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—— (5S,7R)-5-[1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H28F3N5O2
(5S,7R)-5-[1-[(4-ethoxy-3-methoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-anilino-4-oxofuran-3-carboxylate —— C19H14N2O6
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-anilino-4-oxofuran-3-carboxylate
—— 5-[(Z)-N-[[4-(diethylamino)benzoyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylate —— C18H20N3O3S-
5-[(Z)-N-[[4-(diethylamino)benzoyl]amino]-C-methylcarbonimidoyl]thiophene-2-carboxylate
—— 5-[(3S,4R)-4-(4-fluorophenyl)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-3-yl]-1H-pyrazole —— C23H26FN3O2
5-[(3S,4R)-4-(4-fluorophenyl)-1-[[4-(2-methoxyethoxy)phenyl]methyl]pyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-4-(4-fluorophenyl)-1-[(2-methoxy-5-methylphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole —— C22H24FN3O
5-[(3S,4R)-4-(4-fluorophenyl)-1-[(2-methoxy-5-methylphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole
—— (5S,7R)-5-[1-[2-(benzenesulfonyl)ethyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H24F3N5O2S
(5S,7R)-5-[1-[2-(benzenesulfonyl)ethyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5S,7R)-5-[1-[[3-(2-methoxyethoxy)phenyl]methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H28F3N5O2
(5S,7R)-5-[1-[[3-(2-methoxyethoxy)phenyl]methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5S,7R)-5-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H26F3N5O2
(5S,7R)-5-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-[(3S,4R)-1-[(2-methoxy-5-methylphenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole —— C22H25N3O
5-[(3S,4R)-1-[(2-methoxy-5-methylphenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole
—— (5S,7R)-5-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H28F3N5O2
(5S,7R)-5-[1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5S,7R)-5-[1-[3-(2-fluorophenoxy)propyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H25F4N5O
(5S,7R)-5-[1-[3-(2-fluorophenoxy)propyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5S,7R)-5-[1-[(3-prop-2-ynoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H24F3N5O
(5S,7R)-5-[1-[(3-prop-2-ynoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfamoyl)-2-fluorobenzoate —— C16H13FNO6S-
5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfamoyl)-2-fluorobenzoate
—— 5-[(Z)-N-[(2,3-dimethylphenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C16H17N3O2S2
5-[(Z)-N-[(2,3-dimethylphenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— (5S,7R)-5-[1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H26F3N5O2
(5S,7R)-5-[1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-bromo-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)thiophene-2-sulfonamide —— C13H12BrNO4S2
5-bromo-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)thiophene-2-sulfonamide
—— (5S,7R)-5-[1-(4-phenoxybutyl)piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H28F3N5O
(5S,7R)-5-[1-(4-phenoxybutyl)piperidin-4-yl]-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-[(3S,4R)-4-(4-fluorophenyl)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole —— C21H22FN3O
5-[(3S,4R)-4-(4-fluorophenyl)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole
—— (5-methoxythiophen-2-yl)-[4-[(5S,7R)-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone —— C17H20F3N5O2S
(5-methoxythiophen-2-yl)-[4-[(5S,7R)-7-(trifluoromethyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]piperidin-1-yl]methanone
—— 5-[(Z)-N-[(2,4-dimethylphenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid —— C16H17N3O2S2
5-[(Z)-N-[(2,4-dimethylphenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylic acid
—— 5-[(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-(4-fluorophenyl)pyrrolidin-3-yl]-1H-pyrazole —— C23H26FN3O2
5-[(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-(4-fluorophenyl)pyrrolidin-3-yl]-1H-pyrazole
—— 5-[(Z)-N-[(4-ethoxyphenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylate —— C16H16N3O3S2-
5-[(Z)-N-[(4-ethoxyphenyl)carbamothioylamino]-C-methylcarbonimidoyl]thiophene-2-carboxylate
—— 5-[(3S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-(4-fluorophenyl)pyrrolidin-3-yl]-1H-pyrazole —— C22H24FN3O2
5-[(3S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-(4-fluorophenyl)pyrrolidin-3-yl]-1H-pyrazole
—— 5-methyl-3-[(4-methylpiperazin-1-yl)methyl]-2-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridine —— C15H19F3N4
5-methyl-3-[(4-methylpiperazin-1-yl)methyl]-2-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridine
—— 5-[[2-(Cyclopropylcarbamoyl)phenyl]sulfamoyl]-2-fluorobenzoate —— C17H14FN2O5S-
5-[[2-(Cyclopropylcarbamoyl)phenyl]sulfamoyl]-2-fluorobenzoate
—— 5-bromo-N-(2-hydroxy-5-nitrophenyl)thiophene-2-sulfonamide —— C10H7BrN2O5S2
5-bromo-N-(2-hydroxy-5-nitrophenyl)thiophene-2-sulfonamide
—— [5-[[(3S,4R)-3-(dimethylamino)-4-(5-methoxy-1-methylindol-3-yl)pyrrolidin-1-yl]methyl]-2-methoxyphenyl]methanol —— C25H33N3O3
[5-[[(3S,4R)-3-(dimethylamino)-4-(5-methoxy-1-methylindol-3-yl)pyrrolidin-1-yl]methyl]-2-methoxyphenyl]methanol
—— 5-[[2-(Cyclopropylcarbamoyl)phenyl]sulfamoyl]-2-fluorobenzoic acid —— C17H15FN2O5S
5-[[2-(Cyclopropylcarbamoyl)phenyl]sulfamoyl]-2-fluorobenzoic acid
—— (5-Chloro-2-methoxyphenyl)methyl 2-anilino-4-oxofuran-3-carboxylate —— C19H16ClNO5
(5-Chloro-2-methoxyphenyl)methyl 2-anilino-4-oxofuran-3-carboxylate
—— 5-[[2-[[(2R)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoic acid —— C18H19FN2O5S
5-[[2-[[(2R)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoic acid
—— 5-[(3S,4R)-1-[(3,4-difluorophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole —— C21H21F2N3O
5-[(3S,4R)-1-[(3,4-difluorophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole —— C23H27N3O2
5-[(3S,4R)-1-[(4-ethoxy-3-methoxyphenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole
—— 5-[[2-[[(2S)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoate —— C18H18FN2O5S-
5-[[2-[[(2S)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoate
—— 5-methoxy-2-[[[(1R,2S)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]cyclopentyl]amino]methyl]phenol —— C18H24N2O3
5-methoxy-2-[[[(1R,2S)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]cyclopentyl]amino]methyl]phenol
—— 5-[(3S,4R)-4-phenyl-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-pyrazole —— C21H23N3
5-[(3S,4R)-4-phenyl-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-pyrazole
—— [5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-anilino-4-oxofuran-3-carboxylate —— C21H15ClN2O5
[5-(4-Chlorophenyl)-1,3-oxazol-2-yl]methyl 2-anilino-4-oxofuran-3-carboxylate
—— 5-[(3S,4R)-4-(4-methoxyphenyl)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole —— C22H25N3O2
5-[(3S,4R)-4-(4-methoxyphenyl)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-1-[(2-fluorophenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole —— C20H20FN3
5-[(3S,4R)-1-[(2-fluorophenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole
—— 5-[[2-[[(2S)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoic acid —— C18H19FN2O5S
5-[[2-[[(2S)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoic acid
—— 5-[(3S,4R)-1-[[(3R)-oxolan-3-yl]methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole —— C18H23N3O
5-[(3S,4R)-1-[[(3R)-oxolan-3-yl]methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-1-[(3-fluorophenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole —— C20H20FN3
5-[(3S,4R)-1-[(3-fluorophenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-1-(2,2-dimethyl-3-pyrrolidin-1-ylpropyl)-4-phenylpyrrolidin-3-yl]-1H-pyrazole —— C22H32N4
5-[(3S,4R)-1-(2,2-dimethyl-3-pyrrolidin-1-ylpropyl)-4-phenylpyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole —— C24H29N3O2
5-[(3S,4R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole
—— 5-[[2-[[(2R)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoate —— C18H18FN2O5S-
5-[[2-[[(2R)-butan-2-yl]carbamoyl]phenyl]sulfamoyl]-2-fluorobenzoate
—— 5-[(3S,4R)-1-(2-methoxy-5-methylphenyl)sulfonyl-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole —— C22H25N3O4S
5-[(3S,4R)-1-(2-methoxy-5-methylphenyl)sulfonyl-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole —— C23H27N3O
5-[(3S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-phenylpyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-4-(4-methoxyphenyl)-1-[(3,4,5-trimethoxyphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole —— C24H29N3O4
5-[(3S,4R)-4-(4-methoxyphenyl)-1-[(3,4,5-trimethoxyphenyl)methyl]pyrrolidin-3-yl]-1H-pyrazole
—— 5-[(3S,4R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole —— C24H29N3O3
5-[(3S,4R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole
—— [5-[[(3S,4R)-3-(dimethylamino)-4-(1-methylindol-3-yl)pyrrolidin-1-yl]methyl]-2-methoxyphenyl]methanol —— C24H31N3O2
[5-[[(3S,4R)-3-(dimethylamino)-4-(1-methylindol-3-yl)pyrrolidin-1-yl]methyl]-2-methoxyphenyl]methanol
—— 5-[(3S,4R)-1-[(3-fluorophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole —— C21H22FN3O
5-[(3S,4R)-1-[(3-fluorophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]-1H-pyrazole