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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-3-methyl-7-[(5-propylfuran-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H22N2O3
(5S)-3-methyl-7-[(5-propylfuran-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methyl-N-[(1S)-1-(2-pyrazol-1-ylphenyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H18N6
5-methyl-N-[(1S)-1-(2-pyrazol-1-ylphenyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H21N3O4
(5S)-9-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-Methyl-3-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,2-oxazole —— C18H21N5OS
5-Methyl-3-[(4-phenyl-5-piperidin-1-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,2-oxazole
—— (5R)-3-methyl-7-[(5-propylfuran-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H22N2O3
(5R)-3-methyl-7-[(5-propylfuran-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(1S)-1-[(2-cyclopentyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine —— C17H25N7S
5-[(1S)-1-[(2-cyclopentyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine
—— 5-chloro-1-[2-[(3R)-3-(4-chlorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione —— C25H16Cl2FN3O3
5-chloro-1-[2-[(3R)-3-(4-chlorophenyl)-5-(4-fluorophenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl]indole-2,3-dione
—— 5-chloro-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-1-benzofuran-2-carboxamide —— C20H23ClN4O2S
5-chloro-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-1-benzofuran-2-carboxamide
—— (5R)-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H30N4OS2
(5R)-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H30N4OS2
(5S)-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-methyl-2-[[(2R)-oxolan-2-yl]methylsulfanyl]-6-phenyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one —— C21H22N2O2S2
5-methyl-2-[[(2R)-oxolan-2-yl]methylsulfanyl]-6-phenyl-3-prop-2-enylthieno[2,3-d]pyrimidin-4-one
—— 5-chloro-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-2-methoxybenzamide —— C19H25ClN4O2S
5-chloro-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]-2-methoxybenzamide
—— 5-chloro-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]thiophene-2-carboxamide —— C16H21ClN4OS2
5-chloro-N-[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propyl]thiophene-2-carboxamide
—— [5-(5-methylthiophen-2-yl)-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl]methyl 2-(4-methylphenyl)acetate —— C21H18N2O3S2
[5-(5-methylthiophen-2-yl)-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl]methyl 2-(4-methylphenyl)acetate
—— 5-chloro-N-(3-chlorophenyl)-2-fluorobenzamide —— C13H8Cl2FNO
5-chloro-N-(3-chlorophenyl)-2-fluorobenzamide
—— (5R)-7-methyl-2-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H23N5O
(5R)-7-methyl-2-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-N-[(1R)-1-(2-pyrazol-1-ylphenyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H18N6
5-methyl-N-[(1R)-1-(2-pyrazol-1-ylphenyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-methyl-7-[(3S)-3-(1-methylbenzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C20H22N6
5-methyl-7-[(3S)-3-(1-methylbenzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5R)-7-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H22N4O3
(5R)-7-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methylphenyl)acetate —— C18H18N2O4
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(4-methylphenyl)acetate
—— (5-chloro-3-phenyl-1H-indol-2-yl)-[(2R)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone —— C20H17ClN2O2
(5-chloro-3-phenyl-1H-indol-2-yl)-[(2R)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone
—— 5-(4-fluorophenyl)-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(4-fluorophenyl)-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-methyl-7-[(3R)-3-(1-methylbenzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C20H22N6
5-methyl-7-[(3R)-3-(1-methylbenzimidazol-2-yl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5R)-9-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H21N3O4
(5R)-9-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-(4-fluorophenyl)-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C20H18FN5
5-(4-fluorophenyl)-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[4-[[(3S)-3-hydroxypiperidin-3-yl]methyl]piperazin-1-yl]-2-methylpyridazin-3-one —— C15H25N5O2
5-[4-[[(3S)-3-hydroxypiperidin-3-yl]methyl]piperazin-1-yl]-2-methylpyridazin-3-one
—— (5-chloro-3-phenyl-1H-indol-2-yl)-[(2S)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone —— C20H17ClN2O2
(5-chloro-3-phenyl-1H-indol-2-yl)-[(2S)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone
—— (5R)-9-[(4-fluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane —— C19H23FN4
(5R)-9-[(4-fluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane
—— 5-ethyl-7-[(3S)-3-phenylmethoxypiperidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C20H24N4O
5-ethyl-7-[(3S)-3-phenylmethoxypiperidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5S)-7-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H16ClN3O2
(5S)-7-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(3S)-3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazine-1-carbonyl]-1H-pyridin-2-one —— C20H25N3O3
5-[(3S)-3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazine-1-carbonyl]-1H-pyridin-2-one
—— (5R)-7-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H16ClN3O2
(5R)-7-(7-chloroquinolin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(2S)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine —— C20H27N3O
5-[[(2S)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine
—— 5-methyl-N-[(1R)-1-pyridin-3-ylpentyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H21N5
5-methyl-N-[(1R)-1-pyridin-3-ylpentyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[[(2R)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine —— C20H27N3O
5-[[(2R)-2-(3-methoxyphenyl)piperidin-1-yl]methyl]-N,N-dimethylpyridin-2-amine
—— 5-[(3R)-3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazine-1-carbonyl]-1H-pyridin-2-one —— C20H25N3O3
5-[(3R)-3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazine-1-carbonyl]-1H-pyridin-2-one
—— 5-methyl-N-[[(3S)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H21N5
5-methyl-N-[[(3S)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-[(4-fluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane —— C19H23FN4
(5S)-9-[(4-fluorophenyl)methyl]-2-pyrazin-2-yl-2,9-diazaspiro[4.5]decane
—— (5R)-9-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H25N5O2
(5R)-9-[[2-(benzylamino)pyrimidin-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]pyridine-2-carbonitrile —— C19H20N4O2
5-[(2S)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]pyridine-2-carbonitrile
—— 5-methyl-7-[(2R)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]pyrazolo[1,5-a]pyrimidine —— C19H23N5
5-methyl-7-[(2R)-2-methyl-4-(4-methylphenyl)piperazin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-methyl-N-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C18H21N5
5-methyl-N-[[(3R)-2-methyl-3,4-dihydro-1H-isoquinolin-3-yl]methyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]pyridine-2-carbonitrile —— C19H20N4O2
5-[(2R)-4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]pyridine-2-carbonitrile
—— (5R)-3-methyl-9-[(4-methylsulfanylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N2O2S
(5R)-3-methyl-9-[(4-methylsulfanylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[(2,3-difluorophenyl)methyl]-2-(1,3-dihydroxypropan-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24F2N2O3
(5S)-7-[(2,3-difluorophenyl)methyl]-2-(1,3-dihydroxypropan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-3-methyl-9-[(4-methylsulfanylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H22N2O2S
(5S)-3-methyl-9-[(4-methylsulfanylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-chloro-N-[5-(diethylsulfamoyl)-2,3-dimethylphenyl]thiophene-2-carboxamide —— C17H21ClN2O3S2
5-chloro-N-[5-(diethylsulfamoyl)-2,3-dimethylphenyl]thiophene-2-carboxamide
—— 5-methylsulfonyl-N-(2-morpholin-4-ylethyl)-4-[(3R)-piperidin-3-yl]pyrimidin-2-amine —— C16H27N5O3S
5-methylsulfonyl-N-(2-morpholin-4-ylethyl)-4-[(3R)-piperidin-3-yl]pyrimidin-2-amine
—— (5R)-7-amino-1'-[(4-fluorophenyl)methyl]-2,2',4-trioxospiro[1H-pyrano[2,3-d]pyrimidine-5,3'-indole]-6-carbonitrile —— C22H14FN5O4
(5R)-7-amino-1'-[(4-fluorophenyl)methyl]-2,2',4-trioxospiro[1H-pyrano[2,3-d]pyrimidine-5,3'-indole]-6-carbonitrile
—— (5R)-7-[(2,3-difluorophenyl)methyl]-2-(1,3-dihydroxypropan-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24F2N2O3
(5R)-7-[(2,3-difluorophenyl)methyl]-2-(1,3-dihydroxypropan-2-yl)-2,7-diazaspiro[4.5]decan-6-one