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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-3-methyl-9-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5S)-3-methyl-9-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(R)-[(1-methyl-6-propylpyrazolo[3,4-d]pyrimidin-4-yl)amino]-phenylmethyl]-1,3,4-thiadiazol-2-amine —— C18H20N8S
5-[(R)-[(1-methyl-6-propylpyrazolo[3,4-d]pyrimidin-4-yl)amino]-phenylmethyl]-1,3,4-thiadiazol-2-amine
—— 5-chloro-6-oxo-N-[(3R)-1-(2-phenylethyl)piperidin-3-yl]-1H-pyridine-3-carboxamide —— C19H22ClN3O2
5-chloro-6-oxo-N-[(3R)-1-(2-phenylethyl)piperidin-3-yl]-1H-pyridine-3-carboxamide
—— 5-chloro-6-oxo-N-[(3S)-1-(2-phenylethyl)piperidin-3-yl]-1H-pyridine-3-carboxamide —— C19H22ClN3O2
5-chloro-6-oxo-N-[(3S)-1-(2-phenylethyl)piperidin-3-yl]-1H-pyridine-3-carboxamide
—— [(5R)-3,5-dimethyl-4H-1,2-oxazol-5-yl]-(5,6,7,9-tetrahydroimidazo[1,5-a][1,4]diazepin-8-yl)methanone —— C13H18N4O2
[(5R)-3,5-dimethyl-4H-1,2-oxazol-5-yl]-(5,6,7,9-tetrahydroimidazo[1,5-a][1,4]diazepin-8-yl)methanone
—— (5R)-3-methyl-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5R)-3-methyl-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5R)-3-methyl-9-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-phenyl-3-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C18H18N4O
5-phenyl-3-[[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— (5S)-9-[[3-(trifluoromethoxy)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H20F3NO3
(5S)-9-[[3-(trifluoromethoxy)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-methoxy-2-[[(2S)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]pyran-4-one —— C19H23NO4
5-methoxy-2-[[(2S)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]pyran-4-one
—— (5S)-3-methyl-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H20N4O3
(5S)-3-methyl-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(2R)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C15H25N5O3
5-[[(2R)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— [(5S)-3,5-dimethyl-4H-1,2-oxazol-5-yl]-(5,6,7,9-tetrahydroimidazo[1,5-a][1,4]diazepin-8-yl)methanone —— C13H18N4O2
[(5S)-3,5-dimethyl-4H-1,2-oxazol-5-yl]-(5,6,7,9-tetrahydroimidazo[1,5-a][1,4]diazepin-8-yl)methanone
—— 5-[[(2S)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C15H25N5O3
5-[[(2S)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5S)-9-[4-(2-methylimidazol-1-yl)butanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H24N4O3
(5S)-9-[4-(2-methylimidazol-1-yl)butanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[(3-propan-2-ylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H25N3O2
(5S)-9-[(3-propan-2-ylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-7-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H15N5O3
(5R)-7-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18N4O3
(5R)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H23N5O3
(5S)-3-methyl-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(2-phenylquinoline-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C23H21N3O3
(5R)-9-(2-phenylquinoline-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5S)-3-methyl-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18N4O3
(5S)-3-methyl-9-(quinoxaline-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H23N5O3
(5R)-3-methyl-9-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[2-(3,4-dichlorophenyl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H16Cl2N2O3
(5S)-7-[2-(3,4-dichlorophenyl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H21FN2O3
(5R)-9-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-methoxy-2-[[(2R)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]pyran-4-one —— C19H23NO4
5-methoxy-2-[[(2R)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]pyran-4-one
—— (5R)-7-[2-(3,4-dichlorophenyl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H16Cl2N2O3
(5R)-7-[2-(3,4-dichlorophenyl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-ethyl-N-[2-[(2S)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1,2-oxazole-4-carboxamide —— C17H23N5O4
5-ethyl-N-[2-[(2S)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1,2-oxazole-4-carboxamide
—— (5S)-9-(2-phenylquinoline-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C23H21N3O3
(5S)-9-(2-phenylquinoline-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-9-[4-(2-methyltetrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N6O3
(5R)-3-methyl-9-[4-(2-methyltetrazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-[3-(3-oxo-4H-quinoxalin-2-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H24N4O4
(5S)-3-methyl-9-[3-(3-oxo-4H-quinoxalin-2-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[[3-(trifluoromethoxy)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C17H20F3NO3
(5R)-9-[[3-(trifluoromethoxy)phenyl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-7-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H15N5O3
(5S)-7-(imidazo[1,2-b]pyridazine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyridin-2-ylpyrimidine —— C22H25N5O
5-[[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]-2-pyridin-2-ylpyrimidine
—— 5-ethyl-N-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1,2-oxazole-4-carboxamide —— C17H23N5O4
5-ethyl-N-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethyl]-1,2-oxazole-4-carboxamide
—— 5-phenyl-3-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1,2,4-oxadiazole —— C18H18N4O
5-phenyl-3-[[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-[[4-[(2-fluorophenyl)methyl]piperidin-1-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C22H29FN4O
5-[[4-[(2-fluorophenyl)methyl]piperidin-1-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (5S)-9-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H26N4O3
(5S)-9-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[4-[(2-fluorophenyl)methyl]piperidin-1-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C22H29FN4O
5-[[4-[(2-fluorophenyl)methyl]piperidin-1-yl]methyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— (5-methyl-1,2-oxazol-3-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C19H23N3O2
(5-methyl-1,2-oxazol-3-yl)-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5R)-9-(1,3,6-trimethylpyrazolo[3,4-b]pyridine-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H21N5O3
(5R)-9-(1,3,6-trimethylpyrazolo[3,4-b]pyridine-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H20N4O4
(5R)-9-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H20N4O4
(5S)-9-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[(3-propan-2-ylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H25N3O2
(5R)-9-[(3-propan-2-ylimidazol-4-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-(1-benzofuran-5-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N2O3
(5S)-9-(1-benzofuran-5-ylmethyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-ethyl-4-[(3R)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl]-2-methylpyrimidine —— C23H33N5O
5-ethyl-4-[(3R)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl]-2-methylpyrimidine
—— 5-[(5S)-9-(cyclobutylmethyl)-2,9-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-1H-pyridin-4-one —— C20H29N3O2
5-[(5S)-9-(cyclobutylmethyl)-2,9-diazaspiro[4.5]decane-2-carbonyl]-2-methyl-1H-pyridin-4-one
—— 5-[3-[(3R)-3-[methyl(2-pyridin-2-ylethyl)amino]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one —— C19H26N4O3
5-[3-[(3R)-3-[methyl(2-pyridin-2-ylethyl)amino]piperidin-1-yl]-3-oxopropyl]-1,2-oxazol-3-one
—— (5S)-9-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H17N3O4
(5S)-9-(5-phenyl-1,2-oxazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[3-(3-methoxyphenoxy)propyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H26N2O4
(5R)-9-[3-(3-methoxyphenoxy)propyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one