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—— (5S,6R)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-6-(4-fluorophenyl)-1-methylpiperidin-2-one —— C22H30FN3O2
(5S,6R)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-6-(4-fluorophenyl)-1-methylpiperidin-2-one
—— (5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-5-(4-fluorophenyl)-4-methylmorpholin-3-one —— C21H28FN3O3
(5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-5-(4-fluorophenyl)-4-methylmorpholin-3-one
—— 5-methoxy-1,3-dimethyl-4-[(2S)-1-(3-methylsulfonylpropyl)pyrrolidin-2-yl]pyrazole —— C14H25N3O3S
5-methoxy-1,3-dimethyl-4-[(2S)-1-(3-methylsulfonylpropyl)pyrrolidin-2-yl]pyrazole
—— (5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-phenylmorpholin-3-one —— C21H29N3O3
(5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-phenylmorpholin-3-one
—— (5R,6S)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one —— C23H33N3O3
(5R,6S)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-6-(4-methoxyphenyl)-1-methylpiperidin-2-one
—— (5S,6S)-5-(4-chlorophenyl)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methylmorpholin-3-one —— C21H28ClN3O3
(5S,6S)-5-(4-chlorophenyl)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methylmorpholin-3-one
—— (5S,6R)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-1-methyl-6-(4-methylphenyl)piperidin-2-one —— C23H33N3O2
(5S,6R)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-1-methyl-6-(4-methylphenyl)piperidin-2-one
—— (5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-5-(3-fluorophenyl)-4-methylmorpholin-3-one —— C21H28FN3O3
(5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-5-(3-fluorophenyl)-4-methylmorpholin-3-one
—— 5-chloro-1,3-dimethyl-4-[(2R)-1-(2-methylsulfonylethyl)pyrrolidin-2-yl]pyrazole —— C12H20ClN3O2S
5-chloro-1,3-dimethyl-4-[(2R)-1-(2-methylsulfonylethyl)pyrrolidin-2-yl]pyrazole
—— (5S,6S)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-phenylmorpholin-3-one —— C21H29N3O3
(5S,6S)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-phenylmorpholin-3-one
—— (5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-(4-methylphenyl)morpholin-3-one —— C22H31N3O3
(5S,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-(4-methylphenyl)morpholin-3-one
—— (5R,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-phenylmorpholin-3-one —— C21H29N3O3
(5R,6R)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-4-methyl-5-phenylmorpholin-3-one
—— (5-Tert-butyl-2-methylpyrazol-3-yl)-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone —— C18H30N4O
(5-Tert-butyl-2-methylpyrazol-3-yl)-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone
—— 5-methoxy-1,3-dimethyl-4-[(2R)-1-(3-methylsulfonylpropyl)pyrrolidin-2-yl]pyrazole —— C14H25N3O3S
5-methoxy-1,3-dimethyl-4-[(2R)-1-(3-methylsulfonylpropyl)pyrrolidin-2-yl]pyrazole
—— [5-(4-Chlorophenyl)-1,2-oxazol-3-yl]-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone —— C19H22ClN3O2
[5-(4-Chlorophenyl)-1,2-oxazol-3-yl]-[4-(cyclopropylmethyl)-1,4-diazepan-1-yl]methanone
—— 5-chloro-1,3-dimethyl-4-[(2S)-1-(2-methylsulfonylethyl)pyrrolidin-2-yl]pyrazole —— C12H20ClN3O2S
5-chloro-1,3-dimethyl-4-[(2S)-1-(2-methylsulfonylethyl)pyrrolidin-2-yl]pyrazole
—— (5S,6S)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-5-(3-fluorophenyl)-4-methylmorpholin-3-one —— C21H28FN3O3
(5S,6S)-6-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-5-(3-fluorophenyl)-4-methylmorpholin-3-one
—— (5R,6S)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-6-(3-fluorophenyl)-1-methylpiperidin-2-one —— C22H30FN3O2
(5R,6S)-5-[4-(cyclopropylmethyl)-1,4-diazepane-1-carbonyl]-6-(3-fluorophenyl)-1-methylpiperidin-2-one
—— 5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole —— C15H22N4O2
5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole
—— 5-methoxy-4-[(2S)-1-[2-(2-methoxyphenoxy)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole —— C19H27N3O3
5-methoxy-4-[(2S)-1-[2-(2-methoxyphenoxy)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole
—— 5-[(1S)-1-[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C15H23N5O2
5-[(1S)-1-[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-methoxy-1,3-dimethyl-4-[(2R)-1-[[(2S)-oxan-2-yl]methyl]pyrrolidin-2-yl]pyrazole —— C16H27N3O2
5-methoxy-1,3-dimethyl-4-[(2R)-1-[[(2S)-oxan-2-yl]methyl]pyrrolidin-2-yl]pyrazole
—— 5-methoxy-1,3-dimethyl-4-[(2R)-1-[2-(2,2,2-trifluoroethoxy)ethyl]pyrrolidin-2-yl]pyrazole —— C14H22F3N3O2
5-methoxy-1,3-dimethyl-4-[(2R)-1-[2-(2,2,2-trifluoroethoxy)ethyl]pyrrolidin-2-yl]pyrazole
—— 5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-2-methyl-1,3-thiazole —— C15H22N4OS
5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-2-methyl-1,3-thiazole
—— 5-methoxy-4-[(2S)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole —— C19H27N3O2
5-methoxy-4-[(2S)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole
—— 5-tert-butyl-2-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole —— C18H28N4O2
5-tert-butyl-2-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole
—— 5-methoxy-1,3-dimethyl-4-[(2S)-1-[2-(2,2,2-trifluoroethoxy)ethyl]pyrrolidin-2-yl]pyrazole —— C14H22F3N3O2
5-methoxy-1,3-dimethyl-4-[(2S)-1-[2-(2,2,2-trifluoroethoxy)ethyl]pyrrolidin-2-yl]pyrazole
—— 5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole —— C15H22N4O2
5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2-oxazole
—— 5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-propyl-1,2,4-oxadiazole —— C16H25N5O2
5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-propyl-1,2,4-oxadiazole
—— 5-[(1S)-1-[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole —— C15H23N5O2
5-[(1S)-1-[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-propyl-1,2,4-oxadiazole —— C16H25N5O2
5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-propyl-1,2,4-oxadiazole
—— 5-methoxy-4-[(2R)-1-[2-(2-methoxyphenoxy)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole —— C19H27N3O3
5-methoxy-4-[(2R)-1-[2-(2-methoxyphenoxy)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole
—— 5-chloro-4-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]thiadiazole —— C13H18ClN5OS
5-chloro-4-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]thiadiazole
—— 5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C16H25N5O3
5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-methoxy-1,3-dimethyl-4-[(2S)-1-[(1-methylimidazol-2-yl)methyl]pyrrolidin-2-yl]pyrazole —— C15H23N5O
5-methoxy-1,3-dimethyl-4-[(2S)-1-[(1-methylimidazol-2-yl)methyl]pyrrolidin-2-yl]pyrazole
—— 5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C16H25N5O3
5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-methoxy-1,3-dimethyl-4-[(2R)-1-[2-[(R)-phenylsulfinyl]ethyl]pyrrolidin-2-yl]pyrazole —— C18H25N3O2S
5-methoxy-1,3-dimethyl-4-[(2R)-1-[2-[(R)-phenylsulfinyl]ethyl]pyrrolidin-2-yl]pyrazole
—— 5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2,4-oxadiazole —— C14H21N5O2
5-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2,4-oxadiazole
—— 5-methoxy-1,3-dimethyl-4-[(2R)-1-[(1-methylimidazol-2-yl)methyl]pyrrolidin-2-yl]pyrazole —— C15H23N5O
5-methoxy-1,3-dimethyl-4-[(2R)-1-[(1-methylimidazol-2-yl)methyl]pyrrolidin-2-yl]pyrazole
—— 5-methoxy-1,3-dimethyl-4-[(2S)-1-(2-methylsulfonylethyl)pyrrolidin-2-yl]pyrazole —— C13H23N3O3S
5-methoxy-1,3-dimethyl-4-[(2S)-1-(2-methylsulfonylethyl)pyrrolidin-2-yl]pyrazole
—— 5-tert-butyl-2-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole —— C18H28N4O2
5-tert-butyl-2-[[(2S)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole
—— 5-methoxy-1,3-dimethyl-4-[(2S)-1-[2-[(R)-phenylsulfinyl]ethyl]pyrrolidin-2-yl]pyrazole —— C18H25N3O2S
5-methoxy-1,3-dimethyl-4-[(2S)-1-[2-[(R)-phenylsulfinyl]ethyl]pyrrolidin-2-yl]pyrazole
—— 5-chloro-4-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]thiadiazole —— C13H18ClN5OS
5-chloro-4-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]thiadiazole
—— 5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2,4-oxadiazole —— C14H21N5O2
5-[[(2R)-2-(5-methoxy-1,3-dimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-3-methyl-1,2,4-oxadiazole
—— 5-methoxy-4-[(2R)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole —— C19H27N3O2
5-methoxy-4-[(2R)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-yl]-1,3-dimethylpyrazole
—— 5-cyclopropyl-3-[[(2S)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H23N5O
5-cyclopropyl-3-[[(2S)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-methoxy-1,3-dimethyl-4-[(2S)-1-[[(2S)-oxan-2-yl]methyl]pyrrolidin-2-yl]pyrazole —— C16H27N3O2
5-methoxy-1,3-dimethyl-4-[(2S)-1-[[(2S)-oxan-2-yl]methyl]pyrrolidin-2-yl]pyrazole
—— 5-tert-butyl-2-[[(2S)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole —— C18H28N4O
5-tert-butyl-2-[[(2S)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,3-oxazole
—— 5-cyclopropyl-3-[[(2R)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H23N5O
5-cyclopropyl-3-[[(2R)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-{4-[(2-Fluorophenyl)methoxy]phenyl}-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-A]pyrimidine —— C21H15F4N3O
5-{4-[(2-Fluorophenyl)methoxy]phenyl}-2-methyl-7-(trifluoromethyl)pyrazolo[1,5-A]pyrimidine