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—— (5R,6R,7S)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25ClN4O3
(5R,6R,7S)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5R,6S,7R)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25ClN4O3
(5R,6S,7R)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5R,6S,7R)-3-cyano-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-5-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21N5O3
(5R,6S,7R)-3-cyano-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-5-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5R,10bS)-2-(3-chloro-4-ethoxyphenyl)-5-(2-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H23ClN2O2
(5R,10bS)-2-(3-chloro-4-ethoxyphenyl)-5-(2-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— [(5R,10bR)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-hydroxyphenyl)methanone —— C23H18N2O3
[(5R,10bR)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-hydroxyphenyl)methanone
—— (5R,6S,7R)-7-hydroxy-7-methyl-6-N,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C21H21N5O3
(5R,6S,7R)-7-hydroxy-7-methyl-6-N,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (5R,6S,7S)-7-hydroxy-N-(4-methoxyphenyl)-7-methyl-3,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N4O3
(5R,6S,7S)-7-hydroxy-N-(4-methoxyphenyl)-7-methyl-3,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5R,10bR)-9-bromo-5-(2-chloro-5-fluorophenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H15BrClFN2O
(5R,10bR)-9-bromo-5-(2-chloro-5-fluorophenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5,6-dimethyl-2-[[(1R)-1-[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]ethyl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C20H20N4O2S2
5,6-dimethyl-2-[[(1R)-1-[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]ethyl]sulfanylmethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5R,6R,7R)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25ClN4O3
(5R,6R,7R)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5R,6S,7S)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25ClN4O3
(5R,6S,7S)-5-(4-chlorophenyl)-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-3-phenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5S,10bS)-9-bromo-5-(4-ethoxy-3-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H21BrN2O3S
(5S,10bS)-9-bromo-5-(4-ethoxy-3-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,6R,7R)-7-hydroxy-N-(4-methoxyphenyl)-7-methyl-3,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N4O3
(5R,6R,7R)-7-hydroxy-N-(4-methoxyphenyl)-7-methyl-3,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5-Chloro-2-methoxyphenyl)[4-(5-chloro-2-methylphenyl)piperazin-1-yl]methanone —— C19H20Cl2N2O2
(5-Chloro-2-methoxyphenyl)[4-(5-chloro-2-methylphenyl)piperazin-1-yl]methanone
—— (5R,6R,7R)-5-(4-bromophenyl)-3-cyano-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H20BrN5O3
(5R,6R,7R)-5-(4-bromophenyl)-3-cyano-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (5R,6R,7S)-5-(4-bromophenyl)-3-cyano-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H20BrN5O3
(5R,6R,7S)-5-(4-bromophenyl)-3-cyano-7-hydroxy-N-(2-methoxyphenyl)-7-methyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— [(5S,10bR)-2-(4-bromophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-bromophenyl)methanone —— C23H16Br2N2O2
[(5S,10bR)-2-(4-bromophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-bromophenyl)methanone
—— (5S,10bS)-2-(3,4-dimethoxyphenyl)-5-methyl-5-pyridin-3-yl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C24H23N3O3
(5S,10bS)-2-(3,4-dimethoxyphenyl)-5-methyl-5-pyridin-3-yl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (5S,7R)-5-(3,4-dimethylphenyl)-7-(2,3,4-trimethoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C22H26N4O3
(5S,7R)-5-(3,4-dimethylphenyl)-7-(2,3,4-trimethoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— [(5S,10bS)-2-(4-bromophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-methylphenyl)methanone —— C24H19BrN2O2
[(5S,10bS)-2-(4-bromophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-methylphenyl)methanone
—— [(5S,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-phenylphenyl)methanone —— C27H20N2O2S
[(5S,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-phenylphenyl)methanone
—— (5R,10bS)-9-chloro-5-(3,4-dichlorophenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Cl3N2O
(5R,10bS)-9-chloro-5-(3,4-dichlorophenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-5-(2-chloro-5-fluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14ClFN2OS
(5S,10bR)-5-(2-chloro-5-fluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-2-(3-chloro-4-ethoxyphenyl)-5-(2-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H20ClFN2O2
(5R,10bR)-2-(3-chloro-4-ethoxyphenyl)-5-(2-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-9-bromo-5-(2-chloro-5-fluorophenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H15BrClFN2O
(5R,10bS)-9-bromo-5-(2-chloro-5-fluorophenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,7S)-7-phenyl-5-thiophen-2-yl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C15H14N4S
(5S,7S)-7-phenyl-5-thiophen-2-yl-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5R,10bR)-2-(3-chloro-4-ethoxyphenyl)-5-(2,3,4-trimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H27ClN2O5
(5R,10bR)-2-(3-chloro-4-ethoxyphenyl)-5-(2,3,4-trimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,6S,7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C21H20ClN5O2
(5S,6S,7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (5S,10bS)-9-bromo-2-(4-chlorophenyl)-5-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H18BrClN2O2
(5S,10bS)-9-bromo-2-(4-chlorophenyl)-5-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-2-(4-bromophenyl)-5-hexyl-5-methyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C23H27BrN2O
(5S,10bS)-2-(4-bromophenyl)-5-hexyl-5-methyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-5'-bromo-2-(2-chlorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one —— C23H15BrClN3O2
(5R,10bR)-5'-bromo-2-(2-chlorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one
—— (5R,6R,7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C21H20ClN5O2
(5R,6R,7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (5S,10bS)-2-(4-bromophenyl)-5-(2-chloro-6-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H15BrClFN2O
(5S,10bS)-2-(4-bromophenyl)-5-(2-chloro-6-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-9-chloro-5-ethyl-5-methyl-2-thiophen-2-yl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C17H17ClN2OS
(5R,10bS)-9-chloro-5-ethyl-5-methyl-2-thiophen-2-yl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-5-(4-bromophenyl)-9-chloro-2-(4-fluorophenyl)-5-methyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C23H17BrClFN2O
(5R,10bS)-5-(4-bromophenyl)-9-chloro-2-(4-fluorophenyl)-5-methyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-7,9-dichloro-2-(4-methylphenyl)-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H20Cl2N2O
(5R,10bS)-7,9-dichloro-2-(4-methylphenyl)-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bR)-2-(4-bromophenyl)-5-(5-chloro-2-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H15BrClFN2O
(5S,10bR)-2-(4-bromophenyl)-5-(5-chloro-2-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,6R,7S)-5-(3,4-dimethoxyphenyl)-6-N-(2,4-dimethylphenyl)-7-hydroxy-7-methyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C25H29N5O5
(5S,6R,7S)-5-(3,4-dimethoxyphenyl)-6-N-(2,4-dimethylphenyl)-7-hydroxy-7-methyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (5R,10bS)-9-bromo-5-(4-ethoxy-3-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H21BrN2O3S
(5R,10bS)-9-bromo-5-(4-ethoxy-3-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,6R,7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C21H20ClN5O2
(5S,6R,7R)-7-(4-chlorophenyl)-5-methyl-6-N-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (5R,10bS)-2-(4-bromophenyl)-5-methyl-5-propyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C20H21BrN2O
(5R,10bS)-2-(4-bromophenyl)-5-methyl-5-propyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-2-(3-chloro-4-ethoxyphenyl)-5-(2,3,4-trimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H27ClN2O5
(5R,10bS)-2-(3-chloro-4-ethoxyphenyl)-5-(2,3,4-trimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bR)-2-(3-chloro-4-ethoxyphenyl)-5-(2,5-dimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H25ClN2O4
(5R,10bR)-2-(3-chloro-4-ethoxyphenyl)-5-(2,5-dimethoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,6R,7S)-7-hydroxy-N-(4-methoxyphenyl)-7-methyl-3,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C27H26N4O3
(5R,6R,7S)-7-hydroxy-N-(4-methoxyphenyl)-7-methyl-3,5-diphenyl-5,6-dihydro-1H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— [(5S,10bS)-2-(4-bromophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-bromophenyl)methanone —— C23H16Br2N2O2
[(5S,10bS)-2-(4-bromophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-bromophenyl)methanone
—— [(5S,10bS)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-methylphenyl)methanone —— C28H22N2O2
[(5S,10bS)-2-naphthalen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-methylphenyl)methanone
—— (5R,10bS)-2-(3-chloro-4-ethoxyphenyl)-5-(2-chloro-6-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H19Cl2FN2O2
(5R,10bS)-2-(3-chloro-4-ethoxyphenyl)-5-(2-chloro-6-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,7S)-7-(3,4-dimethylphenyl)-5-(3-methoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H22N4O
(5S,7S)-7-(3,4-dimethylphenyl)-5-(3-methoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5R,10bS)-9-bromo-2-(4-chlorophenyl)-5-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H18BrClN2O2
(5R,10bS)-9-bromo-2-(4-chlorophenyl)-5-(2-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-9-chloro-5-(2-chloro-5-fluorophenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17Cl2FN2O2
(5R,10bS)-9-chloro-5-(2-chloro-5-fluorophenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine