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—— 5-[(2-fluorophenyl)methyl]-2-[(3S)-1-methylsulfonylpiperidin-3-yl]pyridine —— C18H21FN2O2S
5-[(2-fluorophenyl)methyl]-2-[(3S)-1-methylsulfonylpiperidin-3-yl]pyridine
—— 5-[[3-(3-chloroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one —— C23H24ClN5O2
5-[[3-(3-chloroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one
—— 5-[[3-(3-Fluoroanilino)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one —— C23H25FN6O
5-[[3-(3-Fluoroanilino)-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one
—— 5-bromo-N-[[2-[(dimethylamino)methyl]phenyl]methyl]pyridine-3-carboxamide —— C16H18BrN3O
5-bromo-N-[[2-[(dimethylamino)methyl]phenyl]methyl]pyridine-3-carboxamide
—— 5-[(3S)-1-(3-fluorophenyl)-5-oxopyrrolidin-3-yl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H14FN5O3
5-[(3S)-1-(3-fluorophenyl)-5-oxopyrrolidin-3-yl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[[3-(3-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-3H-1,3-benzoxazol-2-one —— C20H17FN4O3
5-[[3-(3-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-3H-1,3-benzoxazol-2-one
—— [5-[[(3R)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol —— C26H33N5O2
[5-[[(3R)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol
—— 5-methyl-3-[2-[(2R)-2-[5-[(3-methylpyridin-2-yl)amino]pyridin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]-1,3-benzoxazol-2-one —— C25H25N5O3
5-methyl-3-[2-[(2R)-2-[5-[(3-methylpyridin-2-yl)amino]pyridin-2-yl]pyrrolidin-1-yl]-2-oxoethyl]-1,3-benzoxazol-2-one
—— 5-[(3S)-1-naphthalen-1-yl-5-oxopyrrolidin-3-yl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H17N5O3
5-[(3S)-1-naphthalen-1-yl-5-oxopyrrolidin-3-yl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5-methoxy-1,3-dimethylindol-2-yl)-[(2R)-2-[5-(pyrazin-2-ylamino)pyridin-2-yl]pyrrolidin-1-yl]methanone —— C25H26N6O2
(5-methoxy-1,3-dimethylindol-2-yl)-[(2R)-2-[5-(pyrazin-2-ylamino)pyridin-2-yl]pyrrolidin-1-yl]methanone
—— 5-bromo-2-chloro-N-[[2-[(dimethylamino)methyl]phenyl]methyl]benzamide —— C17H18BrClN2O
5-bromo-2-chloro-N-[[2-[(dimethylamino)methyl]phenyl]methyl]benzamide
—— 5-[(2-fluorophenyl)methyl]-2-[(3R)-1-methylsulfonylpiperidin-3-yl]pyridine —— C18H21FN2O2S
5-[(2-fluorophenyl)methyl]-2-[(3R)-1-methylsulfonylpiperidin-3-yl]pyridine
—— [5-[(2S)-piperidin-2-yl]-1H-pyrazol-4-yl]-pyrrolidin-1-ylmethanone —— C13H20N4O
[5-[(2S)-piperidin-2-yl]-1H-pyrazol-4-yl]-pyrrolidin-1-ylmethanone
—— [5-[[(3S)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol —— C26H33N5O2
[5-[[(3S)-3-[6-(dimethylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]methyl]-2-ethoxyphenyl]methanol
—— [5-[(2R)-piperidin-2-yl]-1H-pyrazol-4-yl]-pyrrolidin-1-ylmethanone —— C13H20N4O
[5-[(2R)-piperidin-2-yl]-1H-pyrazol-4-yl]-pyrrolidin-1-ylmethanone
—— 5-(2H-benzotriazol-5-ylmethyl)-N-(3-fluorophenyl)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-3-amine —— C19H17FN6O
5-(2H-benzotriazol-5-ylmethyl)-N-(3-fluorophenyl)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-3-amine
—— [5-[4-(2,3-Dihydro-1-benzofuran-5-ylmethyl)piperazin-4-ium-1-yl]-5-oxopentyl]urea —— C19H29N4O3+
[5-[4-(2,3-Dihydro-1-benzofuran-5-ylmethyl)piperazin-4-ium-1-yl]-5-oxopentyl]urea
—— 5-[[3-(3,5-difluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one —— C23H23F2N5O2
5-[[3-(3,5-difluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one
—— (5-Chloro-1-benzofuran-2-yl)-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]methanone —— C22H21ClN2O3
(5-Chloro-1-benzofuran-2-yl)-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]methanone
—— 5-[2-[4-(2,3-Dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]-2-oxoethyl]-2,3-dihydro-1,5-benzoxazepin-4-one —— C24H27N3O4
5-[2-[4-(2,3-Dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]-2-oxoethyl]-2,3-dihydro-1,5-benzoxazepin-4-one
—— (5-Chloro-2-methoxyphenyl)-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]methanone —— C21H23ClN2O3
(5-Chloro-2-methoxyphenyl)-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]methanone
—— (5-Chlorothiophen-2-yl)-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]methanone —— C18H19ClN2O2S
(5-Chlorothiophen-2-yl)-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]methanone
—— 5-[3-(4-Methoxyphenoxy)propylsulfanyl]-1-(4-methoxyphenyl)tetrazole —— C18H20N4O3S
5-[3-(4-Methoxyphenoxy)propylsulfanyl]-1-(4-methoxyphenyl)tetrazole
—— (5S,7R)-3-chloro-N-[2-oxo-2-[2-(1H-pyrrole-2-carbonyl)hydrazinyl]ethyl]adamantane-1-carboxamide —— C18H23ClN4O3
(5S,7R)-3-chloro-N-[2-oxo-2-[2-(1H-pyrrole-2-carbonyl)hydrazinyl]ethyl]adamantane-1-carboxamide
—— 5-chloro-N-methyl-N-[2-oxo-2-[2-(1H-pyrrole-2-carbonyl)hydrazinyl]ethyl]thiophene-2-sulfonamide —— C12H13ClN4O4S2
5-chloro-N-methyl-N-[2-oxo-2-[2-(1H-pyrrole-2-carbonyl)hydrazinyl]ethyl]thiophene-2-sulfonamide
—— 5-[(3R)-1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-7-oxo-N-phenyl-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H18FN5O3
5-[(3R)-1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-7-oxo-N-phenyl-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[(3S)-1-(2-methylphenyl)-5-oxopyrrolidin-3-yl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H17N5O3
5-[(3S)-1-(2-methylphenyl)-5-oxopyrrolidin-3-yl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5Z)-3-(3,5-dimethylphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[[(2R)-oxolan-2-yl]methylsulfanyl]imidazol-4-one —— C24H26N2O3S
(5Z)-3-(3,5-dimethylphenyl)-5-[(4-methoxyphenyl)methylidene]-2-[[(2R)-oxolan-2-yl]methylsulfanyl]imidazol-4-one
—— 5-chloro-N-[5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pentyl]thiophene-2-carboxamide —— C19H20ClN3O3S
5-chloro-N-[5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pentyl]thiophene-2-carboxamide
—— 5-chloro-N-[2-(cyclopropylamino)-2-oxoethyl]-1-benzofuran-2-carboxamide —— C14H13ClN2O3
5-chloro-N-[2-(cyclopropylamino)-2-oxoethyl]-1-benzofuran-2-carboxamide
—— 5-bromo-N'-(1H-pyrrole-2-carbonyl)pyridine-3-carbohydrazide —— C11H9BrN4O2
5-bromo-N'-(1H-pyrrole-2-carbonyl)pyridine-3-carbohydrazide
—— 5-[3-(3-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3H-1,3-benzoxazol-2-one —— C20H15FN4O4
5-[3-(3-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3H-1,3-benzoxazol-2-one
—— 5-[(3S)-1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-7-oxo-N-phenyl-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H18FN5O3
5-[(3S)-1-(4-fluorophenyl)-5-oxopyrrolidin-3-yl]-7-oxo-N-phenyl-1H-pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-bromo-N-[2-(cyclopropylamino)-2-oxoethyl]-2-fluorobenzamide —— C12H12BrFN2O2
5-bromo-N-[2-(cyclopropylamino)-2-oxoethyl]-2-fluorobenzamide
—— 5-(cyclohexylsulfamoyl)-N-[2-(cyclopropylamino)-2-oxoethyl]-2-methylbenzamide —— C19H27N3O4S
5-(cyclohexylsulfamoyl)-N-[2-(cyclopropylamino)-2-oxoethyl]-2-methylbenzamide
—— 5-[(2R)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C16H22N6O2
5-[(2R)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2S)-1-[(3-chlorophenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C17H21ClN4O
5-[(2S)-1-[(3-chlorophenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2S)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C17H21FN4O
5-[(2S)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2S)-1-[(2-methoxyphenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C18H24N4O2
5-[(2S)-1-[(2-methoxyphenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2S)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C16H22N6O2
5-[(2S)-1-(1-ethylpyrazole-3-carbonyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2R)-1-[2-(3-chloro-4-fluorophenoxy)acetyl]piperidin-2-yl]-N,N-diethyl-1H-pyrazole-4-carboxamide —— C21H26ClFN4O3
5-[(2R)-1-[2-(3-chloro-4-fluorophenoxy)acetyl]piperidin-2-yl]-N,N-diethyl-1H-pyrazole-4-carboxamide
—— 5-[[3-(3-methoxyanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one —— C24H27N5O3
5-[[3-(3-methoxyanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one
—— 5-[(2R)-1-(1-benzofuran-2-ylmethyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C19H22N4O2
5-[(2R)-1-(1-benzofuran-2-ylmethyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2R)-1-[(2-methoxyphenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C18H24N4O2
5-[(2R)-1-[(2-methoxyphenyl)methyl]pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2S)-1-(1-benzofuran-2-ylmethyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide —— C19H22N4O2
5-[(2S)-1-(1-benzofuran-2-ylmethyl)pyrrolidin-2-yl]-N,N-dimethyl-1H-pyrazole-4-carboxamide
—— 5-[(2S)-1-[2-(3-chloro-4-fluorophenoxy)acetyl]piperidin-2-yl]-N,N-diethyl-1H-pyrazole-4-carboxamide —— C21H26ClFN4O3
5-[(2S)-1-[2-(3-chloro-4-fluorophenoxy)acetyl]piperidin-2-yl]-N,N-diethyl-1H-pyrazole-4-carboxamide
—— 5-[[3-(2-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one —— C23H24FN5O2
5-[[3-(2-fluoroanilino)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl]-1,3,6-trimethylbenzimidazol-2-one
—— 5-[(3-anilino-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl)methyl]-1,3,6-trimethylbenzimidazol-2-one —— C23H25N5O2
5-[(3-anilino-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl)methyl]-1,3,6-trimethylbenzimidazol-2-one
—— (5S)-N-[2-(cyclopropylamino)-2-oxoethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C15H20N2O2S
(5S)-N-[2-(cyclopropylamino)-2-oxoethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-chloro-N-[2-(cyclopropylamino)-2-oxoethyl]-2-methoxybenzamide —— C13H15ClN2O3
5-chloro-N-[2-(cyclopropylamino)-2-oxoethyl]-2-methoxybenzamide