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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C14H19N3O
(5S)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H22N4O3
(5S)-9-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H22N4O3
(5R)-9-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3R)-3-(3,4-difluoroanilino)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C18H20F2N6O
5-[[(3R)-3-(3,4-difluoroanilino)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— (5S)-9-(2,8-dimethylquinoline-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H23N3O3
(5S)-9-(2,8-dimethylquinoline-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-propan-2-yl-7-[(3S)-3-(propoxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C17H26N4O
5-propan-2-yl-7-[(3S)-3-(propoxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— (5R)-7-(2-cyclohexylethyl)-2-(2-hydroxy-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C24H34N2O3
(5R)-7-(2-cyclohexylethyl)-2-(2-hydroxy-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(quinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H19N3O3
(5S)-9-(quinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O4
(5S)-3-methyl-9-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[2-(3,4-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H27NO3
(5R)-9-[2-(3,4-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5,6-dimethyl-N-[[(6S)-4-methyl-1,4-oxazepan-6-yl]methyl]-2-(trifluoromethyl)pyrimidin-4-amine —— C14H21F3N4O
5,6-dimethyl-N-[[(6S)-4-methyl-1,4-oxazepan-6-yl]methyl]-2-(trifluoromethyl)pyrimidin-4-amine
—— (5R)-3-methyl-7-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H21N5O3
(5R)-3-methyl-7-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— [(5R)-9-(2-methoxyethyl)-2,9-diazaspiro[4.5]decan-2-yl]-phenylmethanone —— C18H26N2O2
[(5R)-9-(2-methoxyethyl)-2,9-diazaspiro[4.5]decan-2-yl]-phenylmethanone
—— 5-ethyl-N-[(3R)-5-oxo-1-[[2-(trifluoromethyl)phenyl]methyl]pyrrolidin-3-yl]-1,2-oxazole-4-carboxamide —— C18H18F3N3O3
5-ethyl-N-[(3R)-5-oxo-1-[[2-(trifluoromethyl)phenyl]methyl]pyrrolidin-3-yl]-1,2-oxazole-4-carboxamide
—— [5-(3,4,5-Trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl 6-chloropyridine-3-carboxylate —— C18H16ClN3O6
[5-(3,4,5-Trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]methyl 6-chloropyridine-3-carboxylate
—— [5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 6-chloropyridine-3-carboxylate —— C15H9Cl2N3O3
[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl 6-chloropyridine-3-carboxylate
—— 5-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C18H24N4O3
5-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— 5-propan-2-yl-7-[(3R)-3-(propoxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine —— C17H26N4O
5-propan-2-yl-7-[(3R)-3-(propoxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine
—— 5-methyl-2-[(E)-2-(3-nitrophenyl)ethenyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C16H10N3O5S-
5-methyl-2-[(E)-2-(3-nitrophenyl)ethenyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— (5R)-3-methyl-9-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O4
(5R)-3-methyl-9-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(1S)-1-[(4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine —— C11H11ClN6S
5-[(1S)-1-[(4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine
—— 5-ethyl-N-[(3S)-5-oxo-1-[[2-(trifluoromethyl)phenyl]methyl]pyrrolidin-3-yl]-1,2-oxazole-4-carboxamide —— C18H18F3N3O3
5-ethyl-N-[(3S)-5-oxo-1-[[2-(trifluoromethyl)phenyl]methyl]pyrrolidin-3-yl]-1,2-oxazole-4-carboxamide
—— 5-phenyl-2-[(4-pyridin-1-ium-2-ylpiperazin-1-ium-1-yl)methyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C22H23N5OS+2
5-phenyl-2-[(4-pyridin-1-ium-2-ylpiperazin-1-ium-1-yl)methyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5R)-3-methyl-7-(5-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H20N4O3
(5R)-3-methyl-7-(5-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[2-(benzotriazol-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H19N5O3
(5R)-9-[2-(benzotriazol-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[2-(benzotriazol-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H19N5O3
(5S)-9-[2-(benzotriazol-2-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-7-[3-(1,2,4-triazol-4-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H17N5O3
(5S)-3-methyl-7-[3-(1,2,4-triazol-4-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-7-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H21N5O3
(5S)-3-methyl-7-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-(quinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H19N3O3
(5R)-9-(quinoline-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-3-methyl-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H26N4O2
(5S)-3-methyl-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-chloro-N-[(3S)-1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]-2-methoxybenzamide —— C19H18ClFN2O3
5-chloro-N-[(3S)-1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]-2-methoxybenzamide
—— (5S)-7-(5-hydroxy-1,2-dimethylindole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H21N3O4
(5S)-7-(5-hydroxy-1,2-dimethylindole-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-3-methyl-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H26N4O2
(5R)-3-methyl-9-[(2-propan-2-ylpyrimidin-4-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-[2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H21N3O3S2
(5R)-3-methyl-9-[2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-5-methyl-N-(3-morpholin-4-ylsulfonylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H24N2O4S2
(5R)-5-methyl-N-(3-morpholin-4-ylsulfonylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-9-[2-(3,4-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C19H27NO3
(5S)-9-[2-(3,4-dimethylphenoxy)ethyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5,6-dimethyl-N-[[(6R)-4-methyl-1,4-oxazepan-6-yl]methyl]-2-(trifluoromethyl)pyrimidin-4-amine —— C14H21F3N4O
5,6-dimethyl-N-[[(6R)-4-methyl-1,4-oxazepan-6-yl]methyl]-2-(trifluoromethyl)pyrimidin-4-amine
—— 5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole —— C17H20FN5O2
5-[[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
—— 5-[(1R)-1-[(4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine —— C11H11ClN6S
5-[(1R)-1-[(4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]ethyl]-1,3,4-thiadiazol-2-amine
—— (5R)-3-methyl-9-(2,3,6-trimethylquinoline-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C21H25N3O3
(5R)-3-methyl-9-(2,3,6-trimethylquinoline-4-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(5-phenoxyfuran-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H18N2O5
(5S)-9-(5-phenoxyfuran-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-(2-methoxyethyl)-2-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O3
(5R)-7-(2-methoxyethyl)-2-[2-[methyl(pyridin-3-ylmethyl)amino]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(6-methylpyridine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H19N3O3
(5R)-9-(6-methylpyridine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5-chloropyridin-3-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C20H22ClN3O
(5-chloropyridin-3-yl)-[4-[(2S)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5R)-9-(1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H19N3O3S
(5R)-9-(1,3-benzothiazole-6-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(2R)-2-(3-methoxyphenyl)pyrrolidin-1-yl]sulfonyl-3H-1,3-benzoxazol-2-one —— C18H18N2O5S
5-[(2R)-2-(3-methoxyphenyl)pyrrolidin-1-yl]sulfonyl-3H-1,3-benzoxazol-2-one
—— (5S)-9-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H21N5O3S
(5S)-9-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H22N4O4
(5R)-7-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C16H22N4O4
(5S)-7-[2-(4-acetyl-3,5-dimethylpyrazol-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-9-(6-methylpyridine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H19N3O3
(5S)-9-(6-methylpyridine-2-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one