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—— (5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone —— C18H19FN6O2
(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone
—— (5-Chloro-2-hydroxyphenyl)-[4-(4-chlorophenyl)sulfonylpiperazin-1-yl]methanone —— C17H16Cl2N2O4S
(5-Chloro-2-hydroxyphenyl)-[4-(4-chlorophenyl)sulfonylpiperazin-1-yl]methanone
—— 5-bromo-2-chloro-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)benzamide —— C15H9BrClN3OS
5-bromo-2-chloro-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)benzamide
—— (5S,7R)-3-acetamido-N-[(4-methylphenyl)methyl]adamantane-1-carboxamide —— C21H28N2O2
(5S,7R)-3-acetamido-N-[(4-methylphenyl)methyl]adamantane-1-carboxamide
—— 5-(1,3-benzodioxol-5-yl)-N-(3-ethenoxypropyl)-4-thiophen-2-ylpyrimidin-2-amine —— C20H19N3O3S
5-(1,3-benzodioxol-5-yl)-N-(3-ethenoxypropyl)-4-thiophen-2-ylpyrimidin-2-amine
—— [5-[[Di(propan-2-yl)amino]methyl]furan-2-yl]-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone —— C22H30FN3O3
[5-[[Di(propan-2-yl)amino]methyl]furan-2-yl]-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone
—— (5S,7R)-3-acetamido-N-(5-methyl-1,3-thiazol-2-yl)adamantane-1-carboxamide —— C17H23N3O2S
(5S,7R)-3-acetamido-N-(5-methyl-1,3-thiazol-2-yl)adamantane-1-carboxamide
—— (5S,7R)-3-acetamido-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)adamantane-1-carboxamide —— C21H24N4O2S
(5S,7R)-3-acetamido-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)adamantane-1-carboxamide
—— 5-chloro-2-methoxy-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)benzamide —— C16H12ClN3O2S
5-chloro-2-methoxy-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)benzamide
—— (5S,7R)-3-acetamido-N-(2,2,2-trifluoroethyl)adamantane-1-carboxamide —— C15H21F3N2O2
(5S,7R)-3-acetamido-N-(2,2,2-trifluoroethyl)adamantane-1-carboxamide
—— 5-[1-[(2-Ethylpyrimidin-5-yl)methyl]piperidin-4-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine —— C20H23F3N6
5-[1-[(2-Ethylpyrimidin-5-yl)methyl]piperidin-4-yl]-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
—— [5-(Methoxymethyl)furan-2-yl]-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C20H21F3N4O3
[5-(Methoxymethyl)furan-2-yl]-[4-[2-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— (5S,7R)-3-chloro-N-[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]adamantane-1-carboxamide —— C17H22ClN3O2S
(5S,7R)-3-chloro-N-[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]adamantane-1-carboxamide
—— (5-Hydroxypyridin-3-yl)-[4-[4-methyl-5-(2-methylpyrimidin-4-yl)-1,3-thiazol-2-yl]piperidin-1-yl]methanone —— C20H21N5O2S
(5-Hydroxypyridin-3-yl)-[4-[4-methyl-5-(2-methylpyrimidin-4-yl)-1,3-thiazol-2-yl]piperidin-1-yl]methanone
—— 5-bromo-2-chloro-N-(5-methyl-4-phenyl-1,3-thiazol-2-yl)benzamide —— C17H12BrClN2OS
5-bromo-2-chloro-N-(5-methyl-4-phenyl-1,3-thiazol-2-yl)benzamide
—— 5,6-Bis(3-fluorophenyl)-2-[(2-methoxyphenyl)methyl]-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C24H17F2N5O2
5,6-Bis(3-fluorophenyl)-2-[(2-methoxyphenyl)methyl]-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— 5,6-dimethyl-3-[4-[4-methyl-5-(2-methylpyrimidin-4-yl)-1,3-thiazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H25N5O2S
5,6-dimethyl-3-[4-[4-methyl-5-(2-methylpyrimidin-4-yl)-1,3-thiazol-2-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5,6-Bis(3-methoxyphenyl)-2-methyl-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C19H17N5O3
5,6-Bis(3-methoxyphenyl)-2-methyl-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— [5-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]furan-2-yl]-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone —— C21H22FN3O4
[5-[(3,5-Dimethyl-1,2-oxazol-4-yl)methyl]furan-2-yl]-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone
—— 5-[[(4aR)-1,3,4,4a,5,6,7,8-octahydropyrido[1,2-c]pyrimidin-2-yl]methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole —— C22H26N6O
5-[[(4aR)-1,3,4,4a,5,6,7,8-octahydropyrido[1,2-c]pyrimidin-2-yl]methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole
—— [5-(1,5-Dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone —— C19H20FN5O3
[5-(1,5-Dimethylpyrazol-4-yl)-1,2-oxazol-3-yl]-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone
—— 5-[(3S)-1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H25N7
5-[(3S)-1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5,6-Bis(4-fluorophenyl)-2-(pyridin-3-ylmethyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C22H14F2N6O
5,6-Bis(4-fluorophenyl)-2-(pyridin-3-ylmethyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— 5-bromo-N-(4-thiophen-2-yl-1,3-thiazol-2-yl)pyridine-3-carboxamide —— C13H8BrN3OS2
5-bromo-N-(4-thiophen-2-yl-1,3-thiazol-2-yl)pyridine-3-carboxamide
—— (5,7-Dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone —— C19H20FN5O2
(5,7-Dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[4-(2-fluoropyridin-3-yl)-4-hydroxypiperidin-1-yl]methanone
—— 5,6-Bis(4-fluorophenyl)-2-methyl-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C17H11F2N5O
5,6-Bis(4-fluorophenyl)-2-methyl-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— 5-[(3R)-1-[(2,4-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H21F2N5
5-[(3R)-1-[(2,4-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[[(4aS)-1,3,4,4a,5,6,7,8-octahydropyrido[1,2-c]pyrimidin-2-yl]methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole —— C22H26N6O
5-[[(4aS)-1,3,4,4a,5,6,7,8-octahydropyrido[1,2-c]pyrimidin-2-yl]methyl]-3-[4-(2-methylpyrimidin-4-yl)phenyl]-1,2,4-oxadiazole
—— 5,6-Bis(4-methoxyphenyl)-2-(pyridin-3-ylmethyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C24H20N6O3
5,6-Bis(4-methoxyphenyl)-2-(pyridin-3-ylmethyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— 5-[(3R)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H26N8
5-[(3R)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5,6-Bis(4-fluorophenyl)-2-[(4-methoxyphenyl)methyl]-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C24H17F2N5O2
5,6-Bis(4-fluorophenyl)-2-[(4-methoxyphenyl)methyl]-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— 5-[(3R)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H22ClN5
5-[(3R)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5,6-Bis(3-methoxyphenyl)-2-(2-oxopropyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C21H19N5O4
5,6-Bis(3-methoxyphenyl)-2-(2-oxopropyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— 5,6-Bis(4-methoxyphenyl)-2-(2-oxopropyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one —— C21H19N5O4
5,6-Bis(4-methoxyphenyl)-2-(2-oxopropyl)-[1,2,4]triazolo[3,4-c][1,2,4]triazin-3-one
—— 5-[(3R)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H21F2N5
5-[(3R)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3R)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H21F2N5
5-[(3R)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3R)-1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H25N7
5-[(3R)-1-[(1-ethenyl-3-methylpyrazol-4-yl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3S)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H22ClN5
5-[(3S)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3R)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H22FN5
5-[(3R)-1-[(3-fluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3S)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H26N8
5-[(3S)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(1,3-benzodioxol-5-yl)-N-(furan-2-ylmethyl)-4-thiophen-2-ylpyrimidin-2-amine —— C20H15N3O3S
5-(1,3-benzodioxol-5-yl)-N-(furan-2-ylmethyl)-4-thiophen-2-ylpyrimidin-2-amine
—— 5-[(3S)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H21F2N5
5-[(3S)-1-[(2,3-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(1,3-Benzodioxol-5-yl)-2-(4-methylpiperazin-1-yl)-4-thiophen-2-ylpyrimidine —— C20H20N4O2S
5-(1,3-Benzodioxol-5-yl)-2-(4-methylpiperazin-1-yl)-4-thiophen-2-ylpyrimidine
—— 5-(1,3-benzodioxol-5-yl)-N-(2-morpholin-4-ylethyl)-4-thiophen-2-ylpyrimidin-2-amine —— C21H22N4O3S
5-(1,3-benzodioxol-5-yl)-N-(2-morpholin-4-ylethyl)-4-thiophen-2-ylpyrimidin-2-amine
—— 5-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-pyridin-3-ylpyrimidin-2-amine —— C23H17FN4O2
5-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-pyridin-3-ylpyrimidin-2-amine
—— 5-[(3S)-1-[(2S)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C23H29N5O2
5-[(3S)-1-[(2S)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3S)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H21F2N5
5-[(3S)-1-[(2,5-difluorophenyl)methyl]piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(1,3-benzodioxol-5-yl)-N-[(2-methoxyphenyl)methyl]-4-pyridin-3-ylpyrimidin-2-amine —— C24H20N4O3
5-(1,3-benzodioxol-5-yl)-N-[(2-methoxyphenyl)methyl]-4-pyridin-3-ylpyrimidin-2-amine
—— 5-(1,3-benzodioxol-5-yl)-N-(pyridin-2-ylmethyl)-4-thiophen-2-ylpyrimidin-2-amine —— C21H16N4O2S
5-(1,3-benzodioxol-5-yl)-N-(pyridin-2-ylmethyl)-4-thiophen-2-ylpyrimidin-2-amine
—— 5-[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C17H21N5O
5-[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine