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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-9-(2,1,3-benzothiadiazol-5-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H18N4O2S
(5S)-9-(2,1,3-benzothiadiazol-5-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H22FN3O2S
(5R)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-propan-2-yl-N-[(2R)-2-pyrrolidin-1-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H25N5
5-propan-2-yl-N-[(2R)-2-pyrrolidin-1-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-6-methyl-N-[[(6S)-4-methyl-1,4-oxazepan-6-yl]methyl]thieno[2,3-d]pyrimidin-4-amine —— C16H24N4OS
5-ethyl-6-methyl-N-[[(6S)-4-methyl-1,4-oxazepan-6-yl]methyl]thieno[2,3-d]pyrimidin-4-amine
—— (5S)-9-[4-(1H-pyrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H20N4O3
(5S)-9-[4-(1H-pyrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[3-(5-methyltetrazol-1-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20N6O3
(5S)-9-[3-(5-methyltetrazol-1-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]pyridine-2-carbonitrile —— C22H25FN4O
5-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepane-1-carbonyl]pyridine-2-carbonitrile
—— 5-[(1R)-1-[(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine —— C15H15N9S
5-[(1R)-1-[(1-methyl-6-pyridin-3-ylpyrazolo[3,4-d]pyrimidin-4-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine
—— (5S)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H22FN3O2S
(5S)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-phenyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H18N6
5-phenyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-9-(2,1,3-benzothiadiazol-5-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H18N4O2S
(5R)-9-(2,1,3-benzothiadiazol-5-ylmethyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3R)-3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C14H20N4O3
5-[[(3R)-3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— (5S)-3-methyl-7-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H20N4O3
(5S)-3-methyl-7-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-[3-(4-ethylphenyl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H24N2O3
(5R)-7-[3-(4-ethylphenyl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C20H24N6O2
5-[[methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (5S)-9-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H18ClN3O4
(5S)-9-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-7-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H20N4O3
(5R)-3-methyl-7-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-propan-2-yl-7-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C20H31N5
5-propan-2-yl-7-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5S)-2-(1,3-benzoxazol-2-yl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C23H25N3O3
(5S)-2-(1,3-benzoxazol-2-yl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-3-methyl-1-(2-methylpropyl)-N-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]pyrazole-4-carboxamide —— C17H23ClN4OS
5-chloro-3-methyl-1-(2-methylpropyl)-N-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]pyrazole-4-carboxamide
—— (5R)-9-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H18ClN3O4
(5R)-9-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— [5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl 1,3-benzodioxole-5-carboxylate —— C18H18N2O7S
[5-Amino-4-ethoxycarbonyl-2-(methylcarbamoyl)thiophen-3-yl]methyl 1,3-benzodioxole-5-carboxylate
—— (5R)-2-(1,3-benzoxazol-2-yl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C23H25N3O3
(5R)-2-(1,3-benzoxazol-2-yl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-[3-(4-ethylphenyl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H24N2O3
(5S)-7-[3-(4-ethylphenyl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H28N2O4
(5R)-9-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C20H24N6O2
5-[[methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (5R)-9-[(2,3-dimethoxyphenyl)methyl]-2-ethylsulfonyl-2,9-diazaspiro[4.5]decane —— C19H30N2O4S
(5R)-9-[(2,3-dimethoxyphenyl)methyl]-2-ethylsulfonyl-2,9-diazaspiro[4.5]decane
—— 5-[[(3S)-3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione —— C14H20N4O3
5-[[(3S)-3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl]-1H-pyrimidine-2,4-dione
—— (5S)-9-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H28N2O4
(5S)-9-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-chloro-5-methylsulfanylbenzoate —— C17H12Cl2N2O3S
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-chloro-5-methylsulfanylbenzoate
—— 5-fluoro-1-methyl-2-[[(2R)-2-pyridin-2-ylpiperidin-1-yl]methyl]indole —— C20H22FN3
5-fluoro-1-methyl-2-[[(2R)-2-pyridin-2-ylpiperidin-1-yl]methyl]indole
—— [5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-chloro-5-methylsulfanylbenzoate —— C17H12ClN3O5S
[5-(4-Nitrophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-chloro-5-methylsulfanylbenzoate
—— (5S)-9-[4-(3-fluorophenyl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H21FN2O3
(5S)-9-[4-(3-fluorophenyl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[1-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propyl-1,2,4-oxadiazole —— C16H17N5O3
5-[1-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propyl-1,2,4-oxadiazole
—— 5-cyclopropyl-N-(2,3-dihydro-1H-inden-5-yl)-2-phenylpyrazole-3-carboxamide —— C22H21N3O
5-cyclopropyl-N-(2,3-dihydro-1H-inden-5-yl)-2-phenylpyrazole-3-carboxamide
—— 5-[[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl]-2,1,3-benzothiadiazole —— C18H20N4OS
5-[[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl]-2,1,3-benzothiadiazole
—— (5S)-9-[(2,3-dimethoxyphenyl)methyl]-2-ethylsulfonyl-2,9-diazaspiro[4.5]decane —— C19H30N2O4S
(5S)-9-[(2,3-dimethoxyphenyl)methyl]-2-ethylsulfonyl-2,9-diazaspiro[4.5]decane
—— (5R)-9-[4-(3-fluorophenyl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H21FN2O3
(5R)-9-[4-(3-fluorophenyl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]pyridazin-3-one —— C16H23N5OS
5-[(3R)-3-(aminomethyl)pyrrolidin-1-yl]-2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]pyridazin-3-one
—— 5-methyl-N-(2-pyrrolidin-1-ylphenyl)-1,2-oxazole-3-carboxamide —— C15H17N3O2
5-methyl-N-(2-pyrrolidin-1-ylphenyl)-1,2-oxazole-3-carboxamide
—— 5-[[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H24FN3O2
5-[[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-fluoro-1-methyl-2-[[(2S)-2-pyridin-2-ylpiperidin-1-yl]methyl]indole —— C20H22FN3
5-fluoro-1-methyl-2-[[(2S)-2-pyridin-2-ylpiperidin-1-yl]methyl]indole
—— 5-chloro-N-[[(3R)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]-6-oxo-1H-pyridine-3-carboxamide —— C16H18ClN5O3
5-chloro-N-[[(3R)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]-6-oxo-1H-pyridine-3-carboxamide
—— [5-Chloro-1-[(2-chlorophenyl)methyl]-3-methylpyrazol-4-yl]-(4-propylpiperazin-1-yl)methanone —— C19H24Cl2N4O
[5-Chloro-1-[(2-chlorophenyl)methyl]-3-methylpyrazol-4-yl]-(4-propylpiperazin-1-yl)methanone
—— 5-chloro-3-methyl-1-(2-methylpropyl)-N-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]pyrazole-4-carboxamide —— C17H23ClN4OS
5-chloro-3-methyl-1-(2-methylpropyl)-N-[(6S)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]pyrazole-4-carboxamide
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(2,4-dimethylphenyl)methyl]pyridazin-3-one —— C19H26N4O2
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(2,4-dimethylphenyl)methyl]pyridazin-3-one
—— [5-(phenoxymethyl)furan-2-yl]-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]methanone —— C25H26N2O3
[5-(phenoxymethyl)furan-2-yl]-[4-[(E)-3-phenylprop-2-enyl]piperazin-1-yl]methanone
—— 5-chloro-N-[[(4S)-4-hydroxyazepan-4-yl]methyl]-3-methyl-1-benzothiophene-2-sulfonamide —— C16H21ClN2O3S2
5-chloro-N-[[(4S)-4-hydroxyazepan-4-yl]methyl]-3-methyl-1-benzothiophene-2-sulfonamide
—— 5-methyl-N-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1H-imidazole-4-carboxamide —— C16H22N6O3
5-methyl-N-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1H-imidazole-4-carboxamide
—— 5-[1-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propyl-1,2,4-oxadiazole —— C16H17N5O3
5-[1-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]triazol-4-yl]-3-propyl-1,2,4-oxadiazole