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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-3-methyl-9-(3-methyltriazolo[4,5-b]pyridine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H20N6O3
(5S)-3-methyl-9-(3-methyltriazolo[4,5-b]pyridine-6-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3R)-3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C19H24FN5O2
5-[(3R)-3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— (5R)-7-methyl-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2S
(5R)-7-methyl-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-3-methyl-9-[3-(2-methylimidazol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5R)-3-methyl-9-[3-(2-methylimidazol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-5-(2-chlorophenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione —— C19H14ClN3O2
(5S)-5-(2-chlorophenyl)-2-phenyl-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-dione
—— (5R)-9-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H25N3O3
(5R)-9-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(3,4-dihydro-2H-chromene-6-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N2O4
(5R)-9-(3,4-dihydro-2H-chromene-6-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5-bromofuran-2-yl)[3-(4-fluorophenyl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl]methanone —— C17H13BrFN3O2
(5-bromofuran-2-yl)[3-(4-fluorophenyl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl]methanone
—— 5-bromo-2-(ethylsulfanyl)-N-(4-phenyl-1,2,5-oxadiazol-3-yl)pyrimidine-4-carboxamide —— C15H12BrN5O2S
5-bromo-2-(ethylsulfanyl)-N-(4-phenyl-1,2,5-oxadiazol-3-yl)pyrimidine-4-carboxamide
—— (5S)-7-methyl-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2S
(5S)-7-methyl-2-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(furan-2-yl)-3-(1H-1,2,4-triazol-5-ylamino)cyclohex-2-en-1-one —— C12H12N4O2
(5S)-5-(furan-2-yl)-3-(1H-1,2,4-triazol-5-ylamino)cyclohex-2-en-1-one
—— (5R)-9-(2-ethoxybenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H24N2O4
(5R)-9-(2-ethoxybenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[4-(2-Methoxybenzoyl)piperazin-1-yl]-2-(2-methoxyphenyl)-1,3-oxazole-4-carbonitrile —— C23H22N4O4
5-[4-(2-Methoxybenzoyl)piperazin-1-yl]-2-(2-methoxyphenyl)-1,3-oxazole-4-carbonitrile
—— (5S)-9-[2-(2-ethyl-6-methylpyridin-3-yl)oxyacetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H25N3O4
(5S)-9-[2-(2-ethyl-6-methylpyridin-3-yl)oxyacetyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C18H18ClN3O4
(5S)-7-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-(benzyl(methyl)amino)-4-bromo-2-phenylpyridazin-3(2H)-one —— C18H16BrN3O
5-(benzyl(methyl)amino)-4-bromo-2-phenylpyridazin-3(2H)-one
—— (5S)-9-(2-ethoxybenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H24N2O4
(5S)-9-(2-ethoxybenzoyl)-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H25N3O3
(5S)-9-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-propan-2-yl-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H21N5
5-propan-2-yl-N-[(1R)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R,7R)-7-(3-fluorophenyl)-5-(4-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine —— C17H16FN5O
(5R,7R)-7-(3-fluorophenyl)-5-(4-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine
—— (5R,7S)-7-(3-fluorophenyl)-5-(4-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine —— C17H16FN5O
(5R,7S)-7-(3-fluorophenyl)-5-(4-methoxyphenyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine
—— (5R)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C15H23N3O4
(5R)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— 5-ethoxy-1-(4-methoxybenzyl)-1H-indole-2,3-dione —— C18H17NO4
5-ethoxy-1-(4-methoxybenzyl)-1H-indole-2,3-dione
—— 5-ethyl-N-[(3S)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl]-1,2-oxazole-4-carboxamide —— C18H20FN3O3
5-ethyl-N-[(3S)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl]-1,2-oxazole-4-carboxamide
—— 5-[[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C18H23FN4O2
5-[[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— (5R)-7-(2-cyclohexylethyl)-2-[3-(tetrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H32N6O2
(5R)-7-(2-cyclohexylethyl)-2-[3-(tetrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(2-anilinopyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H19N5O3
(5S)-9-(2-anilinopyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane —— C17H26N2O2
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
—— (5S)-3-methyl-7-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H15N3O3S2
(5S)-3-methyl-7-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-ethyl-N-[(3S)-1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]-4-methyl-1H-pyrazole-3-carboxamide —— C18H21FN4O2
5-ethyl-N-[(3S)-1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl]-4-methyl-1H-pyrazole-3-carboxamide
—— 5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C18H23FN4O2
5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— (5R)-9-(2-anilinopyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C18H19N5O3
(5R)-9-(2-anilinopyrimidine-5-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-ethyl-N-[(3R)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl]-1,2-oxazole-4-carboxamide —— C18H20FN3O3
5-ethyl-N-[(3R)-1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl]-1,2-oxazole-4-carboxamide
—— 5-propan-2-yl-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H21N5
5-propan-2-yl-N-[(1S)-1-pyridin-3-ylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane —— C17H26N2O2
(5S)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
—— 5-methyl-4-[(1S)-3-oxo-1H-2-benzofuran-1-yl]-1,2-dihydropyrazol-3-one —— C12H10N2O3
5-methyl-4-[(1S)-3-oxo-1H-2-benzofuran-1-yl]-1,2-dihydropyrazol-3-one
—— 5-[(3S)-3-(1,3-benzodioxol-5-ylamino)piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H20N4O4
5-[(3S)-3-(1,3-benzodioxol-5-ylamino)piperidine-1-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— 5-[[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23N5O3
5-[[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 5-methyl-4-[(1R)-3-oxo-1H-2-benzofuran-1-yl]-1,2-dihydropyrazol-3-one —— C12H10N2O3
5-methyl-4-[(1R)-3-oxo-1H-2-benzofuran-1-yl]-1,2-dihydropyrazol-3-one
—— 5-[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C20H24N4O4
5-[(3R)-3-(1,3-benzodioxol-5-ylamino)piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— (5S)-9-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H24N4O3
(5S)-9-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(3-chloro-5-fluorobenzoyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H14ClFN2O3
(5S)-9-(3-chloro-5-fluorobenzoyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5,5-Dimethyl-2-(piperidine-1-carbonylamino)-4,7-dihydrothieno[2,3-c]pyran-3-carboxylate —— C16H21N2O4S-
5,5-Dimethyl-2-(piperidine-1-carbonylamino)-4,7-dihydrothieno[2,3-c]pyran-3-carboxylate
—— [5-(methoxymethyl)furan-2-yl]-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone —— C21H26N2O3
[5-(methoxymethyl)furan-2-yl]-[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methanone
—— (5R)-7-[2-(1H-imidazol-2-yl)benzoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H18N4O3
(5R)-7-[2-(1H-imidazol-2-yl)benzoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C17H19N5O3
(5R)-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-7-[2-(1H-imidazol-2-yl)benzoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H18N4O3
(5S)-7-[2-(1H-imidazol-2-yl)benzoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5S)-3-methyl-7-(6,7,8,9-tetrahydro-5H-carbazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C20H23N3O3
(5S)-3-methyl-7-(6,7,8,9-tetrahydro-5H-carbazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-9-(5-ethyl-4-methyl-1H-pyrazole-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5R)-9-(5-ethyl-4-methyl-1H-pyrazole-3-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-3-methyl-7-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H15N3O3S2
(5R)-3-methyl-7-(2-thiophen-2-yl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one