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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(3S)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C19H23N3O4
5-[(3S)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— 5-methyl-1-[2-[(3S)-3-[methyl(2-phenylethyl)amino]piperidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C21H28N4O3
5-methyl-1-[2-[(3S)-3-[methyl(2-phenylethyl)amino]piperidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— (5R)-7-[3-(1H-benzimidazol-2-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H20N4O3
(5R)-7-[3-(1H-benzimidazol-2-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-7-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H17ClN2O5
(5S)-7-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-methyl-1-[2-[(3R)-3-[methyl(2-phenylethyl)amino]piperidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C21H28N4O3
5-methyl-1-[2-[(3R)-3-[methyl(2-phenylethyl)amino]piperidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— 5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(2-phenylsulfanylethyl)pyridazin-3-one —— C18H24N4O2S
5-[(2S)-2-(2-aminoethyl)morpholin-4-yl]-2-(2-phenylsulfanylethyl)pyridazin-3-one
—— (5S)-9-[2-(4-phenylphenyl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C22H24N2O3
(5S)-9-[2-(4-phenylphenyl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-9-(4H-thieno[3,2-b]pyrrole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H19N3O3S
(5R)-3-methyl-9-(4H-thieno[3,2-b]pyrrole-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H17N3O3S2
(5R)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[4-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]sulfonylphenyl]-1,3-oxazole —— C18H17N3O3S
5-[4-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]sulfonylphenyl]-1,3-oxazole
—— (5S)-9-[4-(3,5-dimethylpyrazol-1-yl)butanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H28N4O3
(5S)-9-[4-(3,5-dimethylpyrazol-1-yl)butanoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-3-methyl-7-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H17N5O3
(5R)-3-methyl-7-(2-pyridin-3-ylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-(3-phenylpropyl)-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H30N4O
(5R)-7-(3-phenylpropyl)-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H17N3O3S2
(5S)-9-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H25N3O3
(5R)-9-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[4-(difluoromethoxy)benzoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20F2N2O4
(5S)-9-[4-(difluoromethoxy)benzoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— [5-(2-Bromophenyl)-1,3,4-oxadiazol-2-yl]methyl 6-chloropyridine-3-carboxylate —— C15H9BrClN3O3
[5-(2-Bromophenyl)-1,3,4-oxadiazol-2-yl]methyl 6-chloropyridine-3-carboxylate
—— 5-[[(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]methyl]-2-methylsulfanylpyrimidine —— C15H21N5S
5-[[(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]methyl]-2-methylsulfanylpyrimidine
—— (5R)-2-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H33N5O2
(5R)-2-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(1-ethylindol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H27N3O2
(5R)-9-[(1-ethylindol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20FN3O3
(5S)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-(6-ethyl-1,5-dimethyl-2-oxopyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H23N3O4
(5S)-7-(6-ethyl-1,5-dimethyl-2-oxopyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-2-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H33N5O2
(5S)-2-(6-ethyl-2-pyrrolidin-1-ylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-methyl-7-[3-(1,2,4-triazol-4-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H17N5O3
(5R)-3-methyl-7-[3-(1,2,4-triazol-4-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-chloro-3-[(3R)-3-(3,4-dimethylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one —— C19H22ClN3O2
5-chloro-3-[(3R)-3-(3,4-dimethylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one
—— (5S)-9-[(1-ethylindol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H27N3O2
(5S)-9-[(1-ethylindol-4-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[4-(difluoromethoxy)benzoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20F2N2O4
(5R)-9-[4-(difluoromethoxy)benzoyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(4-methyl-2-phenylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H22N4O3
(5R)-9-(4-methyl-2-phenylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]quinoxaline —— C21H24N4O
5-[[(2R)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]quinoxaline
—— (5R)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H20FN3O3
(5R)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(4-methyl-2-phenylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H22N4O3
(5S)-9-(4-methyl-2-phenylpyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-chloro-3-[(3S)-3-(3,4-dimethylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one —— C19H22ClN3O2
5-chloro-3-[(3S)-3-(3,4-dimethylanilino)piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5-[[(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]methyl]-2-methylsulfanylpyrimidine —— C15H21N5S
5-[[(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]methyl]-2-methylsulfanylpyrimidine
—— (5S)-9-[3-(5-methyltetrazol-1-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N6O3
(5S)-9-[3-(5-methyltetrazol-1-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[4-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]sulfonylphenyl]-1,3-oxazole —— C18H17N3O3S
5-[4-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]sulfonylphenyl]-1,3-oxazole
—— 5-[[(4S)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C14H21N5O3
5-[[(4S)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— (5R)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C14H19N3O
(5R)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(2,8-dimethylquinoline-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C20H23N3O3
(5R)-9-(2,8-dimethylquinoline-4-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]quinoxaline —— C21H24N4O
5-[[(2S)-4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl]quinoxaline
—— 5-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C18H24N4O3
5-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— (5R)-9-[2-oxo-6-(trifluoromethyl)-1H-pyridine-3-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H14F3N3O4
(5R)-9-[2-oxo-6-(trifluoromethyl)-1H-pyridine-3-carbonyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-2-[2-(diethylamino)acetyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H30FN3O2
(5R)-2-[2-(diethylamino)acetyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[3-(5-methyltetrazol-1-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H18N6O3
(5R)-9-[3-(5-methyltetrazol-1-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[[(4R)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C14H21N5O3
5-[[(4R)-4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— (5S)-3-methyl-9-(3-phenyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H21N3O4
(5S)-3-methyl-9-(3-phenyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H20N2O5
(5S)-9-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[[(3S)-3-(3,4-difluoroanilino)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one —— C18H20F2N6O
5-[[(3S)-3-(3,4-difluoroanilino)piperidin-1-yl]methyl]-2-methyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
—— 5-[[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C17H20F2N4O2
5-[[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— (5R)-3-methyl-9-(3-phenyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H21N3O4
(5R)-3-methyl-9-(3-phenyl-1,2-oxazole-4-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-2-[2-(diethylamino)acetyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H30FN3O2
(5S)-2-[2-(diethylamino)acetyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one