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—— (5-Hydroxypyridin-3-yl)-[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-piperidin-1-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C24H28N6O3
(5-Hydroxypyridin-3-yl)-[4-[5-(3-methyl-1,2-oxazol-5-yl)-2-piperidin-1-ylpyrimidin-4-yl]piperidin-1-yl]methanone
—— 5-methylsulfonyl-4-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]-2-pyridin-3-ylpyrimidine —— C20H26N4O3S
5-methylsulfonyl-4-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]-2-pyridin-3-ylpyrimidine
—— 5-tert-butyl-3-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C21H32N6O3
5-tert-butyl-3-[1-[(1R,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— (5-tert-butyl-2-methylpyrazol-3-yl)-[(3R)-3-hydroxy-3-(1,3-thiazol-2-yl)-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone —— C20H28N4O3S
(5-tert-butyl-2-methylpyrazol-3-yl)-[(3R)-3-hydroxy-3-(1,3-thiazol-2-yl)-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone
—— 5-Phenyl-7-(1,3-thiazol-4-ylmethyl)-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C18H16N6OS
5-Phenyl-7-(1,3-thiazol-4-ylmethyl)-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 5-tert-butyl-3-[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C21H32N6O3
5-tert-butyl-3-[1-[(1S,3R)-3-methoxycyclohexanecarbonyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-methyl-3-[1-(2-phenylacetyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C18H20N6O2
5-methyl-3-[1-(2-phenylacetyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-Methylsulfonyl-4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-2-pyrrolidin-1-ylpyrimidine —— C20H27N5O2S
5-Methylsulfonyl-4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-2-pyrrolidin-1-ylpyrimidine
—— (5-methyl-1H-pyrazol-4-yl)-[4-(5-methylsulfonyl-2-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone —— C19H26N6O3S
(5-methyl-1H-pyrazol-4-yl)-[4-(5-methylsulfonyl-2-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone
—— 5-Phenyl-7-(pyridin-2-ylmethyl)-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C20H18N6O
5-Phenyl-7-(pyridin-2-ylmethyl)-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— (5-tert-butyl-2-methylpyrazol-3-yl)-[(3S)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone —— C23H30FN3O3
(5-tert-butyl-2-methylpyrazol-3-yl)-[(3S)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone
—— 5-tert-butyl-3-[1-(thiophene-2-carbonyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C18H22N6O2S
5-tert-butyl-3-[1-(thiophene-2-carbonyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone —— C22H28FN3O3
(5-tert-butyl-1H-pyrazol-3-yl)-[(3S)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone —— C22H28FN3O3
(5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone
—— (5-bromothiophen-2-yl)-[(3R)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone —— C19H19BrFNO3S
(5-bromothiophen-2-yl)-[(3R)-3-(4-fluorophenyl)-3-hydroxy-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone
—— (5-tert-butyl-2-methylpyrazol-3-yl)-[(3S)-3-hydroxy-3-(1,3-thiazol-2-yl)-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone —— C20H28N4O3S
(5-tert-butyl-2-methylpyrazol-3-yl)-[(3S)-3-hydroxy-3-(1,3-thiazol-2-yl)-1-oxa-8-azaspiro[4.5]decan-8-yl]methanone
—— (5S,7R)-7-[4-(difluoromethoxy)phenyl]-5-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine —— C17H15F2N5O
(5S,7R)-7-[4-(difluoromethoxy)phenyl]-5-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine
—— 5-amino-4-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-1-[[(2R)-oxolan-2-yl]methyl]-2H-pyrrol-3-one —— C19H21N3O2S
5-amino-4-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-1-[[(2R)-oxolan-2-yl]methyl]-2H-pyrrol-3-one
—— (5R,7R)-7-[4-(difluoromethoxy)phenyl]-5-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine —— C17H15F2N5O
(5R,7R)-7-[4-(difluoromethoxy)phenyl]-5-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine
—— 5-bromo-2-chloro-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]benzamide —— C16H13BrClNO3
5-bromo-2-chloro-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]benzamide
—— 5-[(3R)-3-[3-(furan-2-yl)-6-oxopyridazin-1-yl]piperidine-1-carbonyl]-1,3-dimethylbenzimidazol-2-one —— C23H23N5O4
5-[(3R)-3-[3-(furan-2-yl)-6-oxopyridazin-1-yl]piperidine-1-carbonyl]-1,3-dimethylbenzimidazol-2-one
—— (5S,7R)-3-chloro-N-methyl-N-[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]adamantane-1-carboxamide —— C20H22ClF3N2O2
(5S,7R)-3-chloro-N-methyl-N-[2-oxo-2-(2,3,4-trifluoroanilino)ethyl]adamantane-1-carboxamide
—— (5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]methanone —— C19H22F3N7O
(5-tert-butyl-1H-pyrazol-3-yl)-[(3R)-3-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]methanone
—— (5-tert-butyl-1H-pyrazol-3-yl)-[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]methanone —— C19H22F3N7O
(5-tert-butyl-1H-pyrazol-3-yl)-[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]piperidin-1-yl]methanone
—— (5-Cyclopropyl-2-methylfuran-3-yl)-[4-(6-methylsulfonyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone —— C20H23N5O4S
(5-Cyclopropyl-2-methylfuran-3-yl)-[4-(6-methylsulfonyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
—— [5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone —— C19H17F3N8O
[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3R)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
—— [5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone —— C19H17F3N8O
[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]-[(3S)-3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
—— (5S)-N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H20N2O2S2
(5S)-N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S,7S)-7-[4-(difluoromethoxy)phenyl]-5-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine —— C17H15F2N5O
(5S,7S)-7-[4-(difluoromethoxy)phenyl]-5-phenyl-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine
—— [5-(Furan-2-yl)-2-sulfanylidene-1,3,4-oxadiazol-3-yl]methyl-[(4-methoxyphenyl)methyl]-methylazanium —— C16H18N3O3S+
[5-(Furan-2-yl)-2-sulfanylidene-1,3,4-oxadiazol-3-yl]methyl-[(4-methoxyphenyl)methyl]-methylazanium
—— (5R)-N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H20N2O2S2
(5R)-N-(5-acetyl-4-methyl-1,3-thiazol-2-yl)-5-ethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(5Z)-5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoate —— C20H22NO5S2-
5-[(5Z)-5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoate
—— 5-[(5Z)-5-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoic acid —— C20H23NO5S2
5-[(5Z)-5-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoic acid
—— (5Z)-2-(3H-1,3-benzothiazol-2-ylidenemethyl)-5-[(3-ethoxy-4-methoxyphenyl)methylidene]-1,3-thiazol-4-one —— C21H18N2O3S2
(5Z)-2-(3H-1,3-benzothiazol-2-ylidenemethyl)-5-[(3-ethoxy-4-methoxyphenyl)methylidene]-1,3-thiazol-4-one
—— 5-[(5Z)-5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoic acid —— C20H23NO5S2
5-[(5Z)-5-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoic acid
—— (5R)-1-butyl-5-(3,5-dimethoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C23H27N3O5
(5R)-1-butyl-5-(3,5-dimethoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— (5R,5aS)-3-methyl-1-phenyl-5,5a,6,7,8,9-hexahydro-4H-pyrazolo[4,3-c]quinolizine-5-carboxylic acid —— C18H21N3O2
(5R,5aS)-3-methyl-1-phenyl-5,5a,6,7,8,9-hexahydro-4H-pyrazolo[4,3-c]quinolizine-5-carboxylic acid
—— 5-[(5Z)-5-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoate —— C20H22NO5S2-
5-[(5Z)-5-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]pentanoate
—— (5R)-1-methyl-5-(2-methylphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C19H19N3O3
(5R)-1-methyl-5-(2-methylphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— 5,6-dimethyl-2-[(3S)-1-(2-thiophen-3-ylacetyl)piperidin-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one —— C19H21N3O2S2
5,6-dimethyl-2-[(3S)-1-(2-thiophen-3-ylacetyl)piperidin-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-[(3S)-3-[3-(furan-2-yl)-6-oxopyridazin-1-yl]piperidine-1-carbonyl]-1,3-dimethylbenzimidazol-2-one —— C23H23N5O4
5-[(3S)-3-[3-(furan-2-yl)-6-oxopyridazin-1-yl]piperidine-1-carbonyl]-1,3-dimethylbenzimidazol-2-one
—— 5,6-dimethyl-2-[(3R)-1-(2-thiophen-3-ylacetyl)piperidin-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one —— C19H21N3O2S2
5,6-dimethyl-2-[(3R)-1-(2-thiophen-3-ylacetyl)piperidin-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5R)-1-ethyl-5-thiophen-2-yl-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C17H17N3O3S
(5R)-1-ethyl-5-thiophen-2-yl-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— 5-pyridin-4-yl-4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidine —— C20H21N5
5-pyridin-4-yl-4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidine
—— [5-ethyl-4-(morpholin-4-ylmethyl)furan-2-yl]-[4-(4-pyridin-4-yl-1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C25H31N5O3
[5-ethyl-4-(morpholin-4-ylmethyl)furan-2-yl]-[4-(4-pyridin-4-yl-1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— (5R)-1-butyl-5-(4-ethoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C23H27N3O4
(5R)-1-butyl-5-(4-ethoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— (5S)-5-(4-ethoxyphenyl)-1-propyl-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C22H25N3O4
(5S)-5-(4-ethoxyphenyl)-1-propyl-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— (5E)-5-[[2-(1,3-benzothiazol-2-yl)hydrazinyl]methylidene]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C15H15N5O3S2
(5E)-5-[[2-(1,3-benzothiazol-2-yl)hydrazinyl]methylidene]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-1-butyl-5-(4-ethoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione —— C23H27N3O4
(5S)-1-butyl-5-(4-ethoxyphenyl)-7,8,9,10-tetrahydro-5H-pyrimido[4,5-b]quinoline-2,4,6-trione
—— (5Z)-5-[[2-(4,6-dimethylpyrimidin-2-yl)hydrazinyl]methylidene]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C14H18N6O3S
(5Z)-5-[[2-(4,6-dimethylpyrimidin-2-yl)hydrazinyl]methylidene]-1-(2-methoxyethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione