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—— 5-(4-methylphenyl)-2-[(2S)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O
5-(4-methylphenyl)-2-[(2S)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— [5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl 1H-indole-2-carboxylate —— C19H13ClN2O3
[5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl 1H-indole-2-carboxylate
—— 5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C19H21FN2O3
5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— 5-(4-methoxyphenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O2
5-(4-methoxyphenyl)-2-[(3S)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— 5-(4-methoxyphenyl)-2-[(2S)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O2
5-(4-methoxyphenyl)-2-[(2S)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— (5R)-N-(3-chloro-4-fluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H17ClFN5O4
(5R)-N-(3-chloro-4-fluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— 5-(4-methoxyphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C23H20N4O2
5-(4-methoxyphenyl)-2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-chloro-5-methylsulfonylbenzoate —— C17H15ClN2O6S
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-chloro-5-methylsulfonylbenzoate
—— (5R)-N-(3-fluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H18FN5O4
(5R)-N-(3-fluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-2-(4-methoxyanilino)-4,7-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H18F3N5O5
(5R)-2-(4-methoxyanilino)-4,7-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-N-(3,4-difluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H17F2N5O4
(5R)-N-(3,4-difluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-(2-methoxyanilino)-N-(3-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H21N5O5
(5S)-2-(2-methoxyanilino)-N-(3-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(2,4-dimethoxyphenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C23H23N5O6
(5S)-N-(2,4-dimethoxyphenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— 5-[3-[(3R)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C18H21FN2O4
5-[3-[(3R)-3-[(4-fluorophenoxy)methyl]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[2-(3,5-dimethylphenoxy)ethylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C15H19N3OS2
5-[2-(3,5-dimethylphenoxy)ethylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— (5S)-2-(2-methoxyanilino)-4,7-dioxo-N-(3,4,5-trimethoxyphenyl)-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C24H25N5O7
(5S)-2-(2-methoxyanilino)-4,7-dioxo-N-(3,4,5-trimethoxyphenyl)-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— 5-(4-methoxyphenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O2
5-(4-methoxyphenyl)-2-[(3R)-3-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— (5R)-N-(3-chloro-4-fluorophenyl)-2-(4-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H17ClFN5O4
(5R)-N-(3-chloro-4-fluorophenyl)-2-(4-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(2,5-dimethoxyphenyl)-2-(4-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C23H23N5O6
(5S)-N-(2,5-dimethoxyphenyl)-2-(4-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-2-(3,5-dichloroanilino)-N-(3-fluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C20H14Cl2FN5O3
(5R)-2-(3,5-dichloroanilino)-N-(3-fluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-(3,5-dichloroanilino)-4,7-dioxo-N-[3-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H14Cl2F3N5O3
(5S)-2-(3,5-dichloroanilino)-4,7-dioxo-N-[3-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— 5-[(6-bromo-1,3-benzodioxol-5-yl)methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C13H12BrN3O2S2
5-[(6-bromo-1,3-benzodioxol-5-yl)methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— (5S)-N-(3-methoxyphenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H18F3N5O4
(5S)-N-(3-methoxyphenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-N-(1,3-benzodioxol-5-yl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H19N5O6
(5R)-N-(1,3-benzodioxol-5-yl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— 5-(4-methoxyphenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one —— C20H22N4O2
5-(4-methoxyphenyl)-2-[(2R)-2-methylpiperidin-1-yl]-1H-pyrido[2,3-d]pyrimidin-4-one
—— (5R)-2-(4-methoxyanilino)-4,7-dioxo-N-[3-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H18F3N5O5
(5R)-2-(4-methoxyanilino)-4,7-dioxo-N-[3-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(3-fluorophenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H15F4N5O3
(5S)-N-(3-fluorophenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-2-(3,5-dichloroanilino)-N-(2-fluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C20H14Cl2FN5O3
(5R)-2-(3,5-dichloroanilino)-N-(2-fluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-N-(3-methoxyphenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H18F3N5O4
(5R)-N-(3-methoxyphenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-(3,5-dichloroanilino)-N-(3,4-difluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C20H13Cl2F2N5O3
(5S)-2-(3,5-dichloroanilino)-N-(3,4-difluorophenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-3-methyl-9-(2-methylquinolin-4-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H21N3O2
(5R)-3-methyl-9-(2-methylquinolin-4-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-2-(2-methoxyanilino)-4,7-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H18F3N5O5
(5R)-2-(2-methoxyanilino)-4,7-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-methyl-5-methylsulfonylbenzoate —— C19H16ClNO5S
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-methyl-5-methylsulfonylbenzoate
—— (5S)-2-(4-methoxyanilino)-N-(3-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H21N5O5
(5S)-2-(4-methoxyanilino)-N-(3-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-(2-methoxyanilino)-4,7-dioxo-N-[2-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H18F3N5O4
(5S)-2-(2-methoxyanilino)-4,7-dioxo-N-[2-(trifluoromethyl)phenyl]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— [5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl (E)-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)prop-2-enoate —— C22H18ClNO5
[5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl (E)-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)prop-2-enoate
—— (5R)-2-(3,5-dichloroanilino)-N-(2-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H17Cl2N5O4
(5R)-2-(3,5-dichloroanilino)-N-(2-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— 5-[[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine —— C14H12FN5OS2
5-[[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-prop-2-enyl-1,3,4-thiadiazol-2-amine
—— (5S)-3-methyl-7-[4-(tetrazol-1-yl)butanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H18N6O3
(5S)-3-methyl-7-[4-(tetrazol-1-yl)butanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-N-(3,4-difluorophenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H14F5N5O3
(5S)-N-(3,4-difluorophenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(4-fluorophenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H15F4N5O3
(5S)-N-(4-fluorophenyl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-N-(3-chloro-4-fluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H17ClFN5O4
(5S)-N-(3-chloro-4-fluorophenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-(4-methoxyanilino)-N-(4-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C22H21N5O5
(5S)-2-(4-methoxyanilino)-N-(4-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-2-(2-methoxyanilino)-4,7-dioxo-N-(3,4,5-trimethoxyphenyl)-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C24H25N5O7
(5R)-2-(2-methoxyanilino)-4,7-dioxo-N-(3,4,5-trimethoxyphenyl)-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— 5-[(2-chloro-7,8-dimethylquinolin-3-yl)methylsulfanyl]-N-(2-methoxyethyl)-1,3,4-thiadiazol-2-amine —— C17H19ClN4OS2
5-[(2-chloro-7,8-dimethylquinolin-3-yl)methylsulfanyl]-N-(2-methoxyethyl)-1,3,4-thiadiazol-2-amine
—— 5-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C19H24N6O2
5-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— (5S)-2-(3,5-dichloroanilino)-N-(4-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C21H17Cl2N5O4
(5S)-2-(3,5-dichloroanilino)-N-(4-methoxyphenyl)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5S)-2-[(2-butyl-1H-imidazol-5-yl)methyl]-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C24H40N4O
(5S)-2-[(2-butyl-1H-imidazol-5-yl)methyl]-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-N-(2,5-dimethoxyphenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C23H23N5O6
(5S)-N-(2,5-dimethoxyphenyl)-2-(2-methoxyanilino)-4,7-dioxo-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide
—— (5R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide —— C23H18F3N5O5
(5R)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4,7-dioxo-2-[3-(trifluoromethyl)anilino]-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-5-carboxamide