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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-7-methyl-2-(1,3,6-trimethylpyrazolo[3,4-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N6O
(5S)-7-methyl-2-(1,3,6-trimethylpyrazolo[3,4-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H23ClN4O2
(5S)-9-[(5-chloro-3-ethyl-1-methylpyrazol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-5-[[(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]-1-methylpyrrolidin-2-one —— C20H23N5O
(5S)-5-[[(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]-1-methylpyrrolidin-2-one
—— (5R)-9-[(2-methoxy-4-methylphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H24N2O3
(5R)-9-[(2-methoxy-4-methylphenyl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— [5-(furan-2-yl)-1,2-oxazol-3-yl]methyl 3-[[(E)-2-(4-methylphenyl)ethenyl]sulfonylamino]propanoate —— C20H20N2O6S
[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl 3-[[(E)-2-(4-methylphenyl)ethenyl]sulfonylamino]propanoate
—— (5R)-5-[[(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]-1-methylpyrrolidin-2-one —— C20H23N5O
(5R)-5-[[(2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]-1-methylpyrrolidin-2-one
—— [5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(2-chloro-6-fluorophenyl)prop-2-enoate —— C19H14ClFN2O3
[5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl (E)-3-(2-chloro-6-fluorophenyl)prop-2-enoate
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 4-fluoro-3-(methoxymethyl)-1-benzothiophene-2-carboxylate —— C19H14FNO5S
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 4-fluoro-3-(methoxymethyl)-1-benzothiophene-2-carboxylate
—— 5-ethyl-2,3-dimethyl-N-[(1S)-1-(6-methylpyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H23N5
5-ethyl-2,3-dimethyl-N-[(1S)-1-(6-methylpyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 4-fluoro-3-(methoxymethyl)-1-benzothiophene-2-carboxylate —— C21H17FN2O4S
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 4-fluoro-3-(methoxymethyl)-1-benzothiophene-2-carboxylate
—— (5R)-2-(3-chloropyridin-2-yl)-9-(cyclopropylmethyl)-2,9-diazaspiro[4.5]decane —— C17H24ClN3
(5R)-2-(3-chloropyridin-2-yl)-9-(cyclopropylmethyl)-2,9-diazaspiro[4.5]decane
—— (5S)-3-methyl-9-(6-methyl-[1,3]dioxolo[4,5-g]quinolin-8-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H21N3O4
(5S)-3-methyl-9-(6-methyl-[1,3]dioxolo[4,5-g]quinolin-8-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-2-(4-methylquinolin-2-yl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C24H26N4O
(5S)-2-(4-methylquinolin-2-yl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-methyl-9-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H31N3O2
(5R)-3-methyl-9-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-1,2,2,5,7,7-hexamethyl-1-azoniabicyclo[2.2.2]octane —— C13H26N+
(5R)-1,2,2,5,7,7-hexamethyl-1-azoniabicyclo[2.2.2]octane
—— 5-fluoro-N,N-dimethyl-2-[(2S)-1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl]oxypyrimidin-4-amine —— C19H26FN5O
5-fluoro-N,N-dimethyl-2-[(2S)-1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl]oxypyrimidin-4-amine
—— (5-methoxyfuran-2-yl)-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone —— C20H26N4O3
(5-methoxyfuran-2-yl)-[(3S)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone
—— (5R)-2-(4-methylquinolin-2-yl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C24H26N4O
(5R)-2-(4-methylquinolin-2-yl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18ClN3O2
(5S)-9-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-1,2,2,5,7,7-hexamethyl-1-azoniabicyclo[2.2.2]octane —— C13H26N+
(5S)-1,2,2,5,7,7-hexamethyl-1-azoniabicyclo[2.2.2]octane
—— (5R)-9-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18ClN3O2
(5R)-9-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5,6-dimethyl-N-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]thieno[2,3-d]pyrimidin-4-amine —— C19H23N5S
5,6-dimethyl-N-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]thieno[2,3-d]pyrimidin-4-amine
—— [5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 1-(2-fluorophenyl)cyclopentane-1-carboxylate —— C22H21FN2O3
[5-(3-Methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 1-(2-fluorophenyl)cyclopentane-1-carboxylate
—— 5-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C17H15FN4O2
5-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 4-(5-chlorothiophen-2-yl)-4-oxobutanoate —— C18H14ClNO4S
(5-Phenyl-1,2-oxazol-3-yl)methyl 4-(5-chlorothiophen-2-yl)-4-oxobutanoate
—— 5-fluoro-N,N-dimethyl-2-[(2R)-1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl]oxypyrimidin-4-amine —— C19H26FN5O
5-fluoro-N,N-dimethyl-2-[(2R)-1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl]oxypyrimidin-4-amine
—— (5R)-3-methyl-9-(6-methyl-[1,3]dioxolo[4,5-g]quinolin-8-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H21N3O4
(5R)-3-methyl-9-(6-methyl-[1,3]dioxolo[4,5-g]quinolin-8-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-methoxyfuran-2-yl)-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone —— C20H26N4O3
(5-methoxyfuran-2-yl)-[(3R)-3-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)piperidin-1-yl]methanone
—— 5-propan-2-yl-N-[[(3R)-1-pyridin-2-ylpiperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H26N6
5-propan-2-yl-N-[[(3R)-1-pyridin-2-ylpiperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-propan-2-yl-N-[[(3S)-1-pyridin-2-ylpiperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H26N6
5-propan-2-yl-N-[[(3S)-1-pyridin-2-ylpiperidin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(2-fluorophenyl)-N-[2-[(2R)-piperidin-2-yl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H22FN5
5-(2-fluorophenyl)-N-[2-[(2R)-piperidin-2-yl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C17H15FN4O2
5-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— 5-[[4-(3-methylphenoxy)piperidin-1-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine —— C22H30N4O2
5-[[4-(3-methylphenoxy)piperidin-1-yl]methyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrimidin-2-amine
—— 5-(2-fluorophenyl)-N-[2-[(2S)-piperidin-2-yl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C19H22FN5
5-(2-fluorophenyl)-N-[2-[(2S)-piperidin-2-yl]ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-ethyl-N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine —— C18H29N5O
5-ethyl-N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O2
(5S)-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(2S)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile —— C16H21N3O
5-[(2S)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile
—— (5-phenyl-1,2-oxazol-3-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C20H16FNO4
(5-phenyl-1,2-oxazol-3-yl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— 5-[(2R)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile —— C16H21N3O
5-[(2R)-1-pyrrolidin-1-ylhex-5-en-2-yl]oxypyridine-2-carbonitrile
—— 5-ethyl-7-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrazolo[1,5-a]pyrimidine —— C19H30N6
5-ethyl-7-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-ethyl-7-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrazolo[1,5-a]pyrimidine —— C19H30N6
5-ethyl-7-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrazolo[1,5-a]pyrimidine
—— [5-(furan-2-yl)-1,2-oxazol-3-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C18H14FNO5
[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate
—— 5-ethyl-N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine —— C18H29N5O
5-ethyl-N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-methyl-1-[3-[2-[5-[(2S)-oxan-2-yl]furan-2-yl]imidazol-1-yl]phenyl]tetrazole —— C20H20N6O2
5-methyl-1-[3-[2-[5-[(2S)-oxan-2-yl]furan-2-yl]imidazol-1-yl]phenyl]tetrazole
—— (5R)-9-(8-chloroquinolin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18ClN3O2
(5R)-9-(8-chloroquinolin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-3-methyl-9-(pyridin-4-ylmethyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H19N3O2
(5S)-3-methyl-9-(pyridin-4-ylmethyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[2-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C19H21N5O3
5-[2-[(3R)-3-(1H-benzimidazol-2-yl)piperidin-1-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (5S)-9-(8-chloroquinolin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18ClN3O2
(5S)-9-(8-chloroquinolin-2-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H25N5O3
(5R)-9-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5-fluoro-2-methoxyphenyl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate —— C18H16F2O4
(5-fluoro-2-methoxyphenyl)methyl (E)-3-(3-fluoro-4-methoxyphenyl)prop-2-enoate