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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-methyl-2-(1-methylimidazol-2-yl)-N-(2-morpholin-4-ylethyl)pyrazolo[1,5-a]pyrimidin-7-amine —— C17H23N7O
5-methyl-2-(1-methylimidazol-2-yl)-N-(2-morpholin-4-ylethyl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine —— C18H19N7
5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[4-(Furan-2-yl)-2-[4-(2-methoxyethyl)piperazin-1-yl]pyrimidin-5-yl]-3-methyl-1,2-oxazole —— C19H23N5O3
5-[4-(Furan-2-yl)-2-[4-(2-methoxyethyl)piperazin-1-yl]pyrimidin-5-yl]-3-methyl-1,2-oxazole
—— 5-Pyrazin-2-yl-2-pyrrolidin-1-yl-4-thiophen-2-ylpyrimidine —— C16H15N5S
5-Pyrazin-2-yl-2-pyrrolidin-1-yl-4-thiophen-2-ylpyrimidine
—— 5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-(3-morpholin-4-ylpropyl)pyrazolo[1,5-a]pyrimidin-7-amine —— C19H27N7O
5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-(3-morpholin-4-ylpropyl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H22N6O
5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5,6-Dimethyl-2-(1-methylimidazol-2-yl)-7-(4-methylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine —— C17H23N7
5,6-Dimethyl-2-(1-methylimidazol-2-yl)-7-(4-methylpiperazin-1-yl)pyrazolo[1,5-a]pyrimidine
—— 5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H22N6O
5,6-dimethyl-2-(1-methylimidazol-2-yl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3S)-3-(2-morpholin-4-yl-5-pyridin-3-ylpyrimidin-4-yl)piperidin-1-yl]-5-oxopentanoic acid —— C23H29N5O4
5-[(3S)-3-(2-morpholin-4-yl-5-pyridin-3-ylpyrimidin-4-yl)piperidin-1-yl]-5-oxopentanoic acid
—— 5-[4-[(3R)-1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-2-pyrrolidin-1-ylpyrimidin-5-yl]-3-methyl-1,2-oxazole —— C23H29N7O
5-[4-[(3R)-1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-2-pyrrolidin-1-ylpyrimidin-5-yl]-3-methyl-1,2-oxazole
—— 5-tert-butyl-3-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C22H30N6O3
5-tert-butyl-3-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-[[[(1R,6R,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine —— C21H27ClN4
5-[[[(1R,6R,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine
—— 5-tert-butyl-3-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C18H24N6OS
5-tert-butyl-3-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-pyrazin-2-ylethyl)pyrimidin-2-amine —— C21H22N8O
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-pyrazin-2-ylethyl)pyrimidin-2-amine
—— 5-(3,4-dimethyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine —— C20H19N7O
5-(3,4-dimethyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
—— 5-(3,4-dimethyl-1,2-oxazol-5-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine —— C18H20N6O3S
5-(3,4-dimethyl-1,2-oxazol-5-yl)-N-[(3R)-1,1-dioxothiolan-3-yl]-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine
—— 5-[4-[(3S)-1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-2-pyrrolidin-1-ylpyrimidin-5-yl]-3-methyl-1,2-oxazole —— C23H29N7O
5-[4-[(3S)-1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-2-pyrrolidin-1-ylpyrimidin-5-yl]-3-methyl-1,2-oxazole
—— (5-Cyclopropyl-2-methylpyrazol-3-yl)-[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-(propan-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C24H31N7O2
(5-Cyclopropyl-2-methylpyrazol-3-yl)-[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-(propan-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— (5-Methylthiophen-2-yl)-[4-[2-(propan-2-ylamino)-5-pyridin-2-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C23H27N5OS
(5-Methylthiophen-2-yl)-[4-[2-(propan-2-ylamino)-5-pyridin-2-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— 5-[[[(1S,6S,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine —— C21H27ClN4
5-[[[(1S,6S,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-[2-(5-methylpyrazol-1-yl)ethyl]pyrimidin-2-amine —— C21H24N8O
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-[2-(5-methylpyrazol-1-yl)ethyl]pyrimidin-2-amine
—— 5-[2-(Azepan-1-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-5-yl]-4-ethyl-3-methyl-1,2-oxazole —— C21H26N6O
5-[2-(Azepan-1-yl)-4-(5-methylpyrazin-2-yl)pyrimidin-5-yl]-4-ethyl-3-methyl-1,2-oxazole
—— (5S,7R)-2-[(2S)-1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine —— C20H27F3N6
(5S,7R)-2-[(2S)-1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]-5-propan-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine
—— 5-[[[(1S,6R,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine —— C21H27ClN4
5-[[[(1S,6R,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(3-piperidin-1-ylpropyl)pyrimidin-2-amine —— C23H31N7O
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(3-piperidin-1-ylpropyl)pyrimidin-2-amine
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-N-[(4-fluorophenyl)methyl]-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine —— C22H21FN6O
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-N-[(4-fluorophenyl)methyl]-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine
—— 5-[[[(1R,6S,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine —— C21H27ClN4
5-[[[(1R,6S,7S,8R)-8-(4-chlorophenyl)-7-bicyclo[4.2.0]octanyl]amino]methyl]-N,N-dimethylpyrimidin-2-amine
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(3-pyridin-2-ylpropyl)pyrimidin-2-amine —— C23H25N7O
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(3-pyridin-2-ylpropyl)pyrimidin-2-amine
—— (5-Methylfuran-2-yl)-[4-(5-methylsulfonyl-2-piperidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone —— C21H28N4O4S
(5-Methylfuran-2-yl)-[4-(5-methylsulfonyl-2-piperidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone
—— 5-(1-ethyl-3-methylpyrazol-4-yl)-N,2-dimethyl-1,1-dioxo-N-phenyl-1,2,6-thiadiazine-3-carboxamide —— C18H21N5O3S
5-(1-ethyl-3-methylpyrazol-4-yl)-N,2-dimethyl-1,1-dioxo-N-phenyl-1,2,6-thiadiazine-3-carboxamide
—— [5-(1-Ethyl-3-methylpyrazol-4-yl)-2-methyl-1,1-dioxo-1,2,6-thiadiazin-3-yl]-(4-ethylpiperazin-1-yl)methanone —— C17H26N6O3S
[5-(1-Ethyl-3-methylpyrazol-4-yl)-2-methyl-1,1-dioxo-1,2,6-thiadiazin-3-yl]-(4-ethylpiperazin-1-yl)methanone
—— 5-[[(1R,12S)-7-tert-butyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]pyrimidin-2-amine —— C20H25N7
5-[[(1R,12S)-7-tert-butyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]pyrimidin-2-amine
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[4-(2,4-dimethoxypyrimidin-5-yl)-4-hydroxypiperidin-1-yl]methanone —— C19H23N3O4S
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[4-(2,4-dimethoxypyrimidin-5-yl)-4-hydroxypiperidin-1-yl]methanone
—— [(5R)-5-tert-butyl-4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl]-[4-(2,4-dimethoxypyrimidin-5-yl)-4-hydroxypiperidin-1-yl]methanone —— C23H32N4O5
[(5R)-5-tert-butyl-4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl]-[4-(2,4-dimethoxypyrimidin-5-yl)-4-hydroxypiperidin-1-yl]methanone
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-morpholin-4-ylethyl)pyrimidin-2-amine —— C21H27N7O2
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-4-(5-methylpyrazin-2-yl)-N-(2-morpholin-4-ylethyl)pyrimidin-2-amine
—— 5-Ethyl-3-methyl-4-(2-piperidin-1-yl-5-pyrazin-2-ylpyrimidin-4-yl)-1,2-oxazole —— C19H22N6O
5-Ethyl-3-methyl-4-(2-piperidin-1-yl-5-pyrazin-2-ylpyrimidin-4-yl)-1,2-oxazole
—— 5-(3-methyl-1,2-oxazol-5-yl)-N-(3-morpholin-4-ylpropyl)-4-thiophen-2-ylpyrimidin-2-amine —— C19H23N5O2S
5-(3-methyl-1,2-oxazol-5-yl)-N-(3-morpholin-4-ylpropyl)-4-thiophen-2-ylpyrimidin-2-amine
—— 5-[4-[(Z)-N-[[2-(3-methoxyanilino)acetyl]amino]-C-methylcarbonimidoyl]phenyl]furan-2-carboxylic acid —— C22H21N3O5
5-[4-[(Z)-N-[[2-(3-methoxyanilino)acetyl]amino]-C-methylcarbonimidoyl]phenyl]furan-2-carboxylic acid
—— 5-(ethylsulfanylmethyl)-3-[1-(furan-3-ylmethyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C17H22N6O2S
5-(ethylsulfanylmethyl)-3-[1-(furan-3-ylmethyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-N-[(3-methoxyphenyl)methyl]-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine —— C23H24N6O2
5-(4-ethyl-3-methyl-1,2-oxazol-5-yl)-N-[(3-methoxyphenyl)methyl]-4-(5-methylpyrazin-2-yl)pyrimidin-2-amine
—— 5-[4-[(Z)-N-[[2-(3-methoxyanilino)acetyl]amino]-C-methylcarbonimidoyl]phenyl]furan-2-carboxylate —— C22H20N3O5-
5-[4-[(Z)-N-[[2-(3-methoxyanilino)acetyl]amino]-C-methylcarbonimidoyl]phenyl]furan-2-carboxylate
—— 5,6-dimethyl-2-(oxan-4-yl)-N-[(1-propylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C22H35N5O
5,6-dimethyl-2-(oxan-4-yl)-N-[(1-propylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(ethylsulfanylmethyl)-3-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C21H30N6O2S
5-(ethylsulfanylmethyl)-3-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-tert-butyl-3-[1-[(2-chlorophenyl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C20H25ClN6O
5-tert-butyl-3-[1-[(2-chlorophenyl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-(ethylsulfanylmethyl)-3-[1-[(2-methylpyrimidin-4-yl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C18H24N8OS
5-(ethylsulfanylmethyl)-3-[1-[(2-methylpyrimidin-4-yl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylthiophen-2-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine —— C19H17N5OS
5-(3-methyl-1,2-oxazol-5-yl)-4-(5-methylthiophen-2-yl)-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
—— 5-(ethylsulfanylmethyl)-3-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C21H30N6O2S
5-(ethylsulfanylmethyl)-3-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5,6-dimethyl-2-(oxan-4-yl)-N-[[(3R)-1-propan-2-ylpiperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C22H35N5O
5,6-dimethyl-2-(oxan-4-yl)-N-[[(3R)-1-propan-2-ylpiperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[[(1S,12R)-7-tert-butyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]pyrimidin-2-amine —— C20H25N7
5-[[(1S,12R)-7-tert-butyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]pyrimidin-2-amine
—— 5-[2-(Azepan-1-yl)-4-(2-methylpyridin-3-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole —— C20H23N5O
5-[2-(Azepan-1-yl)-4-(2-methylpyridin-3-yl)pyrimidin-5-yl]-3-methyl-1,2-oxazole