazin-3-yl)piperidin-3-yl]amino]methyl]benzonitrile —— C19H22FN5
5-fluoro-2-[[methyl-[(3S)-1-(6-methylpyridazin-3-yl)piperidin-3-yl]amino]methyl]benzonitrile
—— 5-{[1-(2-Fluorophenyl)-N-(2-methylpropyl)formamido]methyl}-2-methoxyphenyl ethane-1-sulfonate —— C21H26FNO5S
5-{[1-(2-Fluorophenyl)-N-(2-methylpropyl)formamido]methyl}-2-methoxyphenyl ethane-1-sulfonate