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—— (5-Chlorothiophen-2-yl)-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]methanone —— C17H19ClN2O2S
(5-Chlorothiophen-2-yl)-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]methanone
—— 5-[2-[(3S)-4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C19H30N4O4
5-[2-[(3S)-4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— (5R)-9-[(2-chloro-4-hydroxyphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H19ClN2O3
(5R)-9-[(2-chloro-4-hydroxyphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[2-[(3R)-4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C19H30N4O4
5-[2-[(3R)-4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— 5-(2-fluorophenyl)-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(2-fluorophenyl)-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-7-(dibenzofuran-4-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H20N2O3
(5R)-7-(dibenzofuran-4-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-(dibenzofuran-4-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H20N2O3
(5S)-7-(dibenzofuran-4-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5-Chlorothiophen-2-yl)-[4-[(4-methoxyphenyl)methyl]piperazin-4-ium-1-yl]methanone —— C17H20ClN2O2S+
(5-Chlorothiophen-2-yl)-[4-[(4-methoxyphenyl)methyl]piperazin-4-ium-1-yl]methanone
—— 5-(2-fluorophenyl)-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(2-fluorophenyl)-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5-ethyl-1H-pyrazol-4-yl)-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone —— C20H28N6O
(5-ethyl-1H-pyrazol-4-yl)-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone
—— (5-ethyl-1H-pyrazol-4-yl)-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone —— C20H28N6O
(5-ethyl-1H-pyrazol-4-yl)-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone
—— 5-propan-2-yl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H20N6
5-propan-2-yl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-3-methyl-9-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H23N5O2
(5S)-3-methyl-9-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-acetyl-N-(4-bromophenyl)thiophene-2-carboxamide —— C13H10BrNO2S
5-acetyl-N-(4-bromophenyl)thiophene-2-carboxamide
—— (5R)-3-methyl-9-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H23N5O2
(5R)-3-methyl-9-[(3-phenylpyrazolo[1,5-a]pyrimidin-6-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H18FN3O4
5-[(3S)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-[(4R)-5-[(3,5-dimethyl-1-prop-2-enylpyrazol-4-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-3-methyl-1,2-oxazole —— C19H24N6O
5-[(4R)-5-[(3,5-dimethyl-1-prop-2-enylpyrazol-4-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-4-yl]-3-methyl-1,2-oxazole
—— (5S)-9-[[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H24N4O3
(5S)-9-[[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(2-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H13FN8
5-(2-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-acetyl-N-(3-bromophenyl)thiophene-2-carboxamide —— C13H10BrNO2S
5-acetyl-N-(3-bromophenyl)thiophene-2-carboxamide
—— (5R)-7-[[4-(2-imidazol-1-ylethoxy)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C19H24N4O3
(5R)-7-[[4-(2-imidazol-1-ylethoxy)phenyl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-3-methyl-7-(4-methylquinolin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H19N3O2
(5R)-3-methyl-7-(4-methylquinolin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H24N4O3
(5R)-9-[[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-ethyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H19N5O
5-ethyl-N-[(1R)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(2-fluorophenyl)-N-methyl-N-[(1R)-1-(3-nitrophenyl)ethyl]furan-2-carboxamide —— C20H17FN2O4
5-(2-fluorophenyl)-N-methyl-N-[(1R)-1-(3-nitrophenyl)ethyl]furan-2-carboxamide
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone —— C21H24N4O3
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(2S)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone
—— (5S)-9-[(2,3-difluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane —— C19H22F2N4
(5S)-9-[(2,3-difluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H22N4O3
5-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-chloro-2-fluoro-N-(2-methylphenyl)benzamide —— C14H11ClFNO
5-chloro-2-fluoro-N-(2-methylphenyl)benzamide
—— 5-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H22N4O3
5-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— [5-(imidazol-1-ylmethyl)furan-2-yl]-[(2R)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone —— C21H24N4O3
[5-(imidazol-1-ylmethyl)furan-2-yl]-[(2R)-4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methanone
—— 5-[(2,5-Difluorophenyl)sulfanylmethyl]-3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazole —— C17H14F2N2O3S
5-[(2,5-Difluorophenyl)sulfanylmethyl]-3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazole
—— (5S)-3-methyl-7-(4-methylquinolin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H19N3O2
(5S)-3-methyl-7-(4-methylquinolin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-(2-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H13FN8
5-(2-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H18FN3O4
5-[(3R)-3-[(4-fluorophenoxy)methyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-propan-2-yl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C16H20N6
5-propan-2-yl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(2-fluorophenyl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]furan-2-carboxamide —— C20H17FN2O4
5-(2-fluorophenyl)-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]furan-2-carboxamide
—— 5-[(2,5-Difluorophenyl)sulfanylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C16H12F2N2O2S
5-[(2,5-Difluorophenyl)sulfanylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
—— 5-ethyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H25N5O2
5-ethyl-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-9-[(2,3-difluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane —— C19H22F2N4
(5R)-9-[(2,3-difluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-(2-fluorophenyl)-N-[(3R)-3-imidazol-1-ylbutyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H19FN6
5-(2-fluorophenyl)-N-[(3R)-3-imidazol-1-ylbutyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-N-[(1S)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H19N5O
5-ethyl-N-[(1S)-1-(3-ethyl-1,2-oxazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-5-[2-[4-(2-methoxyethylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-2-oxoethyl]pyrrolidin-2-one —— C17H25N5O3
(5S)-5-[2-[4-(2-methoxyethylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-2-oxoethyl]pyrrolidin-2-one
—— 5-[(1R)-1-[[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]ethyl]-1,3,4-thiadiazol-2-amine —— C16H14FN7S
5-[(1R)-1-[[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]ethyl]-1,3,4-thiadiazol-2-amine
—— 5-fluoro-2-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine —— C18H26FN7
5-fluoro-2-[(3R)-3-[4-methyl-5-(piperidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidine
—— (5R)-5-[2-[4-(2-methoxyethylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-2-oxoethyl]pyrrolidin-2-one —— C17H25N5O3
(5R)-5-[2-[4-(2-methoxyethylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-2-oxoethyl]pyrrolidin-2-one
—— 5-[(1S)-1-[[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]ethyl]-1,3,4-thiadiazol-2-amine —— C16H14FN7S
5-[(1S)-1-[[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino]ethyl]-1,3,4-thiadiazol-2-amine
—— 5-methyl-N-[(2R)-1-pyridin-3-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C15H17N5
5-methyl-N-[(2R)-1-pyridin-3-ylpropan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-chloro-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]-1-benzofuran-2-carboxamide —— C18H15ClN2O4
5-chloro-N-methyl-N-[(1S)-1-(3-nitrophenyl)ethyl]-1-benzofuran-2-carboxamide
—— 5-ethyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H25N5O2
5-ethyl-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pyrazolo[1,5-a]pyrimidin-7-amine