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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-9-(2,1,3-benzoxadiazol-4-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H18N4O3
(5R)-9-(2,1,3-benzoxadiazol-4-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(2R)-1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile —— C18H26N4O
5-[(2R)-1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxypyridine-2-carbonitrile
—— (5S)-9-(2,1,3-benzoxadiazol-4-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H18N4O3
(5S)-9-(2,1,3-benzoxadiazol-4-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 3-(methoxymethyl)benzoate —— C19H17NO4
(5-Phenyl-1,2-oxazol-3-yl)methyl 3-(methoxymethyl)benzoate
—— 5-[(3S)-3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazine-1-carbonyl]-1H-pyridin-2-one —— C21H27N3O3
5-[(3S)-3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazine-1-carbonyl]-1H-pyridin-2-one
—— (5R)-3-methyl-9-(6-piperidin-1-ylpyrimidin-4-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H25N5O2
(5R)-3-methyl-9-(6-piperidin-1-ylpyrimidin-4-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]pyridin-2-amine —— C20H22FN5O
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]pyridin-2-amine
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(2-pyridin-3-ylethyl)pyrimidin-2-amine —— C17H23N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(2-pyridin-3-ylethyl)pyrimidin-2-amine
—— 5-[(6S)-8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C22H28N4O2
5-[(6S)-8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— 5-(Furan-2-yl)-3-[(5-piperidin-1-ylsulfonylpyridin-2-yl)sulfanylmethyl]-1,2-oxazole —— C18H19N3O4S2
5-(Furan-2-yl)-3-[(5-piperidin-1-ylsulfonylpyridin-2-yl)sulfanylmethyl]-1,2-oxazole
—— 5-chloro-N-methyl-N-[[(2R)-oxolan-2-yl]methyl]-3-phenyl-1H-indole-2-carboxamide —— C21H21ClN2O2
5-chloro-N-methyl-N-[[(2R)-oxolan-2-yl]methyl]-3-phenyl-1H-indole-2-carboxamide
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 3-(3-oxo-1,4-benzothiazin-4-yl)propanoate —— C21H19N3O4S
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 3-(3-oxo-1,4-benzothiazin-4-yl)propanoate
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(2-pyridin-3-ylethyl)pyrimidin-2-amine —— C17H23N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(2-pyridin-3-ylethyl)pyrimidin-2-amine
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetate —— C20H15N3O3S
(5-Phenyl-1,2-oxazol-3-yl)methyl 2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetate
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetate —— C20H16N4O3S
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2-pyridin-3-yl-1,3-thiazol-4-yl)acetate
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 4-[(propan-2-ylcarbamoylamino)methyl]benzoate —— C20H21N3O5
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 4-[(propan-2-ylcarbamoylamino)methyl]benzoate
—— 5-(methoxymethyl)-N-[(1S)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H20N6O
5-(methoxymethyl)-N-[(1S)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(methoxymethyl)-N-[(1R)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H20N6O
5-(methoxymethyl)-N-[(1R)-1-(6-methyl-1H-benzimidazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-5-[(2-dibenzofuran-4-ylimidazol-1-yl)methyl]-1-methylpyrrolidin-2-one —— C21H19N3O2
(5R)-5-[(2-dibenzofuran-4-ylimidazol-1-yl)methyl]-1-methylpyrrolidin-2-one
—— (5S)-5-[(2-dibenzofuran-4-ylimidazol-1-yl)methyl]-1-methylpyrrolidin-2-one —— C21H19N3O2
(5S)-5-[(2-dibenzofuran-4-ylimidazol-1-yl)methyl]-1-methylpyrrolidin-2-one
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-2-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
—— 5-[(6S)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C19H24N4O3
5-[(6S)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-(4-fluorophenyl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H16FN7
5-(4-fluorophenyl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(6R)-8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C22H28N4O2
5-[(6R)-8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 3-(2-amino-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoate —— C20H20N6O3
(5-Phenyl-1,2-oxazol-3-yl)methyl 3-(2-amino-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl)propanoate
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-2-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
—— 5-[2-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C19H24N4O3
5-[2-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[[(2S)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methyl]-2-propylpyrimidine —— C20H28N4
5-[[(2S)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]methyl]-2-propylpyrimidine
—— 5-ethyl-7-[(3S)-3-phenylpiperazin-1-yl]pyrazolo[1,5-a]pyrimidine —— C18H21N5
5-ethyl-7-[(3S)-3-phenylpiperazin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-ethyl-7-[(3R)-3-phenylpiperazin-1-yl]pyrazolo[1,5-a]pyrimidine —— C18H21N5
5-ethyl-7-[(3R)-3-phenylpiperazin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5R)-2-(1,3-dihydroxypropan-2-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N2O5
(5R)-2-(1,3-dihydroxypropan-2-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(1,3-dihydroxypropan-2-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N2O5
(5S)-2-(1,3-dihydroxypropan-2-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidin-1-yl]methanone —— C18H17ClFN5O
(5-chloro-2-methylpyrimidin-4-yl)-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidin-1-yl]methanone
—— 5-[(6R)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C19H24N4O3
5-[(6R)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[2-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one —— C19H24N4O3
5-[2-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl]-2-methyl-1H-pyrimidin-6-one
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidin-1-yl]methanone —— C18H17ClFN5O
(5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidin-1-yl]methanone
—— 5-[[(3R)-3-hydroxypiperidin-3-yl]methyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C16H25N3O2S
5-[[(3R)-3-hydroxypiperidin-3-yl]methyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— 5-[(2S)-2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C17H24N4O2
5-[(2S)-2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile —— C19H16FN5O
5-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
—— (5R)-2-(1,3-dihydroxypropan-2-yl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H27FN2O4
(5R)-2-(1,3-dihydroxypropan-2-yl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H32N2O3
(5R)-2-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3S)-3-hydroxypiperidin-3-yl]methyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C16H25N3O2S
5-[[(3S)-3-hydroxypiperidin-3-yl]methyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— [5-[[(4-Ethylphenyl)carbamoyl-propan-2-ylamino]methyl]-2-methoxyphenyl] 3-(trifluoromethyl)benzenesulfonate —— C27H29F3N2O5S
[5-[[(4-Ethylphenyl)carbamoyl-propan-2-ylamino]methyl]-2-methoxyphenyl] 3-(trifluoromethyl)benzenesulfonate
—— 5-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile —— C19H16FN5O
5-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
—— (5R)-3-methyl-9-(2-phenylquinolin-4-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C23H23N3O2
(5R)-3-methyl-9-(2-phenylquinolin-4-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(2-fluorophenyl)-N-[(2R)-1-pyridin-3-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(2-fluorophenyl)-N-[(2R)-1-pyridin-3-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C16H16N4O2
5-[[(2R)-oxolan-2-yl]methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— (5S)-3-methyl-7-[[3-(pyridin-2-ylmethoxy)phenyl]methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H23N3O3
(5S)-3-methyl-7-[[3-(pyridin-2-ylmethoxy)phenyl]methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-2-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H32N2O3
(5S)-2-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-[(4-methylphenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H21N3O4
5-[(3S)-3-[(4-methylphenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione