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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-9-[2-(2-ethylimidazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H20N4O3
(5R)-9-[2-(2-ethylimidazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(3R)-3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H24FN5O2
5-[(3R)-3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H24FN3O2
5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (5S)-3-methyl-9-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H22N4O3
(5S)-3-methyl-9-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H15N3O3S2
(5R)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-9-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H22N4O3
(5R)-3-methyl-9-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-bromo-3-methyl-N-(2,2,2-trifluoroethyl)-1-benzofuran-2-carboxamide —— C12H9BrF3NO2
5-bromo-3-methyl-N-(2,2,2-trifluoroethyl)-1-benzofuran-2-carboxamide
—— 5-(hydroxymethyl)-2-methyl-4-[[methyl-[(3R)-1-(2-phenylethyl)piperidin-3-yl]amino]methyl]pyridin-3-ol —— C22H31N3O2
5-(hydroxymethyl)-2-methyl-4-[[methyl-[(3R)-1-(2-phenylethyl)piperidin-3-yl]amino]methyl]pyridin-3-ol
—— 5-bromo-N-[(1S)-1-(4-sulfamoylphenyl)ethyl]furan-2-carboxamide —— C13H13BrN2O4S
5-bromo-N-[(1S)-1-(4-sulfamoylphenyl)ethyl]furan-2-carboxamide
—— (5S)-3-methyl-7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H21N3O4
(5S)-3-methyl-7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-3-methyl-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H22N4O2S
(5R)-3-methyl-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[2-(1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H18N6O3
(5R)-9-[2-(1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H15N3O3S2
(5S)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(hydroxymethyl)-2-methyl-4-[[methyl-[(3S)-1-(2-phenylethyl)piperidin-3-yl]amino]methyl]pyridin-3-ol —— C22H31N3O2
5-(hydroxymethyl)-2-methyl-4-[[methyl-[(3S)-1-(2-phenylethyl)piperidin-3-yl]amino]methyl]pyridin-3-ol
—— (5R)-N-(2-chlorophenyl)-7-(2,2-dimethylpropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide —— C20H28ClN3O2
(5R)-N-(2-chlorophenyl)-7-(2,2-dimethylpropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-9-(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H16N4O3S
(5S)-9-(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H22N4O2S
(5S)-3-methyl-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H21N3O4
(5R)-9-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H20ClN5O3
(5S)-9-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H25N3O3
(5S)-3-methyl-9-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H16N4O3S
(5R)-9-(2-imidazo[2,1-b][1,3]thiazol-6-ylacetyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H21N3O4
(5S)-9-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-bromo-N-[(1R)-1-(4-sulfamoylphenyl)ethyl]furan-2-carboxamide —— C13H13BrN2O4S
5-bromo-N-[(1R)-1-(4-sulfamoylphenyl)ethyl]furan-2-carboxamide
—— 5-[[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H24FN3O2
5-[[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-(4-methyl-1,4-diazepan-1-yl)-2-[3-[(3S)-3-methylpiperidin-1-yl]-3-oxopropyl]pyridazin-3-one —— C19H31N5O2
5-(4-methyl-1,4-diazepan-1-yl)-2-[3-[(3S)-3-methylpiperidin-1-yl]-3-oxopropyl]pyridazin-3-one
—— (5R)-3-methyl-9-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H25N3O3
(5R)-3-methyl-9-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(1-ethyl-4,6-dimethyl-2-oxopyridine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H25N3O4
(5R)-9-(1-ethyl-4,6-dimethyl-2-oxopyridine-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(4-methyl-1,4-diazepan-1-yl)-2-[3-[(3R)-3-methylpiperidin-1-yl]-3-oxopropyl]pyridazin-3-one —— C19H31N5O2
5-(4-methyl-1,4-diazepan-1-yl)-2-[3-[(3R)-3-methylpiperidin-1-yl]-3-oxopropyl]pyridazin-3-one
—— (5R)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H18F2N2O
(5R)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(3-hydroxy-4-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H18N2O5
(5S)-7-(3-hydroxy-4-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H25N3O4
(5S)-9-[2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H25N3O4
(5R)-9-[2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H18F2N2O
(5S)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(3-hydroxypyridine-2-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H17N3O4
(5S)-9-(3-hydroxypyridine-2-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-5-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1,3-oxazolidin-2-one —— C17H22N2O3
(5R)-5-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1,3-oxazolidin-2-one
—— 5-[[2-[(3S)-morpholin-3-yl]acetyl]amino]pyridine-3-carboxylic acid —— C12H15N3O4
5-[[2-[(3S)-morpholin-3-yl]acetyl]amino]pyridine-3-carboxylic acid
—— (5S)-5-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1,3-oxazolidin-2-one —— C17H22N2O3
(5S)-5-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1,3-oxazolidin-2-one
—— 5-[[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine —— C19H18FN3O
5-[[(2R)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine
—— (5S)-9-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H19F4NO2
(5S)-9-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-(2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H21N5O3
(5S)-9-(2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H20ClN5O3
(5R)-9-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3R)-3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C19H24N4O2
5-[(3R)-3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-chloro-3-methyl-N-(2-methylsulfanyl-1,3-benzothiazol-6-yl)-1-phenylpyrazole-4-carboxamide —— C19H15ClN4OS2
5-chloro-3-methyl-N-(2-methylsulfanyl-1,3-benzothiazol-6-yl)-1-phenylpyrazole-4-carboxamide
—— (5S)-9-[2-(2-ethoxyethyl)-5-methylpyrazole-3-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H24N4O4
(5S)-9-[2-(2-ethoxyethyl)-5-methylpyrazole-3-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[2-(3-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H20N2O4
(5S)-9-[2-(3-hydroxyphenyl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H25N3O4
(5S)-7-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine —— C19H18FN3O
5-[[(2S)-2-(4-fluorophenyl)pyrrolidin-1-yl]methyl]-2-(furan-2-yl)pyrimidine
—— 5-[[(2R)-oxan-2-yl]methylsulfanyl]-1-phenyltetrazole —— C13H16N4OS
5-[[(2R)-oxan-2-yl]methylsulfanyl]-1-phenyltetrazole
—— [5-(methoxymethyl)thiophen-2-yl]-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C21H26N2O2S
[5-(methoxymethyl)thiophen-2-yl]-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— 5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C17H21FN4O2
5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide