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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-9-[3-(5-methyl-2-oxo-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H21N3O5
(5S)-9-[3-(5-methyl-2-oxo-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[3-oxo-3-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]propyl]-1,2-oxazol-3-one —— C20H25N3O3
5-[3-oxo-3-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]propyl]-1,2-oxazol-3-one
—— (5S)-7-(4-tert-butylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H24N2O3
(5S)-7-(4-tert-butylbenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5-chloro-2-methoxyphenyl)-[(3R)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-3-yl]methanone —— C20H24ClN3O3
(5-chloro-2-methoxyphenyl)-[(3R)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-3-yl]methanone
—— 5-(Furan-2-yl)-3-phenyl-2-prop-2-enylsulfanylthieno[2,3-d]pyrimidin-4-one —— C19H14N2O2S2
5-(Furan-2-yl)-3-phenyl-2-prop-2-enylsulfanylthieno[2,3-d]pyrimidin-4-one
—— (5R)-3-methyl-9-(6-methyl-2-oxo-1H-pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H19N3O4
(5R)-3-methyl-9-(6-methyl-2-oxo-1H-pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(2S)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C17H22N4O2
5-[[(2S)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5S)-3-methyl-9-(6-methyl-2-oxo-1H-pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H19N3O4
(5S)-3-methyl-9-(6-methyl-2-oxo-1H-pyridine-3-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-ethoxy-1-[[(3S)-3-hydroxypiperidin-1-yl]methyl]-3-[[(3R)-3-hydroxypiperidin-1-yl]methyl]benzimidazole-2-thione —— C21H32N4O3S
5-ethoxy-1-[[(3S)-3-hydroxypiperidin-1-yl]methyl]-3-[[(3R)-3-hydroxypiperidin-1-yl]methyl]benzimidazole-2-thione
—— 5-[(5S)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carbonyl]pyridine-2-carbonitrile —— C16H18N4O3
5-[(5S)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carbonyl]pyridine-2-carbonitrile
—— (5R)-9-(1,3-thiazol-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C13H18N2O2S
(5R)-9-(1,3-thiazol-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-pyrrolidin-3-yl]pyridin-2-amine —— C18H19N5O
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3S)-pyrrolidin-3-yl]pyridin-2-amine
—— (5R)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5R)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3R)-pyrrolidin-3-yl]pyridin-2-amine —— C18H19N5O
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(3R)-pyrrolidin-3-yl]pyridin-2-amine
—— 5-[2-[(1-Phenyl-4,5,6,7-tetrahydrobenzimidazol-2-yl)sulfanyl]acetyl]-1,3-dihydroindol-2-one —— C23H21N3O2S
5-[2-[(1-Phenyl-4,5,6,7-tetrahydrobenzimidazol-2-yl)sulfanyl]acetyl]-1,3-dihydroindol-2-one
—— 5-[[(5R)-5-[bis(carboxymethyl)amino]-5-carboxypentyl]carbamothioylamino]-2-(3-hydroxy-6-oxoxanthen-9-yl)benzoic acid —— C31H29N3O11S
5-[[(5R)-5-[bis(carboxymethyl)amino]-5-carboxypentyl]carbamothioylamino]-2-(3-hydroxy-6-oxoxanthen-9-yl)benzoic acid
—— 5,6-diamino-3-[(2R)-butan-2-yl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxo-1H-pyrrolo[2,3-c][2,7]naphthyridine-9-carbonitrile —— C21H27N7O2
5,6-diamino-3-[(2R)-butan-2-yl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxo-1H-pyrrolo[2,3-c][2,7]naphthyridine-9-carbonitrile
—— (5R)-9-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H24N4O4
(5R)-9-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5S)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(1,3-thiazol-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one —— C13H18N2O2S
(5S)-9-(1,3-thiazol-2-ylmethyl)-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H24N4O4
(5S)-9-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-ethoxy-1-[[(3S)-3-hydroxypiperidin-1-ium-1-yl]methyl]-3-[[(3R)-3-hydroxypiperidin-1-ium-1-yl]methyl]benzimidazole-2-thione —— C21H34N4O3S+2
5-ethoxy-1-[[(3S)-3-hydroxypiperidin-1-ium-1-yl]methyl]-3-[[(3R)-3-hydroxypiperidin-1-ium-1-yl]methyl]benzimidazole-2-thione
—— (5R,10bS)-2-(4-fluorophenyl)-5-[2-(trifluoromethyl)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H16F4N2O
(5R,10bS)-2-(4-fluorophenyl)-5-[2-(trifluoromethyl)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(5R)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carbonyl]pyridine-2-carbonitrile —— C16H18N4O3
5-[(5R)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carbonyl]pyridine-2-carbonitrile
—— (5-chloro-2-methoxyphenyl)-[(3S)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-3-yl]methanone —— C20H24ClN3O3
(5-chloro-2-methoxyphenyl)-[(3S)-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)piperidin-3-yl]methanone
—— (5R)-9-[2-(1H-imidazol-2-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18N4O3
(5R)-9-[2-(1H-imidazol-2-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[2-(1H-imidazol-2-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H18N4O3
(5S)-9-[2-(1H-imidazol-2-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H20N4O4
(5S)-7-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[[(2R)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C17H22N4O2
5-[[(2R)-2-(2-phenylethyl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-(1H-indol-5-ylmethyl)-2-[[(2S)-2-methylpyrrolidin-1-yl]methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine —— C22H29N5
5-(1H-indol-5-ylmethyl)-2-[[(2S)-2-methylpyrrolidin-1-yl]methyl]-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine
—— 5-[[4-[(3S)-3-(aminomethyl)pyrrolidin-1-yl]-6-oxopyridazin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide —— C17H23N5O3
5-[[4-[(3S)-3-(aminomethyl)pyrrolidin-1-yl]-6-oxopyridazin-1-yl]methyl]-N,N-dimethylfuran-2-carboxamide
—— (5R,7S)-7-(1,3-benzodioxol-5-yl)-5-(4-bromophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H15BrN4O2
(5R,7S)-7-(1,3-benzodioxol-5-yl)-5-(4-bromophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-[(3R)-3-[2-(dimethylamino)ethyl-methylamino]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C20H29N5O2
5-[(3R)-3-[2-(dimethylamino)ethyl-methylamino]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— (5S)-9-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H21N3O5
(5S)-9-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H22N4O3
(5R)-7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S,7R)-7-(1,3-benzodioxol-5-yl)-5-(4-bromophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H15BrN4O2
(5S,7R)-7-(1,3-benzodioxol-5-yl)-5-(4-bromophenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-(4-chlorophenyl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)-3H-thieno[2,3-d]pyrimidin-4-one —— C18H16ClN3O2S
5-(4-chlorophenyl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)-3H-thieno[2,3-d]pyrimidin-4-one
—— (5R)-7-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H20N4O4
(5R)-7-[1-(2-methoxyphenyl)pyrazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-ethyl-N-(6-fluoro-1,3-benzothiazol-2-yl)-4-methylthiophene-2-carboxamide —— C15H13FN2OS2
5-ethyl-N-(6-fluoro-1,3-benzothiazol-2-yl)-4-methylthiophene-2-carboxamide
—— 5-[(3S)-3-[2-(dimethylamino)ethyl-methylamino]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C20H29N5O2
5-[(3S)-3-[2-(dimethylamino)ethyl-methylamino]piperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— 5-bromo-N-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)pyridine-3-carboxamide —— C20H15BrN4O
5-bromo-N-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)pyridine-3-carboxamide
—— (5S)-3-methyl-7-[3-(5-methyl-2-oxo-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H21N3O5
(5S)-3-methyl-7-[3-(5-methyl-2-oxo-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(4-fluorophenyl)sulfamoyl]-2-methyl-N-(pyridin-2-ylmethyl)benzamide —— C20H18FN3O3S
5-[(4-fluorophenyl)sulfamoyl]-2-methyl-N-(pyridin-2-ylmethyl)benzamide
—— (5R)-3-methyl-7-[3-(5-methyl-2-oxo-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H21N3O5
(5R)-3-methyl-7-[3-(5-methyl-2-oxo-1,3-benzoxazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-3-methyl-9-[2-(1,2,4-triazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C13H19N5O3
(5R)-3-methyl-9-[2-(1,2,4-triazol-1-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-7-(7-oxo-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H14N4O4S
(5S)-3-methyl-7-(7-oxo-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[(1R)-1-(benzylsulfamoylamino)ethyl]-1,3,4-thiadiazol-2-amine —— C11H15N5O2S2
5-[(1R)-1-(benzylsulfamoylamino)ethyl]-1,3,4-thiadiazol-2-amine
—— (5S)-5-(4-nitrophenyl)-N-(2-phenylethyl)-4,5-dihydro-1,3-thiazol-2-amine —— C17H17N3O2S
(5S)-5-(4-nitrophenyl)-N-(2-phenylethyl)-4,5-dihydro-1,3-thiazol-2-amine
—— 5-methoxy-3-methyl-N-quinolin-5-yl-1-benzofuran-2-carboxamide —— C20H16N2O3
5-methoxy-3-methyl-N-quinolin-5-yl-1-benzofuran-2-carboxamide
—— (5S)-3-methyl-9-(3-pyridin-2-ylpropanoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H23N3O3
(5S)-3-methyl-9-(3-pyridin-2-ylpropanoyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one