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—— 5-[[2-[(2-Chlorophenyl)methyl]pyrazol-3-yl]amino]-5-oxopentanoic acid —— C15H16ClN3O3
5-[[2-[(2-Chlorophenyl)methyl]pyrazol-3-yl]amino]-5-oxopentanoic acid
—— 5-[[2-[(2-Chlorophenyl)methyl]pyrazol-3-yl]amino]-5-oxopentanoate —— C15H15ClN3O3-
5-[[2-[(2-Chlorophenyl)methyl]pyrazol-3-yl]amino]-5-oxopentanoate
—— 5-bromo-N-[2-[[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl]-N-ethylthiophene-2-carboxamide —— C13H17BrN2O4S2
5-bromo-N-[2-[[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl]-N-ethylthiophene-2-carboxamide
—— [5-[[[(3S,4S)-3-methyl-1-propan-2-ylsulfonylpiperidin-4-yl]amino]methyl]furan-2-yl]methanol —— C15H26N2O4S
[5-[[[(3S,4S)-3-methyl-1-propan-2-ylsulfonylpiperidin-4-yl]amino]methyl]furan-2-yl]methanol
—— 5-[(4-Methoxyphenyl)methylamino]-5-oxopentanoic acid —— C13H17NO4
5-[(4-Methoxyphenyl)methylamino]-5-oxopentanoic acid
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C15H21ClN4O2
(5-chloro-2-methylpyrimidin-4-yl)-[(3S,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5R)-5-[(3S)-1-[(5-butyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl]-5-methylimidazolidine-2,4-dione —— C16H25N5O3
(5R)-5-[(3S)-1-[(5-butyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl]-5-methylimidazolidine-2,4-dione
—— [5-[[[(3R,4S)-3-methyl-1-propan-2-ylsulfonylpiperidin-4-yl]amino]methyl]furan-2-yl]methanol —— C15H26N2O4S
[5-[[[(3R,4S)-3-methyl-1-propan-2-ylsulfonylpiperidin-4-yl]amino]methyl]furan-2-yl]methanol
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3S,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C17H24N6O2
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3S,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3S,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C17H24N6O2
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3S,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5-ethyl-1,3-oxazol-4-yl)-[(3S,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C15H23N3O3
(5-ethyl-1,3-oxazol-4-yl)-[(3S,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5-ethyl-1,3-oxazol-4-yl)-[(3R,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C15H23N3O3
(5-ethyl-1,3-oxazol-4-yl)-[(3R,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C15H21ClN4O2
(5-chloro-2-methylpyrimidin-4-yl)-[(3S,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C15H21ClN4O2
(5-chloro-2-methylpyrimidin-4-yl)-[(3R,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5-ethyl-1,3-oxazol-4-yl)-[(3S,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C15H23N3O3
(5-ethyl-1,3-oxazol-4-yl)-[(3S,4R)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (5-ethyl-1,3-oxazol-4-yl)-[(3R,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C15H23N3O3
(5-ethyl-1,3-oxazol-4-yl)-[(3R,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— 5-chloro-N-[2-[4-(trifluoromethyl)phenyl]ethyl]thiophene-2-sulfonamide —— C13H11ClF3NO2S2
5-chloro-N-[2-[4-(trifluoromethyl)phenyl]ethyl]thiophene-2-sulfonamide
—— (5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3R,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C17H24N6O2
(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[(3R,4S)-3-methyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— 5-propan-2-yl-3-[(3S)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C15H19N7O
5-propan-2-yl-3-[(3S)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— (5-Methyl-1,2-oxazol-3-yl)[4-(phenylsulfonyl)piperazin-1-yl]methanone —— C15H17N3O4S
(5-Methyl-1,2-oxazol-3-yl)[4-(phenylsulfonyl)piperazin-1-yl]methanone
—— 5-[[(3S,8aR)-3-ethyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]isoquinoline —— C18H23N3O2S
5-[[(3S,8aR)-3-ethyl-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]isoquinoline
—— 5-cyclopropyl-3-[(2S)-1-(1,2-oxazol-5-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole —— C13H16N4O2
5-cyclopropyl-3-[(2S)-1-(1,2-oxazol-5-ylmethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-propan-2-yl-3-[(3S)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C18H26N6O
5-propan-2-yl-3-[(3S)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3R)-1-(6-fluoroquinazolin-4-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C17H18FN5O
5-ethyl-3-[(3R)-1-(6-fluoroquinazolin-4-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-methyl-3-[(3R)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C13H15N7O
5-methyl-3-[(3R)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3S)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C14H17N7O
5-ethyl-3-[(3S)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3R)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C14H17N7O
5-ethyl-3-[(3R)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3S)-1-(6-fluoroquinazolin-4-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C17H18FN5O
5-ethyl-3-[(3S)-1-(6-fluoroquinazolin-4-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-methyl-3-[(3S)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C13H15N7O
5-methyl-3-[(3S)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-(2-fluorophenyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)furan-2-carboxamide —— C14H10FN3O2S
5-(2-fluorophenyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)furan-2-carboxamide
—— 5-ethyl-3-[(3R)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]-1,2,4-oxadiazole —— C15H17F3N4O
5-ethyl-3-[(3R)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-propan-2-yl-3-[(3R)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C15H19N7O
5-propan-2-yl-3-[(3R)-1-(7H-purin-6-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3S)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C17H24N6O
5-ethyl-3-[(3S)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3R)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C17H24N6O
5-ethyl-3-[(3R)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2S)-1-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C14H18N4O2
5-cyclopropyl-3-[(2S)-1-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2R)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C16H22N4O2
5-cyclopropyl-3-[(2R)-1-[(5-propan-2-yl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2R)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C14H19N5O2
5-cyclopropyl-3-[(2R)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-propan-2-yl-3-[(3R)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C18H26N6O
5-propan-2-yl-3-[(3R)-1-(4-pyrrolidin-1-ylpyrimidin-2-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2S)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C14H19N5O2
5-cyclopropyl-3-[(2S)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— (5S)-5-benzyl-3-[(1-butyltetrazol-5-yl)methyl]-5-phenylimidazolidine-2,4-dione —— C22H24N6O2
(5S)-5-benzyl-3-[(1-butyltetrazol-5-yl)methyl]-5-phenylimidazolidine-2,4-dione
—— 5-cyclopropyl-3-[(2R)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C14H18N4O2
5-cyclopropyl-3-[(2R)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]-1,2,4-oxadiazole —— C15H17F3N4O
5-ethyl-3-[(3S)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2S)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C14H18N4O2
5-cyclopropyl-3-[(2S)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2R)-1-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C15H21N5O2
5-cyclopropyl-3-[(2R)-1-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2R)-1-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C15H18F3N5O
5-cyclopropyl-3-[(2R)-1-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2R)-1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C15H20N4O2
5-cyclopropyl-3-[(2R)-1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2R)-1-[[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C16H23N5O2
5-cyclopropyl-3-[(2R)-1-[[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2S)-1-[[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C16H23N5O2
5-cyclopropyl-3-[(2S)-1-[[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2S)-1-(2-ethylsulfonylethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole —— C13H21N3O3S
5-cyclopropyl-3-[(2S)-1-(2-ethylsulfonylethyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2S)-1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C15H20N4O2
5-cyclopropyl-3-[(2S)-1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole