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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-1-butyl-5-(4-methoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C22H25N3O4
(5S)-1-butyl-5-(4-methoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— (5-fluoro-2-methoxyphenyl)-[4-[(3R)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone —— C18H25FN2O3
(5-fluoro-2-methoxyphenyl)-[4-[(3R)-3-hydroxypiperidin-1-yl]piperidin-1-yl]methanone
—— (5R)-3-methyl-9-[(4-methylsulfonylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H24N2O4S
(5R)-3-methyl-9-[(4-methylsulfonylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-2-[3-(1H-indol-3-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N3O2
(5S)-2-[3-(1H-indol-3-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(4R)-4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C17H24N4O3
5-[(4R)-4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5R)-9-[6-propan-2-yl-2-(trifluoromethyl)pyrimidin-4-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H21F3N4O2
(5R)-9-[6-propan-2-yl-2-(trifluoromethyl)pyrimidin-4-yl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-Amino-2-(3-hydroxyphenyl)-1,3-oxazole-4-carbonitrile —— C10H7N3O2
5-Amino-2-(3-hydroxyphenyl)-1,3-oxazole-4-carbonitrile
—— (5R)-1-butyl-5-(4-methoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C22H25N3O4
(5R)-1-butyl-5-(4-methoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— 5-ethyl-N-[4-[(2S)-oxolan-2-yl]butyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H24N4O
5-ethyl-N-[4-[(2S)-oxolan-2-yl]butyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5,6-dimethyl-2-[[(1S)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethyl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C17H16N4O2S3
5,6-dimethyl-2-[[(1S)-1-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)ethyl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5S)-7-[4-(diethylaminomethyl)-5-ethylfuran-2-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C19H29N3O4
(5S)-7-[4-(diethylaminomethyl)-5-ethylfuran-2-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(3-methyl-4-oxoquinazoline-7-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H20N4O4
(5S)-9-(3-methyl-4-oxoquinazoline-7-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H28N2O5
(5S)-9-[3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]pyridine-2-carbonitrile —— C21H22N4O
5-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazine-1-carbonyl]pyridine-2-carbonitrile
—— (5R)-2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H28N2O4
(5R)-2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1H-imidazol-5-ylmethyl)-7-(3-methylbut-2-enyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H28N6O
(5R)-5-(1H-imidazol-5-ylmethyl)-7-(3-methylbut-2-enyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— (5R)-9-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22N4O4
(5R)-9-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22N4O4
(5S)-9-[2-(4-methyl-1-oxophthalazin-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H23F2N3O2
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-ethyl-N-[4-[(2R)-oxolan-2-yl]butyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H24N4O
5-ethyl-N-[4-[(2R)-oxolan-2-yl]butyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-methoxy-3-methyl-N-quinolin-8-yl-1-benzofuran-2-carboxamide —— C20H16N2O3
5-methoxy-3-methyl-N-quinolin-8-yl-1-benzofuran-2-carboxamide
—— (5R)-9-[3-(4-oxoquinazolin-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20N4O4
(5R)-9-[3-(4-oxoquinazolin-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H23F2N3O2
5-[[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (5R)-9-[3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H28N2O5
(5R)-9-[3-(3,4-dimethoxyphenyl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H18ClN5O3
(5R)-9-(3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H24N2O3S
(5R)-3-methyl-9-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3,5-dimethylphenyl)methyl]pyridazin-3-one —— C19H26N4O2
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[(3,5-dimethylphenyl)methyl]pyridazin-3-one
—— 5-[3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl]-N-[(3S)-pyrrolidin-3-yl]pyridin-2-amine —— C19H21N5O2
5-[3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl]-N-[(3S)-pyrrolidin-3-yl]pyridin-2-amine
—— (5R)-7-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O4
(5R)-7-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N2O6
(5R)-9-[2-(1,3-benzodioxol-5-yloxy)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C20H24N2O3S
(5R)-9-[[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C18H21N3O3
(5S)-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-3-methyl-7-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H21N3O3
(5R)-3-methyl-7-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C13H16ClN3O4
(5S)-7-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[(1-ethylimidazol-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H23N3O2
(5R)-9-[(1-ethylimidazol-2-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N4O4
(5S)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[2-[(dimethylamino)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C19H29N7O
5-[[2-[(dimethylamino)methyl]-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-5-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (5R)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N4O4
(5R)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H18N4O4
(5S)-7-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-5-(1H-imidazol-5-ylmethyl)-7-(3-methylbut-2-enyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H28N6O
(5S)-5-(1H-imidazol-5-ylmethyl)-7-(3-methylbut-2-enyl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— (5R)-3-methyl-9-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H22N4O3
(5R)-3-methyl-9-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H21N3O3S
(5R)-9-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-chloro-N-[(3R)-1-(1-methylpiperidin-4-yl)piperidin-3-yl]thiophene-2-sulfonamide —— C15H24ClN3O2S2
5-chloro-N-[(3R)-1-(1-methylpiperidin-4-yl)piperidin-3-yl]thiophene-2-sulfonamide
—— 5-[3-[2-[(4S)-2,2-dimethyloxan-4-yl]imidazol-1-yl]propyl]-2H-tetrazole —— C14H22N6O
5-[3-[2-[(4S)-2,2-dimethyloxan-4-yl]imidazol-1-yl]propyl]-2H-tetrazole
—— (5R)-3-methyl-7-[1-methyl-3-(trifluoromethyl)thieno[2,3-c]pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H15F3N4O3S
(5R)-3-methyl-7-[1-methyl-3-(trifluoromethyl)thieno[2,3-c]pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(4-methoxy-2-methylbenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H22N2O4
(5S)-9-(4-methoxy-2-methylbenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-cyano-6-(ethylsulfanyl)-2-methyl-N-(2-methylphenyl)-4-(thiophen-2-yl)pyridine-3-carboxamide —— C21H19N3OS2
5-cyano-6-(ethylsulfanyl)-2-methyl-N-(2-methylphenyl)-4-(thiophen-2-yl)pyridine-3-carboxamide
—— (5S)-9-[[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C20H24N2O3S
(5S)-9-[[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-3-methyl-7-[1-methyl-3-(trifluoromethyl)thieno[2,3-c]pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H15F3N4O3S
(5S)-3-methyl-7-[1-methyl-3-(trifluoromethyl)thieno[2,3-c]pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methoxy-3-methyl-2-[[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1H-indole —— C22H27N3O2
5-methoxy-3-methyl-2-[[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1H-indole