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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-2-thiophen-2-ylpyrimidine —— C20H22N4OS
5-[[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-2-thiophen-2-ylpyrimidine
—— (5R)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane —— C17H26N2
(5R)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
—— (5S)-9-[(2-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C19H23FN4
(5S)-9-[(2-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methoxyphenyl)acetate —— C18H15ClN2O4
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methoxyphenyl)acetate
—— (5R)-3-methyl-7-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H24N4O3
(5R)-3-methyl-7-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane —— C17H26N2
(5S)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
—— 5-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one —— C24H21N3O2S
5-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-6-phenylthieno[2,3-d]pyrimidin-4-one
—— 5-chloro-N-[[(4R)-4-hydroxyazepan-4-yl]methyl]-3-methyl-1-benzothiophene-2-sulfonamide —— C16H21ClN2O3S2
5-chloro-N-[[(4R)-4-hydroxyazepan-4-yl]methyl]-3-methyl-1-benzothiophene-2-sulfonamide
—— (5R)-9-[(2-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane —— C19H23FN4
(5R)-9-[(2-fluorophenyl)methyl]-2-pyrimidin-2-yl-2,9-diazaspiro[4.5]decane
—— (5R)-3-methyl-7-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C13H20N4O2S
(5R)-3-methyl-7-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H20N4O3
(5S)-3-methyl-9-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H19FN2O
(5R)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-propan-2-yl-N-[(1R)-1-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H19N7O
5-propan-2-yl-N-[(1R)-1-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(4-methylpiperazin-1-yl)-2-[2-[(3R)-oxolan-3-yl]ethyl]pyridazin-3-one —— C15H24N4O2
5-(4-methylpiperazin-1-yl)-2-[2-[(3R)-oxolan-3-yl]ethyl]pyridazin-3-one
—— 5-[2-(2-Fluorophenyl)sulfanylethylsulfanyl]-1-(2-methoxy-5-methylphenyl)tetrazole —— C17H17FN4OS2
5-[2-(2-Fluorophenyl)sulfanylethylsulfanyl]-1-(2-methoxy-5-methylphenyl)tetrazole
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methoxyphenyl)acetate —— C16H14N2O5
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methoxyphenyl)acetate
—— 5-[(3R)-3-[2-(dimethylamino)ethyl-methylamino]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C18H27N5O2
5-[(3R)-3-[2-(dimethylamino)ethyl-methylamino]piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[(3R)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C20H27N5O3
5-[(3R)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— (5R)-2-(2,3-dihydrothieno[3,4-b][1,4]dioxine-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N2O5S
(5R)-2-(2,3-dihydrothieno[3,4-b][1,4]dioxine-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-methyl-9-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H24N4O3
(5R)-3-methyl-9-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5,7-dimethyl-N-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide —— C16H18N6OS
5,7-dimethyl-N-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-9-(6-fluoro-4-oxo-1H-quinoline-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H18FN3O4
(5R)-9-(6-fluoro-4-oxo-1H-quinoline-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(6-fluoro-4-oxo-1H-quinoline-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H18FN3O4
(5S)-9-(6-fluoro-4-oxo-1H-quinoline-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-7-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C13H20N4O2S
(5S)-3-methyl-7-[(4-propan-2-ylthiadiazol-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-9-[[1-(3-methylbutyl)benzimidazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C22H32N4O2
(5S)-3-methyl-9-[[1-(3-methylbutyl)benzimidazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-2-(1,3-benzoxazol-2-yl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H21F2N3O2
(5R)-2-(1,3-benzoxazol-2-yl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(2-imidazol-1-ylacetyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H20N4O3
(5R)-9-(2-imidazol-1-ylacetyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-(4-methylpiperazin-1-yl)-2-[2-[(3S)-oxolan-3-yl]ethyl]pyridazin-3-one —— C15H24N4O2
5-(4-methylpiperazin-1-yl)-2-[2-[(3S)-oxolan-3-yl]ethyl]pyridazin-3-one
—— (5R)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C12H20N2O
(5R)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(1,3-benzoxazol-2-yl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H21F2N3O2
(5S)-2-(1,3-benzoxazol-2-yl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole —— C19H22N4O
5-[[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole
—— (5S)-7-(3,5-dichloro-2-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H16Cl2N2O4
(5S)-7-(3,5-dichloro-2-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-N-(2-chlorophenyl)-6-oxo-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide —— C21H23ClN4O2
(5R)-N-(2-chlorophenyl)-6-oxo-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[3-(tetrazol-1-yl)propyl]pyridazin-3-one —— C14H22N8O2
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-[3-(tetrazol-1-yl)propyl]pyridazin-3-one
—— 5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[3-(tetrazol-1-yl)propyl]pyridazin-3-one —— C14H22N8O2
5-[(2R)-2-(2-aminoethyl)morpholin-4-yl]-2-[3-(tetrazol-1-yl)propyl]pyridazin-3-one
—— (5R)-3-methyl-9-[[1-(3-methylbutyl)benzimidazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C22H32N4O2
(5R)-3-methyl-9-[[1-(3-methylbutyl)benzimidazol-2-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H20ClN3O4
(5R)-9-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-N-(2-chlorophenyl)-6-oxo-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide —— C21H23ClN4O2
(5S)-N-(2-chlorophenyl)-6-oxo-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C12H20N2O
(5S)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(3,5-dichloro-2-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H16Cl2N2O4
(5R)-7-(3,5-dichloro-2-methoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H20ClN3O4
(5S)-9-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5-fluoro-1H-indol-3-yl)-[(2S)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone —— C22H21FN2O2
(5-fluoro-1H-indol-3-yl)-[(2S)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone
—— (5-fluoro-1H-indol-3-yl)-[(2R)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone —— C22H21FN2O2
(5-fluoro-1H-indol-3-yl)-[(2R)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]methanone
—— (5S)-9-(2-imidazol-1-ylacetyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C14H20N4O3
(5S)-9-(2-imidazol-1-ylacetyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole —— C19H22N4O
5-[[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]methyl]-3-phenyl-1,2-oxazole
—— (5S)-7-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H20N4O4
(5S)-7-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[(1-benzylimidazol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H22N4O2
(5S)-7-[(1-benzylimidazol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C13H19N5O3S
(5S)-7-[2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-[2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C13H19N5O3S
(5R)-7-[2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H20N4O4
(5R)-7-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one