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—— (5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H24N2O4S2
(5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R)-3-methyl-9-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C12H18N4O2S
(5R)-3-methyl-9-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C12H18N4O2S
(5S)-3-methyl-9-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5Z)-5-[(2-fluorophenyl)methylidene]-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C19H21FN2O4S
(5Z)-5-[(2-fluorophenyl)methylidene]-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— (5S)-5-(4-hydroxyphenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C19H15N3O3
(5S)-5-(4-hydroxyphenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— 5-[(3R)-3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C23H28N2O3
5-[(3R)-3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5Z)-3-[(2S)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one —— C18H22N2O3S3
(5Z)-3-[(2S)-1-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one
—— (5R)-9-(2-ethoxypyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H19N3O4
(5R)-9-(2-ethoxypyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(furan-2-yl)-3-[[(2R)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C19H19N5O2
5-(furan-2-yl)-3-[[(2R)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5Z)-5-[(4-fluorophenyl)methylidene]-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H21FN2O3S2
(5Z)-5-[(4-fluorophenyl)methylidene]-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R)-3-methyl-9-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H21N3O3S
(5R)-3-methyl-9-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[3-(2-methoxyphenoxy)propyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H26N2O4
(5R)-9-[3-(2-methoxyphenoxy)propyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-N-(2,5-dimethoxyphenyl)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H17FN2O4
(5S)-N-(2,5-dimethoxyphenyl)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-3-methyl-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H24N4O2
(5R)-3-methyl-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5Z)-5-[(5-chloro-8-methoxyquinolin-2-yl)methylidene]-3-phenyl-2-thioxoimidazolidin-4-one —— C20H14ClN3O2S
(5Z)-5-[(5-chloro-8-methoxyquinolin-2-yl)methylidene]-3-phenyl-2-thioxoimidazolidin-4-one
—— (5Z)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H24N2O4S2
(5Z)-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(3-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[(3S)-3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one —— C23H28N2O3
5-[(3S)-3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]-2-methyl-1H-pyridin-4-one
—— (5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(3-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C21H26N2O5S
(5Z)-3-[3-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-5-[(3-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— 5-[(3R)-2-oxospiro[1H-indole-3,3'-piperidine]-1'-carbonyl]pyridine-2-carbonitrile —— C19H16N4O2
5-[(3R)-2-oxospiro[1H-indole-3,3'-piperidine]-1'-carbonyl]pyridine-2-carbonitrile
—— (5R)-3-methyl-9-(pyrazolo[1,5-a]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O3
(5R)-3-methyl-9-(pyrazolo[1,5-a]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-4-amino-3-[2-(diethylamino)ethyl]-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C23H27N4O2+
(5R)-4-amino-3-[2-(diethylamino)ethyl]-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— 5-cyano-N-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-2-methyl-6-oxo-1H-pyridine-3-carboxamide —— C20H28N4O2
5-cyano-N-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-2-methyl-6-oxo-1H-pyridine-3-carboxamide
—— (5R)-3-methyl-7-[3-(2-methylimidazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H22N4O2
(5R)-3-methyl-7-[3-(2-methylimidazol-1-yl)propyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[2-(2H-tetrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H16N6O3
(5S)-9-[2-(2H-tetrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-4-amino-5-(2-chlorophenyl)-3-[2-(dimethylamino)ethyl]-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C21H22ClN4O2+
(5S)-4-amino-5-(2-chlorophenyl)-3-[2-(dimethylamino)ethyl]-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— (5S)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-prop-2-enoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H20N2O5
(5S)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-prop-2-enoxyphenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5Z)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethylidene)-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C13H11NO3S2
(5Z)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethylidene)-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-benzylidene-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H22N2O3S2
(5Z)-5-benzylidene-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(furan-2-yl)-3-[[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C19H19N5O2
5-(furan-2-yl)-3-[[(2S)-2-(6-methyl-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5Z)-5-[(2-fluorophenyl)methylidene]-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C19H21FN2O4S
(5Z)-5-[(2-fluorophenyl)methylidene]-3-[2-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— (5R)-9-[2-(2H-tetrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H16N6O3
(5R)-9-[2-(2H-tetrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-fluoro-3-methyl-2-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-indole —— C19H20FN3
5-fluoro-3-methyl-2-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1H-indole
—— [5-[[(6S)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]methyl]-2-ethoxyphenyl]methanol —— C18H28N2O4
[5-[[(6S)-1,11-dioxa-4,8-diazaspiro[5.6]dodecan-4-yl]methyl]-2-ethoxyphenyl]methanol
—— (5S)-9-[3-(4-ethylphenyl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H24N2O3
(5S)-9-[3-(4-ethylphenyl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[3-(4-ethylphenyl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H24N2O3
(5R)-9-[3-(4-ethylphenyl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-cyano-N-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-2-methyl-6-oxo-1H-pyridine-3-carboxamide —— C20H28N4O2
5-cyano-N-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-2-methyl-6-oxo-1H-pyridine-3-carboxamide
—— (5R)-N-(2,5-dimethoxyphenyl)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C18H17FN2O4
(5R)-N-(2,5-dimethoxyphenyl)-3-(4-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-methoxy-2-[[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1H-pyridin-4-one —— C21H25F3N2O2
5-methoxy-2-[[(3R)-3-[2-[2-(trifluoromethyl)phenyl]ethyl]piperidin-1-yl]methyl]-1H-pyridin-4-one
—— 5-bromo-N-(3-(((1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl)amino)-3-oxopropyl)furan-2-carboxamide —— C15H17BrN4O5
5-bromo-N-(3-(((1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl)amino)-3-oxopropyl)furan-2-carboxamide
—— (5S)-9-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H21N5O3
(5S)-9-[3-(benzotriazol-1-yl)propanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(2-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H24N2O4S2
(5Z)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-5-[(2-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-3-methyl-9-(pyrazolo[1,5-a]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N4O3
(5S)-3-methyl-9-(pyrazolo[1,5-a]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-ethyl-N-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1H-pyrazole-4-carboxamide —— C17H24N6O3
5-ethyl-N-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1H-pyrazole-4-carboxamide
—— (5S)-3-methyl-9-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H21N3O3S
(5S)-3-methyl-9-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(2,2-dimethylpropyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,9-diazaspiro[4.5]decane —— C18H32N4O2S
(5R)-9-(2,2-dimethylpropyl)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,9-diazaspiro[4.5]decane
—— (5S)-9-(quinolin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H22N2O2
(5S)-9-(quinolin-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-3-methyl-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H24N4O2
(5S)-3-methyl-9-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5E)-5-benzylidene-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-1,3-thiazolidine-2,4-dione —— C20H24N2O4S
(5E)-5-benzylidene-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-1,3-thiazolidine-2,4-dione
—— (5Z)-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one —— C18H22N2O3S3
(5Z)-3-[3-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropyl]-2-sulfanylidene-5-(thiophen-2-ylmethylidene)-1,3-thiazolidin-4-one
—— (5Z)-5-(furan-2-ylmethylidene)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C17H20N2O5S
(5Z)-5-(furan-2-ylmethylidene)-3-[2-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione