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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-9-[(2-butyl-1H-imidazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H24N4O2
(5S)-9-[(2-butyl-1H-imidazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-N,5-dimethyl-N-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide —— C18H20N4OS2
(5R)-N,5-dimethyl-N-[(2-thiophen-2-yl-1,3-thiazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
—— (5E)-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-5-[(3-nitrophenyl)methylidene]-1,3-thiazol-4-one —— C16H17N3O4S
(5E)-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-5-[(3-nitrophenyl)methylidene]-1,3-thiazol-4-one
—— (5-Acetyl-2-methoxyphenyl)methyl 2-methoxy-5-nitrobenzoate —— C18H17NO7
(5-Acetyl-2-methoxyphenyl)methyl 2-methoxy-5-nitrobenzoate
—— (5S)-7-(cyclobutylmethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C23H29N3O
(5S)-7-(cyclobutylmethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-methoxy-5-nitrobenzoate —— C15H11N3O6S
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-methoxy-5-nitrobenzoate
—— (5S)-7-[[2-(2-hydroxyethoxy)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H22N2O4
(5S)-7-[[2-(2-hydroxyethoxy)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(9H-fluoren-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C22H24N2O2
(5S)-9-(9H-fluoren-2-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-methoxy-5-nitrobenzoate —— C17H13N3O6
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-methoxy-5-nitrobenzoate
—— 5-[2-[(2R)-2-[2-(dimethylamino)ethyl]piperidin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C16H26N4O3
5-[2-[(2R)-2-[2-(dimethylamino)ethyl]piperidin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— 5-(2-fluorophenyl)-N-[(2S)-1-methoxypropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H17FN4O
5-(2-fluorophenyl)-N-[(2S)-1-methoxypropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-methoxy-5-nitrobenzoate —— C17H12ClN3O6
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-methoxy-5-nitrobenzoate
—— (5E)-5-[[4-(2-hydroxyethoxy)-3-methoxyphenyl]methylidene]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C21H20N2O5S
(5E)-5-[[4-(2-hydroxyethoxy)-3-methoxyphenyl]methylidene]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H20FN3O3
5-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5R)-7-(cyclobutylmethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C23H29N3O
(5R)-7-(cyclobutylmethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H26N2O4
(5S)-9-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H26N2O4
(5R)-9-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-propyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C14H19N7
5-propyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-2-(1,3-dihydroxypropan-2-yl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N2O3
(5S)-2-(1,3-dihydroxypropan-2-yl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 4-(furan-2-carbonylamino)benzoate —— C20H14N2O6
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 4-(furan-2-carbonylamino)benzoate
—— 5-bromo-N-[2-[[(1S)-2-methyl-1-thiophen-2-ylpropyl]amino]-2-oxoethyl]furan-2-carboxamide —— C15H17BrN2O3S
5-bromo-N-[2-[[(1S)-2-methyl-1-thiophen-2-ylpropyl]amino]-2-oxoethyl]furan-2-carboxamide
—— 5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H20FN3O3
5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 1-ethyl-2,5-dimethylpyrrole-3-carboxylate —— C19H20N2O3
(5-Phenyl-1,2-oxazol-3-yl)methyl 1-ethyl-2,5-dimethylpyrrole-3-carboxylate
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidin-2-amine —— C16H27N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidin-2-amine
—— [5-(5-Bromothiophen-2-yl)-1,3,4-oxadiazol-2-yl]methyl 1-ethyl-2,5-dimethylpyrrole-3-carboxylate —— C16H16BrN3O3S
[5-(5-Bromothiophen-2-yl)-1,3,4-oxadiazol-2-yl]methyl 1-ethyl-2,5-dimethylpyrrole-3-carboxylate
—— (5S)-3-methyl-7-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H29N3O2
(5S)-3-methyl-7-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H27N7O2
(5S)-9-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-methoxy-2-[(3S)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine —— C19H29N7O
5-methoxy-2-[(3S)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine
—— 5-methyl-N-[[(2R)-morpholin-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C12H17N5O
5-methyl-N-[[(2R)-morpholin-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-3-methyl-7-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H29N3O2
(5R)-3-methyl-7-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methyl-N-[[(2S)-morpholin-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C12H17N5O
5-methyl-N-[[(2S)-morpholin-2-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H32N2O3
(5S)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidin-2-amine —— C16H27N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(2-pyrrolidin-1-ylethyl)pyrimidin-2-amine
—— (5R)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C21H32N2O3
(5R)-9-[[4-(3-hydroxy-3-methylbutyl)phenyl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-2-amine —— C15H21N5O2S2
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-2-amine
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-pent-2-ynylpyridazin-3-one —— C15H22N4O2
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-pent-2-ynylpyridazin-3-one
—— (5R)-9-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H27N7O2
(5R)-9-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-pent-2-ynylpyridazin-3-one —— C15H22N4O2
5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-pent-2-ynylpyridazin-3-one
—— 5-methoxy-2-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine —— C19H29N7O
5-methoxy-2-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine
—— (5S)-5-[[2-[2-(furan-2-yl)pyrimidin-5-yl]imidazol-1-yl]methyl]-1-methylpyrrolidin-2-one —— C17H17N5O2
(5S)-5-[[2-[2-(furan-2-yl)pyrimidin-5-yl]imidazol-1-yl]methyl]-1-methylpyrrolidin-2-one
—— 5-ethyl-2,3-dimethyl-N-[[(3S)-piperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H25N5
5-ethyl-2,3-dimethyl-N-[[(3S)-piperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-2-amine —— C15H21N5O2S2
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-2-amine
—— [5-(methoxymethyl)furan-2-yl]-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methanone —— C19H24N2O4
[5-(methoxymethyl)furan-2-yl]-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methanone
—— 5-chloro-N-[(2S)-1-hydroxypropan-2-yl]-N-methyl-3-phenyl-1H-indole-2-carboxamide —— C19H19ClN2O2
5-chloro-N-[(2S)-1-hydroxypropan-2-yl]-N-methyl-3-phenyl-1H-indole-2-carboxamide
—— 5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[2-(2,4-dimethylphenoxy)ethyl]pyridazin-3-one —— C20H28N4O3
5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[2-(2,4-dimethylphenoxy)ethyl]pyridazin-3-one
—— (5R)-7-(2,2-diphenylethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C21H24N2O2
(5R)-7-(2,2-diphenylethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(1-propyltetrazol-5-yl)methylsulfanyl]-N-[2-(trifluoromethyl)phenyl]-1,3,4-thiadiazol-2-amine —— C14H14F3N7S2
5-[(1-propyltetrazol-5-yl)methylsulfanyl]-N-[2-(trifluoromethyl)phenyl]-1,3,4-thiadiazol-2-amine
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 4-(furan-2-carbonylamino)benzoate —— C22H16N2O5
(5-Phenyl-1,2-oxazol-3-yl)methyl 4-(furan-2-carbonylamino)benzoate
—— (5S)-3-methyl-7-[(4-methylsulfanylphenyl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H20N2O2S
(5S)-3-methyl-7-[(4-methylsulfanylphenyl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(6R)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C19H24N4O3
5-[(6R)-2-ethyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-4-methyl-2-oxo-1H-pyridine-3-carbonitrile