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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[1-[[2-(Dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H26N8
5-[1-[[2-(Dimethylamino)pyrimidin-5-yl]methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-Tert-butyl-11-[(3-methylimidazol-4-yl)methyl]-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C18H24N6O
5-Tert-butyl-11-[(3-methylimidazol-4-yl)methyl]-2,6,7,11-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(phenoxymethyl)-N-[(Z)-(2,4,5-trimethylphenyl)methylideneamino]furan-2-carboxamide —— C22H22N2O3
5-(phenoxymethyl)-N-[(Z)-(2,4,5-trimethylphenyl)methylideneamino]furan-2-carboxamide
—— 5-(phenoxymethyl)-N-[(Z)-(4-propan-2-ylphenyl)methylideneamino]furan-2-carboxamide —— C22H22N2O3
5-(phenoxymethyl)-N-[(Z)-(4-propan-2-ylphenyl)methylideneamino]furan-2-carboxamide
—— 5-(phenoxymethyl)-N-[(Z)-pyridin-3-ylmethylideneamino]furan-2-carboxamide —— C18H15N3O3
5-(phenoxymethyl)-N-[(Z)-pyridin-3-ylmethylideneamino]furan-2-carboxamide
—— 5-[1-[(3-Ethoxy-4-prop-2-ynoxyphenyl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C24H29N5O2
5-[1-[(3-Ethoxy-4-prop-2-ynoxyphenyl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(phenoxymethyl)-N-[(Z)-(2,4,5-trimethoxyphenyl)methylideneamino]furan-2-carboxamide —— C22H22N2O6
5-(phenoxymethyl)-N-[(Z)-(2,4,5-trimethoxyphenyl)methylideneamino]furan-2-carboxamide
—— [5-[[4-(4,5-Dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]methyl]-2-methoxyphenyl]methanol —— C24H34N4O3
[5-[[4-(4,5-Dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]methyl]-2-methoxyphenyl]methanol
—— 5-cyclopropyl-3-[1-(furan-3-ylmethyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C17H20N6O2
5-cyclopropyl-3-[1-(furan-3-ylmethyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(3-methylthiophen-2-yl)-N-(3-morpholin-4-ylpropyl)pyrimidin-2-amine —— C20H25N5O2S
5-(3-methyl-1,2-oxazol-5-yl)-4-(3-methylthiophen-2-yl)-N-(3-morpholin-4-ylpropyl)pyrimidin-2-amine
—— 5-(phenoxymethyl)-N-[(Z)-1-phenylethylideneamino]furan-2-carboxamide —— C20H18N2O3
5-(phenoxymethyl)-N-[(Z)-1-phenylethylideneamino]furan-2-carboxamide
—— 5-[1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C23H28N6O
5-[1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-[1-[(1-Ethyl-3-methylpyrazol-4-yl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C19H27N7
5-[1-[(1-Ethyl-3-methylpyrazol-4-yl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(phenoxymethyl)-N-[(Z)-[2-(trifluoromethyl)phenyl]methylideneamino]furan-2-carboxamide —— C20H15F3N2O3
5-(phenoxymethyl)-N-[(Z)-[2-(trifluoromethyl)phenyl]methylideneamino]furan-2-carboxamide
—— 5-(phenoxymethyl)-N-[(Z)-[4-(trifluoromethyl)phenyl]methylideneamino]furan-2-carboxamide —— C20H15F3N2O3
5-(phenoxymethyl)-N-[(Z)-[4-(trifluoromethyl)phenyl]methylideneamino]furan-2-carboxamide
—— 5-(phenoxymethyl)-N-[(Z)-1-thiophen-2-ylethylideneamino]furan-2-carboxamide —— C18H16N2O3S
5-(phenoxymethyl)-N-[(Z)-1-thiophen-2-ylethylideneamino]furan-2-carboxamide
—— (5-cyclopropyl-2-methylpyrazol-3-yl)-[(1R,5S)-3-(2-fluoropyridin-3-yl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methanone —— C20H23FN4O2
(5-cyclopropyl-2-methylpyrazol-3-yl)-[(1R,5S)-3-(2-fluoropyridin-3-yl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methanone
—— 5-[[4-(4,5-dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]methyl]-N,N-dimethylpyrimidin-2-amine —— C22H33N7O
5-[[4-(4,5-dimethyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]methyl]-N,N-dimethylpyrimidin-2-amine
—— 5-cyclopropyl-3-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C20H26N8O
5-cyclopropyl-3-[1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-[1-[(4-Ethoxyphenyl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine —— C21H27N5O
5-[1-[(4-Ethoxyphenyl)methyl]piperidin-4-yl]-2-methylpyrazolo[1,5-a]pyrimidin-7-amine
—— 5-(phenoxymethyl)-N-[(Z)-1-pyridin-3-ylethylideneamino]furan-2-carboxamide —— C19H17N3O3
5-(phenoxymethyl)-N-[(Z)-1-pyridin-3-ylethylideneamino]furan-2-carboxamide
—— (5R)-3-methyl-5-[2-[4-(4-methyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C20H27N5O4S
(5R)-3-methyl-5-[2-[4-(4-methyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— 5-(phenoxymethyl)-N-[(Z)-1-pyridin-4-ylethylideneamino]furan-2-carboxamide —— C19H17N3O3
5-(phenoxymethyl)-N-[(Z)-1-pyridin-4-ylethylideneamino]furan-2-carboxamide
—— 5-(phenoxymethyl)-N-[(Z)-pyridin-4-ylmethylideneamino]furan-2-carboxamide —— C18H15N3O3
5-(phenoxymethyl)-N-[(Z)-pyridin-4-ylmethylideneamino]furan-2-carboxamide
—— 5-(1,5-dimethylpyrazol-4-yl)-2-methyl-1,1-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,2,6-thiadiazine-3-carboxamide —— C17H16F3N5O4S
5-(1,5-dimethylpyrazol-4-yl)-2-methyl-1,1-dioxo-N-[4-(trifluoromethoxy)phenyl]-1,2,6-thiadiazine-3-carboxamide
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-morpholin-4-yl-2-oxoethyl)-6-thiophen-2-ylpyridazin-3-one —— C18H18N4O4S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-morpholin-4-yl-2-oxoethyl)-6-thiophen-2-ylpyridazin-3-one
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-piperidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one —— C19H22N4O2S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-piperidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one
—— (5S)-3-methyl-5-[2-[4-(4-methyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione —— C20H27N5O4S
(5S)-3-methyl-5-[2-[4-(4-methyl-6-morpholin-4-ylpyrimidin-2-yl)piperidin-1-yl]-2-oxoethyl]-1,3-thiazolidine-2,4-dione
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine —— C23H23N7O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
—— 5-(3-methyl-1,2-oxazol-5-yl)-2-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-6-thiophen-2-ylpyridazin-3-one —— C20H22N4O3S
5-(3-methyl-1,2-oxazol-5-yl)-2-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-6-thiophen-2-ylpyridazin-3-one
—— [5-(1-methylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C20H19N7O2
[5-(1-methylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 5-(1,3-dimethylpyrazol-4-yl)-2-methyl-N-(5-methyl-1,2-oxazol-3-yl)-1,1-dioxo-1,2,6-thiadiazine-3-carboxamide —— C14H16N6O4S
5-(1,3-dimethylpyrazol-4-yl)-2-methyl-N-(5-methyl-1,2-oxazol-3-yl)-1,1-dioxo-1,2,6-thiadiazine-3-carboxamide
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one —— C18H18N4O3S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-oxo-2-pyrrolidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one
—— 5-(phenoxymethyl)-N-[(Z)-[(E)-3-phenylprop-2-enylidene]amino]furan-2-carboxamide —— C21H18N2O3
5-(phenoxymethyl)-N-[(Z)-[(E)-3-phenylprop-2-enylidene]amino]furan-2-carboxamide
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-[(2-methylphenyl)methyl]-6-thiophen-2-ylpyridazin-3-one —— C20H17N3O2S
5-(3-Methyl-1,2-oxazol-5-yl)-2-[(2-methylphenyl)methyl]-6-thiophen-2-ylpyridazin-3-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-2-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-6-thiophen-2-ylpyridazin-3-one —— C20H22N4O3S
5-(3-methyl-1,2-oxazol-5-yl)-2-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-6-thiophen-2-ylpyridazin-3-one
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(3-oxo-3-phenylpropyl)-6-thiophen-2-ylpyridazin-3-one —— C21H17N3O3S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(3-oxo-3-phenylpropyl)-6-thiophen-2-ylpyridazin-3-one
—— 5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-[(1S)-1-phenylethyl]pyrimidin-2-amine —— C25H26N6O2
5-(3-methyl-1,2-oxazol-5-yl)-4-(6-morpholin-4-ylpyridin-3-yl)-N-[(1S)-1-phenylethyl]pyrimidin-2-amine
—— 5-[4-[(Z)-C-methyl-N-[[2-(2-oxoazepan-1-yl)acetyl]amino]carbonimidoyl]phenyl]furan-2-carboxylic acid —— C21H23N3O5
5-[4-[(Z)-C-methyl-N-[[2-(2-oxoazepan-1-yl)acetyl]amino]carbonimidoyl]phenyl]furan-2-carboxylic acid
—— [5-methyl-4-(morpholin-4-ylmethyl)furan-2-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C23H27N5O3
[5-methyl-4-(morpholin-4-ylmethyl)furan-2-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 5,6-dimethyl-2-(2-methylfuran-3-yl)-N-(3-morpholin-4-ylpropyl)pyrazolo[1,5-a]pyrimidin-7-amine —— C20H27N5O2
5,6-dimethyl-2-(2-methylfuran-3-yl)-N-(3-morpholin-4-ylpropyl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 5-cyclopropyl-3-[1-[2-(2,5-dimethoxyphenyl)acetyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C22H26N6O4
5-cyclopropyl-3-[1-[2-(2,5-dimethoxyphenyl)acetyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— [5-(1-methylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C20H19N7O2
[5-(1-methylpyrazol-4-yl)-1,2-oxazol-3-yl]-[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-oxo-2-piperidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one —— C19H20N4O3S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(2-oxo-2-piperidin-1-ylethyl)-6-thiophen-2-ylpyridazin-3-one
—— 5-(3-Methyl-1,2-oxazol-5-yl)-2-(pyridin-3-ylmethyl)-6-thiophen-2-ylpyridazin-3-one —— C18H14N4O2S
5-(3-Methyl-1,2-oxazol-5-yl)-2-(pyridin-3-ylmethyl)-6-thiophen-2-ylpyridazin-3-one
—— 5-cyclopropyl-3-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C19H18F2N6O2
5-cyclopropyl-3-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-cyclopropyl-3-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C19H18F2N6O2
5-cyclopropyl-3-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-methoxy-2-[[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]phenol —— C20H22N4O2
5-methoxy-2-[[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]phenol
—— [5-methyl-4-(morpholin-4-ylmethyl)furan-2-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone —— C23H27N5O3
[5-methyl-4-(morpholin-4-ylmethyl)furan-2-yl]-[(1S,12R)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methanone
—— 5,6-dimethyl-2-(oxan-4-yl)-N-(2-pyridin-4-ylethyl)pyrazolo[1,5-a]pyrimidin-7-amine —— C20H25N5O
5,6-dimethyl-2-(oxan-4-yl)-N-(2-pyridin-4-ylethyl)pyrazolo[1,5-a]pyrimidin-7-amine