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—— 5-methyl-3-[(3S)-1-(6-methylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C13H16N6OS
5-methyl-3-[(3S)-1-(6-methylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3S)-1-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-3-yl]-1,2,4-oxadiazole —— C15H19N7O
5-ethyl-3-[(3S)-1-(5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3S)-1-thieno[2,3-d]pyrimidin-4-ylpiperidin-3-yl]-1,2,4-oxadiazole —— C15H17N5OS
5-ethyl-3-[(3S)-1-thieno[2,3-d]pyrimidin-4-ylpiperidin-3-yl]-1,2,4-oxadiazole
—— 5-propan-2-yl-3-[(3R)-1-quinoxalin-2-ylpiperidin-3-yl]-1,2,4-oxadiazole —— C18H21N5O
5-propan-2-yl-3-[(3R)-1-quinoxalin-2-ylpiperidin-3-yl]-1,2,4-oxadiazole
—— 5-(methylsulfamoyl)-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide —— C14H18N4O4S
5-(methylsulfamoyl)-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide
—— 5-ethyl-3-[(2R)-1-thieno[2,3-d]pyrimidin-4-ylpyrrolidin-2-yl]-1,2,4-oxadiazole —— C14H15N5OS
5-ethyl-3-[(2R)-1-thieno[2,3-d]pyrimidin-4-ylpyrrolidin-2-yl]-1,2,4-oxadiazole
—— 5-methyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1H-pyrazole-3-carboxamide —— C13H17N5O
5-methyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1H-pyrazole-3-carboxamide
—— 5-(methylsulfamoyl)-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide —— C14H18N4O4S
5-(methylsulfamoyl)-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide
—— 5-ethyl-3-[(3S)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-3-yl]-1,2,4-oxadiazole —— C14H16F3N5O
5-ethyl-3-[(3S)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-ethyl-3-[(3R)-1-thieno[3,2-d]pyrimidin-4-ylpiperidin-3-yl]-1,2,4-oxadiazole —— C15H17N5OS
5-ethyl-3-[(3R)-1-thieno[3,2-d]pyrimidin-4-ylpiperidin-3-yl]-1,2,4-oxadiazole
—— 5-bromo-3-methyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide —— C14H16BrN3O2
5-bromo-3-methyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide
—— 5-cyclopropyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1H-pyrazole-3-carboxamide —— C15H19N5O
5-cyclopropyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1H-pyrazole-3-carboxamide
—— 5-cyclopropyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1H-pyrazole-3-carboxamide —— C15H19N5O
5-cyclopropyl-N-[(6S)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-1H-pyrazole-3-carboxamide
—— 5-chloro-2-propan-2-yloxy-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]benzamide —— C17H20ClN3O2
5-chloro-2-propan-2-yloxy-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]benzamide
—— 5-Methyl-1-(2-methylphenyl)-3-(2-methylpropyl)pyrazole-4-carboxylate —— C16H19N2O2-
5-Methyl-1-(2-methylphenyl)-3-(2-methylpropyl)pyrazole-4-carboxylate
—— 5-ethyl-3-methyl-1-(2-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-4-carboxamide —— C19H25N3O2
5-ethyl-3-methyl-1-(2-methylphenyl)-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-4-carboxamide
—— [5-Ethyl-1-(4-fluorophenyl)-3-(2-methylpropyl)pyrazol-4-yl]-(4-ethylpiperazin-4-ium-1-yl)methanone —— C22H32FN4O+
[5-Ethyl-1-(4-fluorophenyl)-3-(2-methylpropyl)pyrazol-4-yl]-(4-ethylpiperazin-4-ium-1-yl)methanone
—— 5-ethyl-1-(4-fluorophenyl)-N-(furan-2-ylmethyl)-3-propylpyrazole-4-carboxamide —— C20H22FN3O2
5-ethyl-1-(4-fluorophenyl)-N-(furan-2-ylmethyl)-3-propylpyrazole-4-carboxamide
—— [5-Ethyl-1-(3-fluorophenyl)-3-propylpyrazol-4-yl]-(4-ethylpiperazin-1-yl)methanone —— C21H29FN4O
[5-Ethyl-1-(3-fluorophenyl)-3-propylpyrazol-4-yl]-(4-ethylpiperazin-1-yl)methanone
—— 5-ethyl-3-methyl-1-(2-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-4-carboxamide —— C19H25N3O2
5-ethyl-3-methyl-1-(2-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-4-carboxamide
—— 5-methyl-1-(2-methylphenyl)-N-(2-methylpropyl)-3-propylpyrazole-4-carboxamide —— C19H27N3O
5-methyl-1-(2-methylphenyl)-N-(2-methylpropyl)-3-propylpyrazole-4-carboxamide
—— (5-Methyl-1-phenyl-3-propylpyrazol-4-yl)-piperidin-1-ylmethanone —— C19H25N3O
(5-Methyl-1-phenyl-3-propylpyrazol-4-yl)-piperidin-1-ylmethanone
—— 5-Methyl-1-(2-methylphenyl)-3-(2-methylpropyl)pyrazole-4-carboxylic acid —— C16H20N2O2
5-Methyl-1-(2-methylphenyl)-3-(2-methylpropyl)pyrazole-4-carboxylic acid
—— 5-methyl-N-(4-phenoxypyridin-3-yl)-1H-pyrazole-3-carboxamide —— C16H14N4O2
5-methyl-N-(4-phenoxypyridin-3-yl)-1H-pyrazole-3-carboxamide
—— 5-methyl-1-(2-methylphenyl)-N,3-bis(2-methylpropyl)pyrazole-4-carboxamide —— C20H29N3O
5-methyl-1-(2-methylphenyl)-N,3-bis(2-methylpropyl)pyrazole-4-carboxamide
—— 5-methyl-N-(2-methylpropyl)-1-phenyl-3-propylpyrazole-4-carboxamide —— C18H25N3O
5-methyl-N-(2-methylpropyl)-1-phenyl-3-propylpyrazole-4-carboxamide
—— 5-oxo-N-(1,3-thiazol-2-ylmethyl)-N-(2,2,2-trifluoroethyl)-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C13H11F3N4O2S2
5-oxo-N-(1,3-thiazol-2-ylmethyl)-N-(2,2,2-trifluoroethyl)-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-Methyl-3-(2-methylpropyl)-1-(4-nitrophenyl)pyrazole-4-carboxylate —— C15H16N3O4-
5-Methyl-3-(2-methylpropyl)-1-(4-nitrophenyl)pyrazole-4-carboxylate
—— 5-ethyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide —— C15H19N3O2
5-ethyl-N-[(6R)-2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]furan-2-carboxamide
—— [5-Ethyl-1-(3-fluorophenyl)-3-propylpyrazol-4-yl]-(4-ethylpiperazin-4-ium-1-yl)methanone —— C21H30FN4O+
[5-Ethyl-1-(3-fluorophenyl)-3-propylpyrazol-4-yl]-(4-ethylpiperazin-4-ium-1-yl)methanone
—— 5-Methyl-3-(2-methylpropyl)-1-(4-nitrophenyl)pyrazole-4-carboxylic acid —— C15H17N3O4
5-Methyl-3-(2-methylpropyl)-1-(4-nitrophenyl)pyrazole-4-carboxylic acid
—— 5-Methyl-1-phenyl-3-propylpyrazole-4-carboxylate —— C14H15N2O2-
5-Methyl-1-phenyl-3-propylpyrazole-4-carboxylate
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1S)-1-cyclopropylethyl]-N-(4-methoxyphenyl)pentanamide —— C22H31N3O3S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-N-[(1S)-1-cyclopropylethyl]-N-(4-methoxyphenyl)pentanamide
—— 5-methyl-N-[[(2S)-oxolan-2-yl]methyl]-N-[3-oxo-3-(propan-2-ylamino)propyl]pyrazine-2-carboxamide —— C17H26N4O3
5-methyl-N-[[(2S)-oxolan-2-yl]methyl]-N-[3-oxo-3-(propan-2-ylamino)propyl]pyrazine-2-carboxamide
—— [5-Methyl-1-(4-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-piperidin-1-ylmethanone —— C21H29N3O
[5-Methyl-1-(4-methylphenyl)-3-(2-methylpropyl)pyrazol-4-yl]-piperidin-1-ylmethanone
—— [5-Ethyl-1-(4-fluorophenyl)-3-(2-methylpropyl)pyrazol-4-yl]-morpholin-4-ylmethanone —— C20H26FN3O2
[5-Ethyl-1-(4-fluorophenyl)-3-(2-methylpropyl)pyrazol-4-yl]-morpholin-4-ylmethanone
—— 5-(4-methoxyphenyl)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pentanamide —— C19H25N3O2
5-(4-methoxyphenyl)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pentanamide
—— 5-ethyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]thiophene-2-carboxamide —— C14H17N3OS
5-ethyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]thiophene-2-carboxamide
—— 5-chloro-2-(diethylamino)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyrimidine-4-carboxamide —— C16H21ClN6O
5-chloro-2-(diethylamino)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyrimidine-4-carboxamide
—— 5-(4-methoxyphenyl)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pentanamide —— C19H25N3O2
5-(4-methoxyphenyl)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pentanamide
—— 5-chloro-2-(diethylamino)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyrimidine-4-carboxamide —— C16H21ClN6O
5-chloro-2-(diethylamino)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyrimidine-4-carboxamide
—— 5-ethyl-4-methyl-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]thiophene-2-carboxamide —— C15H19N3OS
5-ethyl-4-methyl-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]thiophene-2-carboxamide
—— 5-ethyl-4-methyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]thiophene-2-carboxamide —— C15H19N3OS
5-ethyl-4-methyl-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]thiophene-2-carboxamide
—— [5-[[[(2R)-butan-2-yl]-(thiophene-2-carbonyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C18H23NO5S2
[5-[[[(2R)-butan-2-yl]-(thiophene-2-carbonyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— [5-[[[(2R)-butan-2-yl]-(furan-2-carbonyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate —— C20H27NO6S
[5-[[[(2R)-butan-2-yl]-(furan-2-carbonyl)amino]methyl]-2-methoxyphenyl] propane-2-sulfonate
—— 5-propan-2-yl-3-[(3S)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole —— C17H24N4O
5-propan-2-yl-3-[(3S)-1-[(1S)-1-pyridin-4-ylethyl]piperidin-3-yl]-1,2,4-oxadiazole
—— 5-acetamido-2-fluoro-N-[(1R)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]benzamide —— C18H17FN2O3
5-acetamido-2-fluoro-N-[(1R)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]benzamide
—— 5-{[N-Cyclopropyl-1-(thiophen-2-YL)formamido]methyl}-2-methoxyphenyl propane-2-sulfonate —— C19H23NO5S2
5-{[N-Cyclopropyl-1-(thiophen-2-YL)formamido]methyl}-2-methoxyphenyl propane-2-sulfonate
—— 5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-1,3-dimethylpyrazolo[3,4-b]pyridine —— C15H21N5O2S
5-[[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]sulfonyl]-1,3-dimethylpyrazolo[3,4-b]pyridine
—— [5-(2-fluorophenyl)-1,2-oxazol-3-yl]-[(2S)-2-(1-methylpyrrol-2-yl)azepan-1-yl]methanone —— C21H22FN3O2
[5-(2-fluorophenyl)-1,2-oxazol-3-yl]-[(2S)-2-(1-methylpyrrol-2-yl)azepan-1-yl]methanone