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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-chloro-N-[(3S)-1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-2-carboxamide —— C21H18ClN3O2
5-chloro-N-[(3S)-1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-2-carboxamide
—— 5-chloro-N-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-6-oxo-1H-pyridine-3-carboxamide —— C18H26ClN3O2
5-chloro-N-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-6-oxo-1H-pyridine-3-carboxamide
—— (5R)-9-(2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H23N3O4
(5R)-9-(2-oxo-5,6,7,8-tetrahydro-1H-quinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5R)-9-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-7-(5-propan-2-yl-1,2-oxazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H19N3O4
(5S)-3-methyl-7-(5-propan-2-yl-1,2-oxazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methyl-N-[(3S)-5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide —— C18H22N4O2
5-methyl-N-[(3S)-5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S)-9-(1-ethyl-3,5-dimethylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H24N4O3
(5S)-9-(1-ethyl-3,5-dimethylpyrazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-2-ethylsulfonyl-9-(2-phenylethyl)-2,9-diazaspiro[4.5]decane —— C18H28N2O2S
(5S)-2-ethylsulfonyl-9-(2-phenylethyl)-2,9-diazaspiro[4.5]decane
—— (5R)-9-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O4
(5R)-9-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C19H22N4O3
5-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-propyl-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H24N6
5-propyl-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[2-[(3R)-3-(3,4-dimethylanilino)piperidin-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione —— C20H26N4O3
5-[2-[(3R)-3-(3,4-dimethylanilino)piperidin-1-yl]-2-oxoethyl]-3-methyl-1H-pyrimidine-2,4-dione
—— 5-propyl-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H24N6
5-propyl-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-[3-(4,6-dimethyl-2-oxo-1H-pyrimidin-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H24N4O4
(5S)-9-[3-(4,6-dimethyl-2-oxo-1H-pyrimidin-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(5-phenoxyfuran-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H20N2O5
(5S)-9-(5-phenoxyfuran-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-7-(5-propan-2-yl-1,2-oxazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H19N3O4
(5R)-3-methyl-7-(5-propan-2-yl-1,2-oxazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(3R)-3-(4-fluoroanilino)piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C21H21FN4O2
5-[(3R)-3-(4-fluoroanilino)piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— (5-Methyl-1,3,4-oxadiazol-2-yl)methyl 2-(4-phenylphenyl)acetate —— C18H16N2O3
(5-Methyl-1,3,4-oxadiazol-2-yl)methyl 2-(4-phenylphenyl)acetate
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C20H23F2N5O
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— 5-chloro-N-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-6-oxo-1H-pyridine-3-carboxamide —— C18H26ClN3O2
5-chloro-N-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-6-oxo-1H-pyridine-3-carboxamide
—— (5R)-9-[3-(4,6-dimethyl-2-oxo-1H-pyrimidin-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H24N4O4
(5R)-9-[3-(4,6-dimethyl-2-oxo-1H-pyrimidin-5-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C19H22N4O3
5-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-phenylphenyl)acetate —— C21H16N2O4
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-phenylphenyl)acetate
—— (5R)-9-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H22N2O3
(5R)-9-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5-fluoro-1H-indol-2-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C23H24FN3O
(5-fluoro-1H-indol-2-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5S)-9-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5S)-9-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[3-[(3S)-3-(3-fluoroanilino)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C17H20FN3O3
5-[3-[(3S)-3-(3-fluoroanilino)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— 5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-pyrrolidin-3-yl]pyridin-2-amine —— C20H23N5O
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-pyrrolidin-3-yl]pyridin-2-amine
—— 5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-[(3R)-pyrrolidin-3-yl]pyridin-2-amine —— C20H23N5O
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-[(3R)-pyrrolidin-3-yl]pyridin-2-amine
—— (5-fluoro-1H-indol-2-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C23H24FN3O
(5-fluoro-1H-indol-2-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— 5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C20H23F2N5O
5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— (5S)-9-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H22N2O3
(5S)-9-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-methyl-N-[(3S)-1-[[4-(2-methylpropyl)phenyl]methyl]piperidin-3-yl]-1,2-oxazole-4-sulfonamide —— C20H29N3O3S
5-methyl-N-[(3S)-1-[[4-(2-methylpropyl)phenyl]methyl]piperidin-3-yl]-1,2-oxazole-4-sulfonamide
—— (5R)-3-methyl-7-[2-([1,2,4]triazolo[4,3-b]pyridazin-6-yloxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H16N6O4
(5R)-3-methyl-7-[2-([1,2,4]triazolo[4,3-b]pyridazin-6-yloxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H32N2O3
(5R)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-fluorophenyl)-N-[(1R)-2-methyl-1-(2-methyl-1,2,4-triazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H20FN7
5-(2-fluorophenyl)-N-[(1R)-2-methyl-1-(2-methyl-1,2,4-triazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(2-fluorophenyl)-N-[(1S)-2-methyl-1-(2-methyl-1,2,4-triazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H20FN7
5-(2-fluorophenyl)-N-[(1S)-2-methyl-1-(2-methyl-1,2,4-triazol-3-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H32N2O3
(5S)-2-(cyclobutylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(1-benzoxepine-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H20N2O4
(5R)-9-(1-benzoxepine-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— [5-(2-chlorophenyl)furan-2-yl]-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone —— C17H18ClNO4
[5-(2-chlorophenyl)furan-2-yl]-[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methanone
—— (5S)-3-methyl-7-[2-([1,2,4]triazolo[4,3-b]pyridazin-6-yloxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H16N6O4
(5S)-3-methyl-7-[2-([1,2,4]triazolo[4,3-b]pyridazin-6-yloxy)acetyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H17F3N4O2
(5S)-3-methyl-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H20N4O3
(5R)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-Bromo-1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]pyridin-2-one —— C15H12BrNO4
5-Bromo-1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]pyridin-2-one
—— (5S)-9-[2-(2,3-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H27NO3
(5S)-9-[2-(2,3-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-2-(1H-indole-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C23H24N4O2
(5R)-2-(1H-indole-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C21H29N3O3
5-[(3S)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-3-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3-propan-2-ylimidazol-4-yl)methyl]pyridazin-3-one —— C17H26N6O2
5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3-propan-2-ylimidazol-4-yl)methyl]pyridazin-3-one
—— (5R)-9-[2-(2,3-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H27NO3
(5R)-9-[2-(2,3-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[3-[(3R)-3-(3-fluoroanilino)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C17H20FN3O3
5-[3-[(3R)-3-(3-fluoroanilino)piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one