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—— 5-ethyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H21N5
5-ethyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-9-[3-(2-ethylimidazol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C15H22N4O3
(5R)-9-[3-(2-ethylimidazol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H17N5O3
(5R)-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-(2,2-dimethylpropyl)-2-(6-methyl-4-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O3
(5S)-7-(2,2-dimethylpropyl)-2-(6-methyl-4-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-N-(6-chloropyridin-3-yl)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide —— C15H19ClN4O3
(5R)-N-(6-chloropyridin-3-yl)-3-methyl-2-oxo-1-oxa-3,9-diazaspiro[4.6]undecane-9-carboxamide
—— (5S)-5-(2-phenylethyl)-2-[2-(trifluoromethyl)phenyl]-5,6-dihydropyrazolo[3,4-e][1,3]oxazin-7-one —— C20H16F3N3O2
(5S)-5-(2-phenylethyl)-2-[2-(trifluoromethyl)phenyl]-5,6-dihydropyrazolo[3,4-e][1,3]oxazin-7-one
—— 5-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C17H22N4O3
5-[(3S)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— 5-ethyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H21N5
5-ethyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-(2-pyridin-4-ylsulfanylacetyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H19N3O3S
(5S)-9-(2-pyridin-4-ylsulfanylacetyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H25N3O3
(5S)-9-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5R)-9-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one —— C16H25N3O3
(5R)-9-[[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl]-1-oxa-9-azaspiro[4.6]undecan-8-one
—— (5S)-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H17N5O3
(5S)-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H22N4O4
(5S)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(2S)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C17H18N4O2
5-[(2S)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[2-[(2S)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C20H23N3O4
5-[2-[(2S)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (5R)-9-(2-pyridin-4-ylsulfanylacetyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C15H19N3O3S
(5R)-9-(2-pyridin-4-ylsulfanylacetyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(5-propylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H22N2O3S
(5R)-9-(5-propylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[2-[(2R)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione —— C20H23N3O4
5-[2-[(2R)-2-hydroxyspiro[1,2-dihydroindene-3,4'-piperidine]-1'-yl]-2-oxoethyl]-6-methyl-1H-pyrimidine-2,4-dione
—— (5R)-9-[3-(3-oxo-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23N3O5
(5R)-9-[3-(3-oxo-1,4-benzoxazin-4-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C14H22N4O4
(5R)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O
(5S)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(4-imidazol-1-ylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O2
(5R)-9-[(4-imidazol-1-ylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-tert-butyl-4-[[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl]furan-2-carboxamide —— C16H26N2O4
5-tert-butyl-4-[[(3R)-3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl]furan-2-carboxamide
—— (5S)-7-[(4-propan-2-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N2O
(5S)-7-[(4-propan-2-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[(4-imidazol-1-ylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O2
(5S)-9-[(4-imidazol-1-ylphenyl)methyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5R)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C23H28N4O4
(5R)-7-[(2,3-dimethoxyphenyl)methyl]-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O
(5R)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C17H18N4O2
5-[(2R)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— (5S)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C18H22N4O3
(5S)-9-[2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— 5-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one —— C17H22N4O3
5-[(3R)-3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl]-2-phenyl-1H-pyrazol-3-one
—— 5-phenyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H17N7
5-phenyl-N-[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5R)-9-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H25ClN2O3
(5R)-9-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H25ClN2O3
(5S)-9-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-(5-propylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C16H22N2O3S
(5S)-9-(5-propylthiophene-3-carbonyl)-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-7-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H17N3O4
(5S)-7-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H17N3O4
(5R)-7-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-phenyl-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine —— C17H17N7
5-phenyl-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
—— (5S)-9-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H23N3O4
(5S)-9-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5S)-9-(4-oxo-1H-quinoline-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H17N3O4
(5S)-9-(4-oxo-1H-quinoline-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-(4-oxo-1H-quinoline-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C17H17N3O4
(5R)-9-(4-oxo-1H-quinoline-2-carbonyl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-9-[3-(2-methylindol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H25N3O3
(5R)-9-[3-(2-methylindol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5R)-9-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C19H23N3O4
(5R)-9-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— (5R)-7-[(4-propan-2-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H26N2O
(5R)-7-[(4-propan-2-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[3-(2-methylindol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C20H25N3O3
(5S)-9-[3-(2-methylindol-1-yl)propanoyl]-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-2-(4-methylphenyl)sulfonyl-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H25N3O3S
(5S)-2-(4-methylphenyl)sulfonyl-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(4-methylphenyl)sulfonyl-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H25N3O3S
(5R)-2-(4-methylphenyl)sulfonyl-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23FN4O2
(5R)-9-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H23FN4O2
(5S)-9-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-9-[4-(dimethylamino)naphthalene-1-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C22H27N3O3
(5S)-9-[4-(dimethylamino)naphthalene-1-carbonyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one